Target Details
| UniProt AC | P51451 |
|---|---|
| Gene Symbol | BLK |
| Protein Name | Tyrosine-protein kinase Blk |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 388
- Clinical molecules 48
- Avg pChEMBL 7.08
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (388)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GCBJDOWIQHMCMR
|
6.4 | Ki | 84 | — | |
GKFFFOLFBJUEFN
|
6.4 | Ki | 3 | — | |
GMYYMEOGFRKSFS
|
6.4 | Ki | 29 | — | |
HRZOUBQYVUXBNS
|
6.4 | Ki | 38 | — | |
KIOLXAWQJUDVMS
|
6.4 | Ki | 5 | — | |
KROLCVQARUUHNV
|
6.4 | Ki | 12 | — | |
MASJMHFQMYAPJR
|
6.4 | Ki | 41 | — | |
MZDKLVOWGIOKTN
|
6.4 | Ki | 80 | — | |
NXNQLECPAXXYTR
|
6.4 | Ki | 29 | — | |
RTDSHUGNRVXRHN
|
6.4 | Ki | 51 | — | |
YDWMUCKJUNLURC
|
6.4 | Ki | 24 | — | |
ZHTVWJDQZBBZHV
|
6.4 | Ki | 9 | — | |
ZLVOTRRGLSDLPF
|
6.4 | Ki | 36 | — | |
ITTRLTNMFYIYPA
|
6.4 | IC50 | 17 | — | |
DYOUYPOJLPRXSV
|
6.3 | IC50 | 2 | — | |
YJAJTLZIWHYGPF
|
6.3 | IC50 | 3 | — | |
SBRIQINKAOKMMM
|
6.3 | IC50 | 6 | — | |
BMGQWWVMWDBQGC
|
6.3 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.3 | Kd | 91 | Yes | |
HHZIURLSWUIHRB
|
6.3 | Kd | 57 | Yes | |
IOBVCHJTLVPPBR
|
6.3 | Ki | 39 | — | |
OQNPAZRZCXFOBC
|
6.3 | Ki | 11 | — | |
PSCJSWRVCKUMSL
|
6.3 | Ki | 35 | — | |
RITAVMQDGBJQJZ
|
6.3 | Ki | 33 | — | |
RJZDECGDCKOHBV
|
6.3 | Ki | 70 | — | |
RMTJSBZCZKCYHB
|
6.3 | IC50 | 13 | — | |
TVLFEDKEAOXRCZ
|
6.3 | Ki | 22 | — | |
XYZNKCSDQRKAFR
|
6.3 | Ki | 53 | — | |
YEPNVBNYCRGZRX
|
6.3 | Ki | 26 | — | |
YMIJUBCSOKSFRU
|
6.3 | Ki | 87 | — | |
ZQQVWTACALNOAJ
|
6.3 | Ki | 11 | — | |
GLBZSOQDAOLMGC
|
6.3 | IC50 | 23 | Yes | |
KTUFNOKKBVMGRW
|
6.3 | Kd | 38 | Yes | |
YZNIHXUBUWEUCM
|
6.3 | IC50 | 14 | — | |
CLUYEBBJSXKZNL
|
6.3 | IC50 | 2 | — | |
DPZGKYJHTOSMIA
|
6.3 | IC50 | 8 | — | |
HXBVFFZAZCNTBQ
|
6.3 | IC50 | 2 | — | |
KUCNBQPAJZRQMJ
|
6.3 | IC50 | 11 | — | |
KZRDVFBPXXGSPD
|
6.3 | IC50 | 9 | — | |
MJQGHLODJHABRA
|
6.3 | IC50 | 10 | — | |
NNJUAJKDRBFVRD
|
6.3 | IC50 | 2 | — | |
QUFURWJAQILIFO
|
6.3 | IC50 | 9 | — | |
JIBBGYSUSKAPDY
|
6.2 | IC50 | 19 | — | |
PIDFACDPHSZEFT
|
6.2 | IC50 | 4 | — | |
CEJHRMYKGWBHHX
|
6.2 | IC50 | 3 | — | |
ZZSBPGIGIUFJRA
|
6.2 | Kd | 46 | — | |
DJOJKIGNNDWGRS
|
6.2 | Ki | 13 | — | |
FJZXDUKUMALHNP
|
6.2 | Ki | 10 | — | |
FONINLXADYUZFI
|
6.2 | Ki | 25 | — | |
LYNBNVBMAGDJRW
|
6.2 | Ki | 81 | — |