Target Details
| UniProt AC | P51617 |
|---|---|
| Gene Symbol | IRAK1 |
| Protein Name | Interleukin-1 receptor-associated kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00531 (Death) PF00069 (Pkinase) |
Summary
- Multi-target molecules 312
- Clinical molecules 15
- Avg pChEMBL 6.84
KEGG Pathways (20)
- Alcoholic liver disease
- Chagas disease
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- Neurotrophin signaling pathway
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Yersinia infection
Active Molecules (312)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MURKOANUFGPGGP
|
7.2 | IC50 | 2 | — | |
JOGIYNFTOOGHNQ
|
7.1 | IC50 | 3 | — | |
MHRNVFQJUUXQIG
|
7.1 | IC50 | 2 | — | |
SWPXADMCNLNAGW
|
7.1 | IC50 | 10 | — | |
UUTHPYJPFVUVPN
|
7.1 | Ki | 3 | — | |
DKXHSOUZPMHNIZ
|
7.1 | Ki | 51 | Yes | |
FUMCKNCUEAQHCV
|
7.1 | Ki | 103 | — | |
GCBJDOWIQHMCMR
|
7.1 | Ki | 84 | — | |
JOBAEWAZUAPIKW
|
7.1 | IC50 | 2 | — | |
MHRNVFQJUUXQIG
|
7.1 | IC50 | 2 | — | |
WAOZMJFYNREQLU
|
7.1 | IC50 | 2 | — | |
YMIJUBCSOKSFRU
|
7.1 | Ki | 87 | — | |
HXJNPTQRPZSTHS
|
7.1 | IC50 | 2 | — | |
QITLDLOFVQLFFF
|
7.1 | IC50 | 2 | — | |
OWSBCGNMLGHERL
|
7.1 | IC50 | 2 | — | |
HXUCFPZSRWJRRN
|
7.0 | IC50 | 3 | — | |
CFBKGVOKLIQQJD
|
7.0 | IC50 | 3 | — | |
YMEYAMDEQBMREG
|
7.0 | IC50 | 3 | — | |
FXKMVTAKVQDJJT
|
7.0 | Ki | 2 | — | |
AKLWVZFHNFDHCQ
|
7.0 | IC50 | 3 | — | |
MEBULVBTXSYJKD
|
7.0 | IC50 | 3 | — | |
RKUKAACYUCUJEE
|
7.0 | Ki | 58 | — | |
SRCLLEDPPXOXGH
|
7.0 | IC50 | 3 | — | |
XMWONVHOMANOOY
|
7.0 | IC50 | 3 | — | |
LVDGPLKQEUXHAV
|
7.0 | IC50 | 2 | — | |
CVWXJKQAOSCOAB
|
6.9 | IC50 | 35 | — | |
KPKVXBUKMZIGPN
|
6.9 | IC50 | 3 | — | |
KSJNXKBKMYLRSO
|
6.9 | IC50 | 3 | — | |
XZXHXSATPCNXJR
|
6.9 | Kd | 165 | Yes | |
HHVUHFYJIYORJI
|
6.9 | IC50 | 3 | — | |
MURKOANUFGPGGP
|
6.9 | IC50 | 2 | — | |
ADMFLILDQJSEIK
|
6.9 | Ki | 72 | — | |
MUYFQIQEBJQOGI
|
6.9 | IC50 | 2 | — | |
QONPPIZSNSSCSK
|
6.9 | Ki | 45 | Yes | |
SYLTYCLPHHSEIJ
|
6.9 | Ki | 27 | — | |
TVLFEDKEAOXRCZ
|
6.9 | Ki | 22 | — | |
UZWDCWONPYILKI
|
6.9 | Kd | 47 | — | |
WINHZLLDWRZWRT
|
6.9 | Ki | 66 | — | |
ODPGGGTTYSGTGO
|
6.9 | Kd | 153 | — | |
UZBFFCBUJQNOPY
|
6.9 | IC50 | 3 | — | |
UBKAKYFRDGQVJG
|
6.8 | IC50 | 3 | — | |
ZEMQCNHEKKILBX
|
6.8 | IC50 | 3 | — | |
DUOPMZXNVCHSKJ
|
6.8 | IC50 | 3 | — | |
XGALLCVXEZPNRQ
|
6.8 | Kd | 39 | Yes | |
SZFYZDIPRMLBDC
|
6.8 | Kd | 9 | — | |
FTEUGWHCWRSIJU
|
6.8 | IC50 | 3 | — | |
HXYSWTZEQZNVDR
|
6.8 | IC50 | 3 | — | |
CLRFYTGANQZOBS
|
6.8 | Ki | 41 | — | |
MIKAKZKNMYZLDX
|
6.8 | Ki | 42 | — | |
NLUPJKQOKWBWFC
|
6.8 | Ki | 69 | — |