Target Details
| UniProt AC | P51617 |
|---|---|
| Gene Symbol | IRAK1 |
| Protein Name | Interleukin-1 receptor-associated kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00531 (Death) PF00069 (Pkinase) |
Summary
- Multi-target molecules 312
- Clinical molecules 15
- Avg pChEMBL 6.84
KEGG Pathways (20)
- Alcoholic liver disease
- Chagas disease
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- Neurotrophin signaling pathway
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Yersinia infection
Active Molecules (312)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DJVYXMINSBMUHH
|
7.6 | IC50 | 8 | — | |
RPGMSHCJIWHISY
|
7.6 | IC50 | 3 | — | |
RPGMSHCJIWHISY
|
7.6 | IC50 | 3 | — | |
MCOWNEICYXDEPL
|
7.5 | IC50 | 3 | — | |
MMKIEBBLOVSLAS
|
7.5 | IC50 | 3 | — | |
CMKUJKFQBWYWBJ
|
7.5 | IC50 | 3 | — | |
MWKSRKSEWLRPBL
|
7.5 | Kd | 1075 | — | |
RZHTUCWWEKMCNM
|
7.5 | IC50 | 2 | — | |
HXQKDULUOFXHDI
|
7.5 | IC50 | 2 | — | |
UDFDIIVNIYWXDM
|
7.5 | Ki | 74 | — | |
YEHCNYAQEBQCCS
|
7.5 | Ki | 74 | — | |
ZQKNIPQNEVNCDY
|
7.5 | IC50 | 8 | — | |
YUANXHKOYHEHOW
|
7.5 | IC50 | 2 | — | |
CZYCPCNQYXFAPQ
|
7.5 | IC50 | 2 | — | |
FQBRQRVXPUQKLG
|
7.5 | IC50 | 10 | — | |
GPQARSZTOBDAFR
|
7.5 | IC50 | 2 | — | |
PKAXKMPZRBQIOO
|
7.5 | IC50 | 3 | — | |
RDBXDKAXTSZQAP
|
7.4 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
7.4 | IC50 | 92 | — | |
HKSZLNNOFSGOKW
|
7.4 | IC50 | 408 | — | |
HWXVIOGONBBTBY
|
7.4 | IC50 | 27 | — | |
VVQWKIHKNXGJKG
|
7.4 | IC50 | 2 | — | |
XPHWIERLJBFPFV
|
7.4 | Ki | 69 | — | |
FQGLEOSEPJEJPE
|
7.4 | IC50 | 2 | — | |
NTKWIHLGLPIAOG
|
7.4 | IC50 | 2 | — | |
FLXHMSFCIMZSJT
|
7.4 | IC50 | 3 | — | |
VDJSCKUWUKCUEK
|
7.4 | IC50 | 2 | — | |
YCFRZMCRPHNZOC
|
7.4 | IC50 | 7 | — | |
YCFRZMCRPHNZOC
|
7.4 | IC50 | 6 | — | |
QQWUGDVOUVUTOY
|
7.3 | Kd | 231 | Yes | |
QPKFIZDVDMZSPR
|
7.3 | Ki | 3 | — | |
YYLKKYCXAOBSRM
|
7.3 | Kd | 191 | — | |
KTEIFNKAUNYNJU
|
7.3 | Kd | 114 | — | |
CLEGDJQQHUTCOW
|
7.3 | Ki | 43 | — | |
SUULIUKTZNKMMB
|
7.3 | Ki | 10 | — | |
XFWUTMHVDGPWLH
|
7.3 | Ki | 75 | — | |
SNNSTEZDXSIKQW
|
7.3 | IC50 | 3 | — | |
RKSPQOPBECGSGM
|
7.3 | IC50 | 3 | — | |
BNVZRFQNZWYPQH
|
7.3 | IC50 | 2 | — | |
YZPJEKZOTFSOHR
|
7.2 | IC50 | 2 | — | |
PWCLOPMRUGHLET
|
7.2 | IC50 | 2 | — | |
AZIKDQBYCZVPSU
|
7.2 | IC50 | 3 | — | |
KZVISSXNPKKESH
|
7.2 | IC50 | 3 | — | |
VRHHAMWTRSVIEX
|
7.2 | Kd | 5 | — | |
JZTOUVBEZONDKA
|
7.2 | Ki | 80 | — | |
RYYNGWLOYLRZLK
|
7.2 | Ki | 104 | — | |
STCDSEJQOLKGFJ
|
7.2 | IC50 | 2 | — | |
FPQNRXITKTZFMF
|
7.2 | Kd | 13 | — | |
FUOKGTYXSNVQIW
|
7.2 | IC50 | 3 | — | |
MINWMNHFXQZNMG
|
7.2 | IC50 | 2 | — |