Target Details
| UniProt AC | P51452 |
|---|---|
| Gene Symbol | DUSP3 |
| Protein Name | Dual specificity protein phosphatase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00782 (DSPc) |
Summary
- Multi-target molecules 38
- Clinical molecules 1
- Avg pChEMBL 6.29
KEGG Pathways (1)
Active Molecules (38)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LCOYYIYBAKWSIQ
|
7.1 | IC50 | 3 | — | |
VCMZPVCCQDEZRB
|
6.7 | IC50 | 2 | — | |
HBNOSXCFGXWLCL
|
6.7 | IC50 | 2 | — | |
HNDWHMKTONQBSA
|
6.6 | IC50 | 3 | — | |
NMLOLMOZTQCQJF
|
6.5 | IC50 | 2 | — | |
GGZKBXVGDIISFQ
|
6.5 | IC50 | 2 | — | |
QIRQGNZQWCVFAG
|
6.5 | IC50 | 2 | — | |
AQNQKVLAOFOLOO
|
6.5 | IC50 | 2 | — | |
OJWCRZGASOCMRF
|
6.5 | IC50 | 2 | — | |
PBERWSCWYDTVLM
|
6.5 | IC50 | 2 | — | |
KGOAMMKJVQZGLF
|
6.5 | IC50 | 2 | — | |
WWPIFOBKKAFENH
|
6.4 | IC50 | 2 | — | |
WRFNFMUNJVHPGT
|
6.4 | IC50 | 3 | — | |
VZRHEZSOEBDPOH
|
6.4 | IC50 | 2 | — | |
WBNVGVTYQBOUQG
|
6.3 | IC50 | 2 | — | |
KKWJOTGFSWWYJO
|
6.3 | IC50 | 3 | — | |
QEAYLNJEDDOYNQ
|
6.3 | IC50 | 2 | — | |
BFJXGNDCJKJBPA
|
6.3 | IC50 | 2 | — | |
GROJNADPOMHDCI
|
6.3 | IC50 | 2 | — | |
FKZHXROWVQMDAU
|
6.2 | IC50 | 2 | — | |
JFRYLPFKWKOMBZ
|
6.2 | IC50 | 2 | — | |
VDHAPQOXKYQZDW
|
6.2 | IC50 | 2 | — | |
CLLDGZJVIZEVBU
|
6.1 | IC50 | 2 | — | |
LWULRPYIMPIYQD
|
6.1 | IC50 | 2 | — | |
RZODWLFHOZGYSH
|
6.1 | IC50 | 2 | — | |
YJOYTQQCKRNIPB
|
6.1 | IC50 | 2 | — | |
CCGJOMGWGAAKFE
|
6.1 | IC50 | 2 | — | |
KJRKWHJEHFSIPH
|
6.1 | IC50 | 2 | — | |
GXEHDKDVKTUCMK
|
6.1 | IC50 | 2 | — | |
WVNQJOXFTBTXOE
|
6.1 | IC50 | 6 | — | |
YSWVIGJDOZEAPY
|
6.1 | IC50 | 2 | — | |
AVMJNCJSYBFURN
|
6.1 | IC50 | 4 | Yes | |
VDWPBBYWLISYQY
|
6.1 | IC50 | 2 | — | |
IOSUGCLQHJKTCK
|
6.0 | IC50 | 2 | — | |
LKBYYUZEKINDPS
|
6.0 | IC50 | 6 | — | |
NWGYQTVHIXHPJH
|
6.0 | IC50 | 2 | — | |
RUQGCDMXFBOTMW
|
6.0 | IC50 | 2 | — | |
SLGRAIAQIAUZAQ
|
6.0 | IC50 | 16 | — |