Target Details
| UniProt AC | P51160 |
|---|---|
| Gene Symbol | PDE6C |
| Protein Name | Cone cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha' |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01590 (GAF) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 70
- Clinical molecules 0
- Avg pChEMBL 7.42
KEGG Pathways (2)
Associated Diseases (2)
Active Molecules (70)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
REZGGXNDEMKIQB
|
6.4 | Ki | 8 | — | |
UEHYTJCPYRCAPM
|
6.4 | IC50 | 8 | — | |
SRUIZVZXCPBTGE
|
6.3 | IC50 | 3 | — | |
CIKOPVDFPXGTDP
|
6.3 | IC50 | 8 | — | |
BWVJYTGTOWKCOX
|
6.3 | IC50 | 8 | — | |
SDYQZLQJADODFL
|
6.3 | Ki | 7 | — | |
XJCFZDNOEIPPIC
|
6.3 | IC50 | 7 | — | |
PUJFXPWIBOJQHB
|
6.2 | IC50 | 12 | — | |
UEMKDTSBXWIJFQ
|
6.2 | IC50 | 7 | — | |
VFFZRVLFFCXMEW
|
6.2 | Ki | 7 | — | |
WTHIWWQIRPIFLQ
|
6.2 | IC50 | 8 | — | |
HLUWBLAYMFWHOF
|
6.1 | IC50 | 8 | — | |
INLBUQIADGPECI
|
6.1 | IC50 | 2 | — | |
RPLZXBUKXSYWDQ
|
6.1 | IC50 | 10 | — | |
RCUCFFJDNMXZAV
|
6.1 | Ki | 7 | — | |
SGZFBLCNGYGISG
|
6.1 | IC50 | 8 | — | |
QBLWGJRSTWQUGT
|
6.0 | IC50 | 8 | — | |
JITUOVWOCIXEEZ
|
6.0 | IC50 | 23 | — | |
NWOYPSQSXFBTCX
|
6.0 | IC50 | 6 | — | |
OWWOVESWHWBLEI
|
6.0 | IC50 | 6 | — |