Target Details
| UniProt AC | P51451 |
|---|---|
| Gene Symbol | BLK |
| Protein Name | Tyrosine-protein kinase Blk |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 388
- Clinical molecules 48
- Avg pChEMBL 7.08
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (388)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KJRVCMVPIKELBC
|
9.7 | IC50 | 12 | — | |
SSDFTYWIYVWCIE
|
9.7 | IC50 | 17 | — | |
ZBNZXTGUTAYRHI
|
9.7 | Kd | 102 | Yes | |
LCYSSHSIKSARGO
|
9.3 | IC50 | 19 | — | |
NNGVMERLTTVLQP
|
9.3 | IC50 | 8 | — | |
XYFPWWZEPKGCCK
|
9.3 | IC50 | 34 | — | |
CXBBWVXSZINRCS
|
9.1 | Ki | 41 | — | |
OWRXHGAFWZFFCW
|
9.0 | Ki | 113 | — | |
SFCBIFOAGRZJNX
|
9.0 | Kd | 22 | — | |
UOOZSMNSBYVUGZ
|
9.0 | Ki | 32 | — | |
RNOAOAWBMHREKO
|
8.9 | IC50 | 15 | — | |
WVXNSAVVKYZVOE
|
8.9 | IC50 | 92 | — | |
ULMCFLZUGRSEQA
|
8.9 | Ki | 17 | — | |
BJMXICGJKUALLN
|
8.8 | IC50 | 8 | — | |
VAARYSWULJUGST
|
8.8 | Kd | 119 | Yes | |
HKSZLNNOFSGOKW
|
8.8 | Ki | 118 | — | |
KCPKCAYWGNEVBR
|
8.8 | IC50 | 7 | — | |
MCCCQFAOMZMZKE
|
8.8 | Ki | 52 | — | |
RBXYGQNZRVPDNB
|
8.8 | Ki | 34 | — | |
XKZINYYXWJEYEL
|
8.7 | Ki | 37 | — | |
KZMQPYCXSAGLTB
|
8.7 | IC50 | 8 | — | |
PZWSKESWDIFAFK
|
8.6 | IC50 | 9 | — | |
WPHKIQPVPYJNAX
|
8.6 | Ki | 81 | — | |
HKSZLNNOFSGOKW
|
8.6 | IC50 | 408 | — | |
KNARVZUUCLIBGV
|
8.5 | Ki | 33 | — | |
UGEJLCNSVIVALC
|
8.5 | Ki | 41 | — | |
XOOAAYRIVATZNM
|
8.5 | Ki | 55 | — | |
ZCCJKVBTHCOISJ
|
8.5 | Ki | 46 | — | |
UBPYILGKFZZVDX
|
8.5 | Kd | 130 | Yes | |
SMOPKEHQPPXRSH
|
8.4 | IC50 | 8 | — | |
CQBBMNXXVMOFCA
|
8.3 | Ki | 39 | — | |
IRBVGTPPFBYDKX
|
8.3 | IC50 | 9 | — | |
MHCPAORAYMTGCZ
|
8.3 | Ki | 37 | — | |
ULHGAQSVFPOUDY
|
8.3 | Ki | 43 | — | |
CXQHYVUVSFXTMY
|
8.3 | Kd | 154 | — | |
JTHOLYGYPAXIFD
|
8.3 | IC50 | 2 | — | |
SEJGTFPOEJWEGG
|
8.3 | Kd | 149 | — | |
YEVYGRCYEKDRGH
|
8.2 | IC50 | 2 | — | |
BTWVWABAWDKQNJ
|
8.2 | IC50 | 8 | — | |
LCFFREMLXLZNHE
|
8.2 | IC50 | 5 | — | |
QJIVDCJIPGAKQZ
|
8.2 | Ki | 25 | — | |
JLONRANGHBAJIS
|
8.2 | IC50 | 2 | — | |
GDRLJBDXWDATLA
|
8.1 | IC50 | 13 | — | |
RVCKMZIQUFKZFD
|
8.1 | IC50 | 7 | — | |
KPZGJWPPVXZLDN
|
8.1 | IC50 | 10 | — | |
SRSQULBCTWSVKL
|
8.1 | IC50 | 15 | — | |
AWZWOMPLEBTAGQ
|
8.1 | IC50 | 2 | — | |
NYBJZNNMOLQLJD
|
8.1 | IC50 | 2 | — | |
OPHSZSZDICRBPP
|
8.1 | IC50 | 16 | — | |
VKBFHTIUXUCYRQ
|
8.1 | Ki | 66 | — |