Target Details
| UniProt AC | P51451 |
|---|---|
| Gene Symbol | BLK |
| Protein Name | Tyrosine-protein kinase Blk |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 388
- Clinical molecules 48
- Avg pChEMBL 7.08
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (388)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WINHZLLDWRZWRT
|
7.2 | Ki | 66 | — | |
WINHZLLDWRZWRT
|
7.2 | Kd | 201 | Yes | |
UHTHHESEBZOYNR
|
7.2 | Kd | 66 | Yes | |
HHFBDROWDBDFBR
|
7.2 | Kd | 40 | Yes | |
BLWDOLCMBQDSMT
|
7.2 | IC50 | 4 | — | |
LNCCSXUMNALGKS
|
7.1 | IC50 | 2 | — | |
OPKHZFMFWCMAPS
|
7.1 | IC50 | 6 | — | |
JWNAINYXINYHML
|
7.1 | IC50 | 3 | — | |
OSAWFUCUZJNEID
|
7.1 | IC50 | 20 | — | |
LAUHLGUSVSJYCI
|
7.1 | IC50 | 16 | — | |
WVUNYSQLFKLYNI
|
7.1 | Kd | 46 | Yes | |
DLPARMNJOHFOLU
|
7.1 | Ki | 14 | Yes | |
DZSUJUOJJJCWGG
|
7.1 | Ki | 55 | Yes | |
GALVWTFFXPRMQM
|
7.1 | Ki | 20 | — | |
NRGYZNJPCGRCLV
|
7.1 | Ki | 52 | — | |
OTVCFDOYUHREFJ
|
7.1 | Ki | 26 | — | |
SFPWNTQWFFNJIH
|
7.1 | Ki | 48 | — | |
XCHWBXBDZRJVDP
|
7.1 | Ki | 51 | — | |
ZVWRFVCNQOECJS
|
7.1 | Ki | 71 | — | |
DQHVUKLVCBJBLM
|
7.1 | IC50 | 8 | — | |
AHBFBRPGNOVEBK
|
7.1 | IC50 | 11 | — | |
JXVBUPCEADJXCV
|
7.1 | IC50 | 4 | — | |
JWNPDZNEKVCWMY
|
7.1 | Kd | 57 | Yes | |
UFEYPVTVHUTYJF
|
7.0 | IC50 | 4 | — | |
NZIQNLGMMJGSQU
|
7.0 | IC50 | 6 | — | |
FGPPXNCHKYRZCI
|
7.0 | IC50 | 6 | — | |
KNVOICXEDILAGT
|
7.0 | Ki | 17 | — | |
LVECPYVAIBNSRV
|
7.0 | Ki | 33 | — | |
MTCHQDWUHQADSY
|
7.0 | Ki | 29 | — | |
OMIQRSKHABIPRH
|
7.0 | IC50 | 15 | — | |
PTVPBWWDGZSEAF
|
7.0 | Ki | 63 | — | |
RTYJMUXLFRYRBU
|
7.0 | Ki | 35 | — | |
RYYNGWLOYLRZLK
|
7.0 | Ki | 104 | — | |
WUWDLXZGHZSWQZ
|
7.0 | Ki | 41 | — | |
XJSFDMGICAWQFS
|
7.0 | Ki | 60 | — | |
XYXLUJQBBIBJFV
|
7.0 | Ki | 36 | — | |
TWWKXZDIDHDHRF
|
7.0 | IC50 | 7 | — | |
KTEIFNKAUNYNJU
|
7.0 | Kd | 114 | — | |
ZATZMKDSRSJODQ
|
7.0 | IC50 | 2 | — | |
SHPFDGWALWEPGS
|
6.9 | Kd | 35 | — | |
XXJWYDDUDKYVKI
|
6.9 | Kd | 52 | — | |
CMZKQVFPFYPHOD
|
6.9 | IC50 | 3 | — | |
DBXOMQJZSQLQED
|
6.9 | Ki | 12 | — | |
DMTDZFGYURLLKX
|
6.9 | Ki | 13 | Yes | |
JZTOUVBEZONDKA
|
6.9 | Ki | 80 | — | |
KUNZDWIFPOMUOX
|
6.9 | Ki | 36 | — | |
NFMGZVPRGVERNN
|
6.9 | Ki | 44 | — | |
NHFDRBXTEDBWCZ
|
6.9 | Ki | 41 | — | |
NWAUBAGBGOPJLF
|
6.9 | Ki | 51 | Yes | |
NZVDDFRUBIEKLV
|
6.9 | Ki | 20 | — |