Target Details
| UniProt AC | P51617 |
|---|---|
| Gene Symbol | IRAK1 |
| Protein Name | Interleukin-1 receptor-associated kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00531 (Death) PF00069 (Pkinase) |
Summary
- Multi-target molecules 312
- Clinical molecules 15
- Avg pChEMBL 6.84
KEGG Pathways (20)
- Alcoholic liver disease
- Chagas disease
- Coronavirus disease - COVID-19
- Epstein-Barr virus infection
- Hepatitis B
- Herpes simplex virus 1 infection
- Human immunodeficiency virus 1 infection
- Leishmaniasis
- Lipid and atherosclerosis
- MAPK signaling pathway
- Measles
- NF-kappa B signaling pathway
- Neurotrophin signaling pathway
- Pathogenic Escherichia coli infection
- Pertussis
- Salmonella infection
- Toll-like receptor signaling pathway
- Toxoplasmosis
- Tuberculosis
- Yersinia infection
Active Molecules (312)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KQDKXYWFBHTGIX
|
8.9 | IC50 | 2 | — | |
QQIQOMIKWUAMAA
|
8.7 | IC50 | 7 | — | |
WMZGRDMNDXPHMF
|
8.3 | IC50 | 2 | — | |
ZMZGUJSLGMATGF
|
8.3 | IC50 | 5 | — | |
GZYCQQBRSRIFII
|
8.2 | Kd | 7 | — | |
WSTUJEXAPHIEIM
|
8.2 | Kd | 10 | — | |
VMZCRJAQNNOYPK
|
8.2 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
8.2 | Kd | 289 | Yes | |
KLAHVJUJQYVKPO
|
8.2 | IC50 | 2 | — | |
WBVTVMHUUOONFL
|
8.2 | IC50 | 2 | — | |
FUFJXODRNRQIRI
|
8.1 | IC50 | 2 | — | |
HCHLTTBJHNWMPS
|
8.1 | IC50 | 2 | — | |
XBMMPGPTZWUPAP
|
8.1 | IC50 | 2 | — | |
LYADGAGFYYXXIO
|
8.1 | IC50 | 82 | — | |
WQVPGYMGERDXLH
|
8.1 | IC50 | 2 | — | |
NHHQJBCNYHBUSI
|
8.0 | Kd | 220 | — | |
OTAZAWFIQUEVLG
|
8.0 | IC50 | 3 | — | |
DQEKCEBMQCYICP
|
7.9 | Ki | 3 | — | |
GHMRUNOHAHJNNA
|
7.9 | Ki | 29 | — | |
IAQIZJLJAOFQPG
|
7.9 | IC50 | 2 | — | |
PNKALLUVKOKYHZ
|
7.9 | Ki | 32 | — | |
ATVTUVKVZSYFBE
|
7.9 | Kd | 7 | — | |
IDGNCVHQDDOPND
|
7.8 | IC50 | 6 | — | |
RADRIIWGHYFWPP
|
7.8 | IC50 | 4 | — | |
RAFFLDOJXQAJPF
|
7.8 | IC50 | 2 | — | |
WINHZLLDWRZWRT
|
7.8 | Kd | 201 | Yes | |
YLJPQGVBJWZONC
|
7.8 | IC50 | 6 | — | |
IWAWFGKTGNXQLY
|
7.8 | IC50 | 2 | — | |
QYGMZFLXMWJYRJ
|
7.8 | Ki | 14 | — | |
DGUFRRJUHIZTQE
|
7.7 | Ki | 3 | — | |
FRKBJIBHJMIOHI
|
7.7 | IC50 | 2 | — | |
JGNYWVKGPUWQDG
|
7.7 | IC50 | 2 | — | |
UEFCSGDOOJJXTN
|
7.7 | IC50 | 46 | — | |
GCYXEGSPUDSZJY
|
7.7 | Ki | 82 | — | |
VBIYDORVDCFKHM
|
7.7 | Ki | 13 | — | |
UXNHXSBDEPPEKO
|
7.7 | IC50 | 2 | — | |
GZNUMHPRTTZGTC
|
7.7 | IC50 | 3 | — | |
IQBCZHKBLZWXEM
|
7.7 | IC50 | 3 | — | |
VBVMZSHPPUKQDJ
|
7.7 | IC50 | 2 | — | |
HTJGFHHVVPNDMR
|
7.7 | IC50 | 6 | — | |
IALDYVNFZAPNJV
|
7.7 | IC50 | 11 | — | |
YISMQBFJYDFMAL
|
7.7 | IC50 | 46 | — | |
IGZHZHVJEZFVIH
|
7.6 | IC50 | 2 | — | |
OSATXCGVOWUMIG
|
7.6 | Ki | 2 | — | |
MVJMMLFMPWITEJ
|
7.6 | Ki | 110 | — | |
QSSMDRNGJZDMSQ
|
7.6 | IC50 | 3 | — | |
YGDAYHUWESEYBV
|
7.6 | IC50 | 2 | — | |
DJVYXMINSBMUHH
|
7.6 | IC50 | 8 | — | |
OCDYJTRAVKONSS
|
7.6 | IC50 | 3 | — | |
CTNPALGJUAXMMC
|
7.6 | Kd | 151 | — |