Target Details
| UniProt AC | P51449 |
|---|---|
| Gene Symbol | RORC |
| Protein Name | Nuclear receptor ROR-gamma |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 95
- Clinical molecules 0
- Avg pChEMBL 7.36
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (95)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZDHFRWUXYBOYAJ
|
7.2 | IC50 | 2 | — | |
LNDNBCFVCPXIRA
|
7.2 | IC50 | 2 | — | |
WUZNZQZEJJUMBN
|
7.2 | IC50 | 2 | — | |
QBKPVUOATLEJDS
|
7.1 | IC50 | 2 | — | |
QBIGUDRHHJTXKG
|
7.0 | IC50 | 2 | — | |
LTMHDMANZUZIPE
|
7.0 | Kd | 10 | — | |
OZBSSKGBKHOLGA
|
7.0 | Ki | 2 | — | |
AFZMZLHHVUIZBS
|
6.9 | IC50 | 2 | — | |
WCGUUGGRBIKTOS
|
6.9 | IC50 | 5 | — | |
ZBVWPYZPEXTFFC
|
6.9 | IC50 | 2 | — | |
AFZMZLHHVUIZBS
|
6.8 | IC50 | 2 | — | |
ILXLMNLDODDHOQ
|
6.8 | Ki | 2 | — | |
WUZNZQZEJJUMBN
|
6.8 | IC50 | 2 | — | |
AFZMZLHHVUIZBS
|
6.8 | IC50 | 2 | — | |
SHGAZHPCJJPHSC
|
6.7 | IC50 | 13 | — | |
ASEWBZJHLDHXLR
|
6.7 | Ki | 2 | — | |
ACTPLOYOROGJBM
|
6.6 | IC50 | 2 | — | |
QWFSPUISXUYUCI
|
6.6 | IC50 | 2 | — | |
SGIWFELWJPNFDH
|
6.6 | IC50 | 6 | — | |
LRZLWEPJKYOTMH
|
6.5 | IC50 | 2 | — | |
OYCQSCPHBYKGHN
|
6.5 | IC50 | 2 | — | |
YPTBGUKCVIWVDD
|
6.5 | IC50 | 2 | — | |
PDAASAKPBNZZQB
|
6.4 | IC50 | 2 | — | |
DATNOEKWAMTIHN
|
6.3 | IC50 | 2 | — | |
JXWVEYDXIMPHDP
|
6.3 | IC50 | 2 | — | |
OGODHXWGKYDWLS
|
6.3 | IC50 | 2 | — | |
AKMCELRJWFESNG
|
6.3 | IC50 | 2 | — | |
AZVDUNZVEKRQNT
|
6.3 | IC50 | 2 | — | |
FGXJJPWNKQTSEM
|
6.3 | IC50 | 2 | — | |
FXTXQRXJLIGODT
|
6.3 | IC50 | 2 | — | |
HFMXKUVVFZSMNI
|
6.3 | IC50 | 2 | — | |
HTLJGDDOXOYDIA
|
6.3 | IC50 | 2 | — | |
IVJZFFBZAPYDHF
|
6.3 | IC50 | 2 | — | |
LDYXWSQWGGILQQ
|
6.3 | IC50 | 2 | — | |
MGNNUHSXEBVLGO
|
6.3 | IC50 | 2 | — | |
QCNYOMWEVRZCBH
|
6.3 | IC50 | 2 | — | |
RKEKMGUGGBHNDU
|
6.3 | IC50 | 2 | — | |
RYXBKDXGNAYCOV
|
6.3 | IC50 | 2 | — | |
BXVPMFQBRUNLCJ
|
6.2 | IC50 | 2 | — | |
KBOKCQLFWLAHHN
|
6.2 | IC50 | 2 | — | |
DSIYRAHIZDXKRO
|
6.1 | IC50 | 2 | — | |
HEPPZYJPFBGTKA
|
6.1 | IC50 | 2 | — | |
IEMKKJCNFFIONU
|
6.0 | IC50 | 2 | — | |
OKKXBHWKOBOMGK
|
6.0 | Ki | 2 | — | |
GZBZDZWXLLKUTQ
|
6.0 | IC50 | 2 | — |