Target Details
| UniProt AC | P51451 |
|---|---|
| Gene Symbol | BLK |
| Protein Name | Tyrosine-protein kinase Blk |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 388
- Clinical molecules 48
- Avg pChEMBL 7.08
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (388)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QDOBTYVGPGFRCM
|
6.2 | Ki | 11 | — | |
QYZOGCMHVIGURT
|
6.2 | Ki | 26 | Yes | |
RIUZPIBUSOHUKF
|
6.2 | Ki | 23 | — | |
UPPYTUNUGKDPSA
|
6.2 | Ki | 7 | — | |
VNGYQBMDQMDALH
|
6.2 | Ki | 25 | — | |
ZAARMHXLYCHRAK
|
6.2 | Ki | 20 | — | |
JOOXLOJCABQBSG
|
6.2 | Kd | 139 | — | |
MVCOAUNKQVWQHZ
|
6.2 | Kd | 54 | Yes | |
PFTXFNSHFZLJNT
|
6.1 | IC50 | 17 | — | |
CTNPALGJUAXMMC
|
6.1 | Kd | 151 | — | |
GEGCXGMFUYJULA
|
6.1 | Ki | 30 | Yes | |
HBHOKIDZSIYNGE
|
6.1 | Ki | 3 | — | |
HCNIBOQWDVOZKF
|
6.1 | Ki | 26 | — | |
IJRBJCMLWLFMIN
|
6.1 | Ki | 17 | — | |
KTEIFNKAUNYNJU
|
6.1 | Ki | 48 | — | |
MLDQJTXFUGDVEO
|
6.1 | Ki | 85 | Yes | |
OPHDFABOUWVUBL
|
6.1 | IC50 | 4 | — | |
PNKALLUVKOKYHZ
|
6.1 | Ki | 32 | — | |
PYXQMJSGJIJHJT
|
6.1 | Ki | 28 | — | |
QEWSTOOMTBAUAG
|
6.1 | Ki | 17 | — | |
RWEHAHIEUDLKGT
|
6.1 | Ki | 33 | — | |
UWDBNTXEKYRMSG
|
6.1 | Ki | 26 | — | |
WCAKSXQRFBVWDG
|
6.1 | Ki | 10 | — | |
BMYBPXJXNNXUJF
|
6.1 | IC50 | 4 | — | |
DYIBUWLFYBFBBS
|
6.1 | IC50 | 5 | — | |
XISIJMIPHPQCQQ
|
6.0 | IC50 | 9 | — | |
DZIPQNPWTUXXSJ
|
6.0 | Ki | 18 | — | |
FTIAKTLRFKSDFR
|
6.0 | Ki | 10 | Yes | |
GHMRUNOHAHJNNA
|
6.0 | Ki | 29 | — | |
GKHIVNAUVKXIIY
|
6.0 | Ki | 4 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KAKFXRYHYUPXSU
|
6.0 | Ki | 16 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KOHNRDPXFDZZJF
|
6.0 | Ki | 31 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
QMMMGQKKOKYDMN
|
6.0 | Ki | 5 | — | |
VCSQVKQFGYRGEH
|
6.0 | Ki | 13 | — | |
XGALLCVXEZPNRQ
|
6.0 | Ki | 39 | Yes |