Target Details
| UniProt AC | P51451 |
|---|---|
| Gene Symbol | BLK |
| Protein Name | Tyrosine-protein kinase Blk |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 388
- Clinical molecules 48
- Avg pChEMBL 7.08
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (388)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LSFLAQVDISHMNB
|
6.7 | Ki | 13 | — | |
NSKFXNDKPCVDIN
|
6.7 | Ki | 12 | — | |
QONPPIZSNSSCSK
|
6.7 | Ki | 45 | Yes | |
SJMFZIGFOIPNPE
|
6.7 | Ki | 10 | — | |
UORAPQCBWYIISR
|
6.7 | IC50 | 15 | — | |
ULXXDDBFHOBEHA
|
6.7 | Kd | 15 | Yes | |
UKYJKXMPIDEQFF
|
6.6 | IC50 | 16 | — | |
MFAQYJIYDMLAIM
|
6.6 | Kd | 130 | Yes | |
ILXFYIOJPFUYGX
|
6.6 | IC50 | 5 | — | |
DJLORVJVWIBDME
|
6.6 | Ki | 24 | — | |
FGSVLADZCDNNOC
|
6.6 | Ki | 11 | — | |
GDYZFFBMSBDTAA
|
6.6 | Ki | 60 | — | |
GQGMUKOYILWOIQ
|
6.6 | Ki | 25 | — | |
GXFGHUNNGNQSMQ
|
6.6 | Ki | 19 | — | |
NRSGWEVTVGZDFC
|
6.6 | Ki | 50 | — | |
QKPLUKMJEKRAJD
|
6.6 | Ki | 30 | Yes | |
RKLGMDOZEOTQEM
|
6.6 | Ki | 12 | — | |
SXXRMKLCTXMFPH
|
6.6 | IC50 | 5 | — | |
UTQPKPHUIMHAAN
|
6.6 | Ki | 22 | — | |
WHKWRDQKKUPBMN
|
6.6 | Ki | 7 | — | |
YACXOXQTGJXYNX
|
6.6 | Ki | 11 | — | |
WDTHDWKPTWWHLS
|
6.5 | IC50 | 13 | — | |
ZHLODYGHLUYMDJ
|
6.5 | IC50 | 7 | — | |
COWVAFPFSREMEQ
|
6.5 | IC50 | 5 | — | |
YTIWDAUDJMCXOD
|
6.5 | IC50 | 5 | — | |
GXANJKDFGYJBEM
|
6.5 | IC50 | 5 | — | |
WMMNTQFZCHUZSM
|
6.5 | IC50 | 14 | — | |
FOONBYIHFUMRSX
|
6.5 | Ki | 12 | — | |
HXHAJRMTJXHJJZ
|
6.5 | Ki | 52 | Yes | |
KTQYQHLIMZOBSM
|
6.5 | Ki | 12 | — | |
KWSZYBNXNYRQCC
|
6.5 | Ki | 21 | — | |
MIKAKZKNMYZLDX
|
6.5 | Ki | 42 | — | |
MPVGZUGXCQEXTM
|
6.5 | Ki | 61 | Yes | |
PKCDDUHJAFVJJB
|
6.5 | Ki | 13 | — | |
QPORZABOFXPRHM
|
6.5 | Ki | 18 | — | |
RGZXAQQHXALOBL
|
6.5 | Kd | 10 | — | |
RPGBQFNDFPEOON
|
6.5 | Ki | 22 | — | |
UPITUWGOTMBQLX
|
6.5 | Ki | 13 | — | |
XKZQZMSAWVDRSP
|
6.5 | IC50 | 39 | Yes | |
ZXLFIHLBHMLHFJ
|
6.5 | Ki | 31 | — | |
FJNULDLUBJRUJN
|
6.5 | IC50 | 5 | — | |
JGLBGBDMKMGQFA
|
6.5 | IC50 | 5 | — | |
VUDJPBPVCUEFHU
|
6.5 | IC50 | 5 | — | |
RTRNJQOBEOISFQ
|
6.4 | IC50 | 5 | — | |
FDVSOQRNTAPCHB
|
6.4 | IC50 | 8 | Yes | |
PUIXMSRTTHLNKI
|
6.4 | IC50 | 12 | — | |
SFMJNHNUOVADRW
|
6.4 | IC50 | 7 | — | |
XZXHXSATPCNXJR
|
6.4 | Kd | 165 | Yes | |
CQWQFVNFRPNLID
|
6.4 | IC50 | 2 | — | |
DOLVPVSWTLFZMQ
|
6.4 | Ki | 17 | — |