Target Details
| UniProt AC | P51451 |
|---|---|
| Gene Symbol | BLK |
| Protein Name | Tyrosine-protein kinase Blk |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 388
- Clinical molecules 48
- Avg pChEMBL 7.08
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (388)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ORRHVRJUSPCILV
|
7.5 | Ki | 16 | — | |
VWVYILCFSYNJHF
|
7.5 | Ki | 49 | — | |
XNEPVLVYFUGJLF
|
7.5 | Ki | 27 | — | |
CBRJPFGIXUFMTM
|
7.5 | Ki | 7 | — | |
XNVVTSSPSNFSCT
|
7.5 | IC50 | 3 | — | |
XXKYXXNDMNIKFT
|
7.5 | IC50 | 2 | — | |
PTHVKCSYXICMAR
|
7.4 | IC50 | 14 | — | |
ZVPDNRVYHLRXLX
|
7.4 | IC50 | 35 | Yes | |
CZQVOIDVDAVDFW
|
7.4 | Ki | 18 | — | |
NRZYTPAJGVTKIM
|
7.4 | Ki | 38 | — | |
NSYXCWYWACQNOH
|
7.4 | Ki | 10 | — | |
XKFTZKGMDDZMJI
|
7.4 | Ki | 56 | — | |
ZLHFILGSQDJULK
|
7.4 | Ki | 37 | Yes | |
SZFYZDIPRMLBDC
|
7.4 | IC50 | 9 | — | |
HJURBXZLFARTFO
|
7.4 | IC50 | 2 | — | |
XYFZVVYVIFJBIS
|
7.4 | IC50 | 17 | — | |
RJVBLELKWSSFMN
|
7.4 | IC50 | 2 | — | |
OMZCMEYTWSXEPZ
|
7.3 | Kd | 43 | Yes | |
OSVUGUHRKMMBSE
|
7.3 | Kd | 170 | — | |
OXQLPBHQZPVYQX
|
7.3 | IC50 | 2 | — | |
FDVSOQRNTAPCHB
|
7.3 | IC50 | 7 | Yes | |
DKSNLQYRZJKYOC
|
7.3 | Ki | 51 | — | |
GZYUJXFTHLKPAK
|
7.3 | IC50 | 16 | — | |
HKZKELVPGXJIMW
|
7.3 | Ki | 41 | — | |
LYHDXABKNJMNEZ
|
7.3 | Ki | 10 | — | |
MVJMMLFMPWITEJ
|
7.3 | Ki | 110 | — | |
NFKMFNBKEOQNPZ
|
7.3 | Ki | 43 | — | |
XFWUTMHVDGPWLH
|
7.3 | Ki | 75 | — | |
UORAPQCBWYIISR
|
7.3 | IC50 | 12 | — | |
VTJHGMZHVOXJPG
|
7.3 | IC50 | 15 | — | |
HSYNEJBNGIWWIC
|
7.3 | IC50 | 2 | — | |
IBCGPVVKHZXWNX
|
7.3 | IC50 | 7 | — | |
LLRUOFRCNQYKAO
|
7.3 | IC50 | 3 | — | |
NJKRMPNUGZAMJN
|
7.3 | IC50 | 5 | — | |
XNJQHXBRQQSGDT
|
7.3 | IC50 | 2 | — | |
CEUSZLVORFRBCV
|
7.2 | IC50 | 13 | — | |
ASMLDRAEBPYENO
|
7.2 | IC50 | 10 | — | |
JBTQYTBFFKJOSI
|
7.2 | IC50 | 2 | — | |
MIMOHMCANSGXIG
|
7.2 | IC50 | 15 | — | |
BLQYVHBZHAISJM
|
7.2 | Ki | 54 | — | |
DCTBPIBEQFLAOQ
|
7.2 | Ki | 13 | — | |
GWMATETWMAQOFL
|
7.2 | Ki | 36 | — | |
IAKGNUWZPSPEKU
|
7.2 | Ki | 19 | — | |
JAMDNXUAYUHJLJ
|
7.2 | Ki | 40 | — | |
LGHBDVLAHHANMX
|
7.2 | Ki | 53 | — | |
LRLDYTTWQIFWBD
|
7.2 | Ki | 25 | — | |
NXSJMRCTGYTSTK
|
7.2 | Kd | 200 | — | |
SRUYMJRFVGLQDV
|
7.2 | Ki | 37 | — | |
UOVCGJXDGOGOCZ
|
7.2 | Ki | 59 | — | |
UUWNXFJBBYAMDT
|
7.2 | Ki | 46 | — |