Target Details
| UniProt AC | P51451 |
|---|---|
| Gene Symbol | BLK |
| Protein Name | Tyrosine-protein kinase Blk |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 388
- Clinical molecules 48
- Avg pChEMBL 7.08
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (388)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
8.0 | IC50 | 213 | — | |
ADLPKFFMGIJZIM
|
8.0 | Ki | 44 | — | |
FLEAYYMORDPWAJ
|
8.0 | Ki | 90 | — | |
LXURGGKEOPHREO
|
8.0 | IC50 | 13 | — | |
GUBJNPWVIUFSTR
|
8.0 | Kd | 103 | — | |
WAXWZMRXSJUAGV
|
8.0 | IC50 | 2 | — | |
LQSGDXCDNZWTJN
|
7.9 | IC50 | 17 | — | |
JSDGKSMNPHJDFK
|
7.9 | Ki | 35 | — | |
OWFXKTOLFUQPDJ
|
7.9 | Ki | 36 | — | |
WZZXMNBOPNKKSX
|
7.9 | Ki | 10 | — | |
XBYVOPRDASFDMY
|
7.9 | Ki | 42 | — | |
XHORJSJFHVABEA
|
7.9 | Ki | 49 | — | |
PPGPPDAKFCUXOF
|
7.9 | IC50 | 2 | — | |
FOKYFSPHYRIEJZ
|
7.8 | IC50 | 2 | — | |
FCXFBAVJAPHCTG
|
7.8 | IC50 | 3 | — | |
CFIBXVQLBVNOHW
|
7.8 | Ki | 64 | — | |
CNTCGRJDUJEUDG
|
7.8 | Ki | 37 | — | |
RWSXMGOKPQHHNZ
|
7.8 | IC50 | 2 | — | |
UXQLMVSZSYZFID
|
7.8 | Ki | 12 | — | |
YHVHYWYQEFELOW
|
7.8 | IC50 | 44 | — | |
YMSXHRWUGLAAKL
|
7.8 | IC50 | 14 | Yes | |
ZKHDDJKHTPLPOQ
|
7.8 | Ki | 62 | — | |
ZWVZORIKUNOTCS
|
7.8 | Ki | 69 | — | |
FUZSHLVNKZZEKR
|
7.8 | IC50 | 16 | — | |
MRXCLHVAIIGTOJ
|
7.8 | IC50 | 2 | — | |
WDENQIQQYWYTPO
|
7.8 | Kd | 8 | — | |
BNRXMSGHPVYSDK
|
7.7 | IC50 | 24 | — | |
JUSWPUDQOKINJO
|
7.7 | IC50 | 16 | — | |
MULNSLQVKKUPJN
|
7.7 | Ki | 41 | — | |
TVJRDCQUZMGBAB
|
7.7 | IC50 | 13 | — | |
CVWXJKQAOSCOAB
|
7.7 | IC50 | 35 | — | |
VYZQSAKXLMEDCB
|
7.7 | IC50 | 9 | — | |
CDISOBGWDHAHGF
|
7.7 | IC50 | 16 | — | |
LZECOFRPCLZCOI
|
7.7 | IC50 | 4 | — | |
ZRYMMWAJAFUANM
|
7.6 | IC50 | 7 | — | |
BIKYDWLMTPRSQL
|
7.6 | Ki | 50 | — | |
MQRDVGBWWVWMEN
|
7.6 | Ki | 47 | — | |
NHHQJBCNYHBUSI
|
7.6 | Kd | 220 | — | |
RVHUGWYTNUUGPJ
|
7.6 | IC50 | 2 | — | |
YISMQBFJYDFMAL
|
7.6 | IC50 | 46 | — | |
LSJWYMSFUWBGPN
|
7.5 | IC50 | 17 | — | |
JMVDIGHUQAXWIE
|
7.5 | IC50 | 10 | — | |
ODPGGGTTYSGTGO
|
7.5 | Kd | 153 | — | |
XJVQNHKBZSHCJV
|
7.5 | IC50 | 2 | — | |
DASFSPDIWCMVRW
|
7.5 | Ki | 21 | — | |
GCIKSSRWRFVXBI
|
7.5 | Ki | 109 | Yes | |
KKYPRNBBPBRJQX
|
7.5 | Ki | 40 | — | |
KNACLJBHKVSTDL
|
7.5 | Ki | 40 | — | |
MFMXAWQGPQXDRJ
|
7.5 | Ki | 27 | — | |
MICOMLRETSSUOK
|
7.5 | IC50 | 3 | — |