Target Details
| UniProt AC | P51531 |
|---|---|
| Gene Symbol | SMARCA2 |
| Protein Name | SWI/SNF-related matrix-associated actin-dependent regulator of chromatin subfamily A member 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07533 (BRK) PF00439 (Bromodomain) PF00271 (Helicase_C) PF07529 (HSA) PF08880 (QLQ) PF14619 (SnAC) PF00176 (SNF2-rel_dom) |
Summary
- Multi-target molecules 66
- Clinical molecules 0
- Avg pChEMBL 7.37
KEGG Pathways (3)
Associated Diseases (2)
Active Molecules (66)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IHWHEWSGCAIVIM
|
7.0 | IC50 | 2 | — | |
LAMLMRYWDMUTPN
|
7.0 | IC50 | 3 | — | |
QQVCUSPUMMUFTD
|
7.0 | Kd | 3 | — | |
SZKHGLTYXIDOFH
|
6.9 | Kd | 3 | — | |
ICVVDNFTMKQVQK
|
6.7 | IC50 | 3 | — | |
HFIPFTAKXMECCX
|
6.7 | Kd | 2 | — | |
QBSVEUFIPREFRZ
|
6.7 | IC50 | 2 | — | |
VLPRXFLUVHYBBT
|
6.6 | Kd | 3 | — | |
SIWZRTOJDAJYHG
|
6.6 | IC50 | 3 | — | |
YIQNHNMFVVDQQU
|
6.5 | IC50 | 3 | — | |
DHDZFJQQXROKLC
|
6.5 | Kd | 3 | — | |
LTOWBWFTKOUSOO
|
6.3 | IC50 | 3 | — | |
HCMYOXQNMXWNNB
|
6.3 | IC50 | 2 | — | |
IVARZBJJMMUJHI
|
6.1 | IC50 | 2 | — | |
APFPJIWYBJHIHN
|
6.0 | IC50 | 2 | — | |
GZFJPALDEYOFHA
|
6.0 | IC50 | 6 | — |