Target Details
| UniProt AC | P51451 |
|---|---|
| Gene Symbol | BLK |
| Protein Name | Tyrosine-protein kinase Blk |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 388
- Clinical molecules 48
- Avg pChEMBL 7.08
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (388)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PQNWNVWJXPSZFR
|
6.9 | Ki | 21 | — | |
PUPCRRRSBUYJAD
|
6.9 | Ki | 44 | Yes | |
QXRJBJVCBQSLTA
|
6.9 | Ki | 29 | — | |
RPDVCUCXMGWTFA
|
6.9 | Ki | 10 | — | |
RYAVJHIPOWNWDE
|
6.9 | Ki | 38 | — | |
VUHZDNOPEVGHEO
|
6.9 | Ki | 29 | — | |
XLFYOIVELARSKP
|
6.9 | Ki | 33 | — | |
YDOPLCNFRXOHCC
|
6.9 | Ki | 28 | — | |
QQWUGDVOUVUTOY
|
6.9 | Kd | 231 | Yes | |
AILRADAXUVEEIR
|
6.9 | IC50 | 75 | — | |
APPXQUDJLJXULP
|
6.9 | IC50 | 47 | — | |
KHTYLSIHFRAWQO
|
6.9 | IC50 | 2 | — | |
BLYRPGBSIKAIAU
|
6.8 | IC50 | 24 | Yes | |
PYNRTYJUAIYHTF
|
6.8 | IC50 | 2 | — | |
PYNRTYJUAIYHTF
|
6.8 | IC50 | 2 | — | |
JIJDVLXBQGQRQM
|
6.8 | IC50 | 3 | — | |
WJEOLQLKVOPQFV
|
6.8 | Kd | 24 | — | |
NPYHVKHWRDSLAV
|
6.8 | IC50 | 3 | — | |
ACNCCUVYXQGPKZ
|
6.8 | Ki | 31 | — | |
BDPBZUHWAVABDM
|
6.8 | Ki | 11 | — | |
BHSOPYVVEZFHDB
|
6.8 | Ki | 25 | Yes | |
DXQBCGUEDOHNHP
|
6.8 | IC50 | 12 | — | |
FQYLJBVSYHZWLT
|
6.8 | Ki | 35 | Yes | |
GCYXEGSPUDSZJY
|
6.8 | Ki | 82 | — | |
GSXRCPJTNIGKSZ
|
6.8 | Ki | 43 | — | |
HQPNLIKXAPLWBQ
|
6.8 | Ki | 12 | Yes | |
SLKAFUZHONQYQY
|
6.8 | IC50 | 5 | — | |
UGXCBYVBIJACEK
|
6.8 | IC50 | 8 | — | |
UIARLYUEJFELEN
|
6.8 | Kd | 289 | Yes | |
UUVMNPKFPGJBNX
|
6.8 | Ki | 10 | — | |
UXMNYFJHEBEDJS
|
6.8 | Ki | 19 | Yes | |
WOLATEJXXTXCRC
|
6.8 | IC50 | 2 | — | |
BYWUIYIFSMRUSS
|
6.8 | Ki | 3 | — | |
DYLDTESCOKKPMG
|
6.8 | IC50 | 3 | — | |
WIZIQUFUGUEWKY
|
6.8 | IC50 | 6 | — | |
ZFDGMDVYMNWICG
|
6.8 | IC50 | 10 | — | |
YHCSNQVEOHUGIM
|
6.8 | IC50 | 2 | — | |
GFHLXZJWIUHXCL
|
6.8 | IC50 | 5 | — | |
WJZRVTHUECQQTM
|
6.7 | IC50 | 2 | — | |
AAKJLRGGTJKAMG
|
6.7 | Kd | 50 | Yes | |
BZWACBLCIHAEKY
|
6.7 | IC50 | 5 | — | |
PIQCTGMSNWUMAF
|
6.7 | Kd | 137 | Yes | |
QRDCOOSKIFYKIQ
|
6.7 | Kd | 8 | — | |
VMTZCKPMAFGPEN
|
6.7 | Ki | 3 | — | |
BSFNGHCTZDCQBF
|
6.7 | Ki | 93 | — | |
HAYYBYPASCDWEQ
|
6.7 | Ki | 47 | — | |
HEUSUIRCBWROMH
|
6.7 | Ki | 64 | — | |
IKENQUDOTQBCJH
|
6.7 | Kd | 18 | — | |
ISVHLTLEHRZKJC
|
6.7 | Ki | 19 | — | |
KRIUNPBAQZGFQA
|
6.7 | Ki | 76 | — |