Target Details
| UniProt AC | P51449 |
|---|---|
| Gene Symbol | RORC |
| Protein Name | Nuclear receptor ROR-gamma |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 95
- Clinical molecules 0
- Avg pChEMBL 7.36
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (95)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZDBJECNSNPXCFS
|
9.2 | IC50 | 2 | — | |
JFBZAEQCYPRNMQ
|
9.2 | IC50 | 2 | — | |
KXWLXPUSRXLJCK
|
9.1 | IC50 | 2 | — | |
SLMOKTWBUBMWJO
|
9.1 | IC50 | 2 | — | |
KYIGOCCCBXRHNJ
|
9.0 | IC50 | 43 | — | |
IORGFFCZJYGRQD
|
9.0 | IC50 | 2 | — | |
QLKWBZGQDXUAPZ
|
9.0 | IC50 | 2 | — | |
FOOFCMISAIJPLF
|
8.9 | IC50 | 2 | — | |
PSFPATVFAWGHAJ
|
8.8 | IC50 | 2 | — | |
VICVDIVPAGQTTO
|
8.8 | IC50 | 2 | — | |
SPDXXZUHXTYAPT
|
8.7 | IC50 | 2 | — | |
FQNXGRKEBPOPHJ
|
8.6 | IC50 | 2 | — | |
NSAOHDFDPAPARQ
|
8.5 | IC50 | 2 | — | |
BENOEPUDOPGLCP
|
8.5 | IC50 | 2 | — | |
KIAHYBIZSGNTBR
|
8.4 | IC50 | 2 | — | |
ZHSFCHXKHOJYIG
|
8.4 | IC50 | 2 | — | |
KEKCGMLTBGENHB
|
8.4 | Ki | 2 | — | |
HCTASJAOJYRGPC
|
8.4 | IC50 | 2 | — | |
CZZWOGGSAFJKEU
|
8.4 | IC50 | 2 | — | |
ULYHXRTUZSKYEU
|
8.4 | IC50 | 2 | — | |
ISWGZOZQPRMRJA
|
8.3 | IC50 | 2 | — | |
MNUCRODXGZMPCU
|
8.3 | IC50 | 3 | — | |
GPALVRLYDQFPIU
|
8.3 | IC50 | 2 | — | |
DANLZOIRUUHIIX
|
8.2 | IC50 | 2 | — | |
LRJKAYGDKHTSDL
|
8.1 | IC50 | 2 | — | |
FPEPDZZKOGUYFO
|
8.1 | IC50 | 2 | — | |
IOWMKBFJCNLRTC
|
8.0 | Ki | 3 | — | |
OYXZMSRRJOYLLO
|
8.0 | Ki | 2 | — | |
OYXZMSRRJOYLLO
|
8.0 | Ki | 2 | — | |
XFHHIVHARPRKCG
|
8.0 | IC50 | 2 | — | |
GZCDNIGGYFEPLV
|
7.9 | IC50 | 2 | — | |
PWNQDXFSXNJRRQ
|
7.8 | IC50 | 3 | — | |
MREFIIMUWJNTII
|
7.7 | IC50 | 2 | — | |
GRWNPFJXINLSNF
|
7.7 | IC50 | 2 | — | |
SBHFAQDIXHCJBY
|
7.7 | IC50 | 2 | — | |
VHGGVTVFPZUWCU
|
7.6 | IC50 | 2 | — | |
XNZJHNCNFWAVAE
|
7.5 | IC50 | 3 | — | |
TUMWNEOCLIEIOQ
|
7.5 | IC50 | 2 | — | |
VTRHQLPYGVWKKI
|
7.5 | IC50 | 2 | — | |
HJJYGXDBXQAVQG
|
7.4 | IC50 | 2 | — | |
KEKPYTHQPDLLDE
|
7.4 | IC50 | 2 | — | |
HVDDJVICMSYNIS
|
7.4 | IC50 | 2 | — | |
QYYZXEPEVBXNNA
|
7.4 | IC50 | 2 | — | |
AVHWMAVUUHFRKE
|
7.3 | IC50 | 2 | — | |
QQIBJFMXQBDPGQ
|
7.3 | IC50 | 2 | — | |
FYIJFWZBSFEMNI
|
7.3 | IC50 | 2 | — | |
MGOPCYIZHYONRL
|
7.3 | IC50 | 2 | — | |
WWWWYLGWKNWDLQ
|
7.3 | IC50 | 2 | — | |
AVHWMAVUUHFRKE
|
7.3 | IC50 | 2 | — | |
JKDVOVFYDAXBSL
|
7.2 | IC50 | 2 | — |