Target Details
| UniProt AC | P51160 |
|---|---|
| Gene Symbol | PDE6C |
| Protein Name | Cone cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha' |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01590 (GAF) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 70
- Clinical molecules 0
- Avg pChEMBL 7.42
KEGG Pathways (2)
Associated Diseases (2)
Active Molecules (70)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UJLHNYPXKZJKLV
|
10.0 | IC50 | 24 | — | |
KXCOKRBRUWINCT
|
9.9 | IC50 | 24 | — | |
GDXUQGMYOAPPJF
|
9.9 | IC50 | 6 | — | |
KPFFPWNKWSYQFT
|
9.8 | IC50 | 24 | — | |
GOBQSCBEINUNFL
|
9.6 | IC50 | 24 | — | |
AFCWMWBOATWMJV
|
9.5 | IC50 | 24 | — | |
DKSKKVAOIPURFT
|
9.5 | IC50 | 24 | — | |
YJBDHZKAVGNHET
|
9.1 | IC50 | 2 | — | |
BPBDCOLBZYWXHD
|
9.0 | IC50 | 24 | — | |
FMMIDZWTNQYEIY
|
9.0 | IC50 | 24 | — | |
IFMLEMDUMAPODC
|
8.9 | IC50 | 3 | — | |
VNWKVRSLWCIUCC
|
8.9 | IC50 | 7 | — | |
AANJEOKXWMXQIE
|
8.8 | IC50 | 2 | — | |
NGFDENLSEDFSFN
|
8.8 | IC50 | 4 | — | |
RNHNQORGLGCJLQ
|
8.8 | IC50 | 3 | — | |
HIEBSPLRWFLZPT
|
8.7 | IC50 | 7 | — | |
RNHNQORGLGCJLQ
|
8.6 | IC50 | 2 | — | |
WFSWUBOROARLDR
|
8.6 | IC50 | 7 | — | |
DRWIDCWXXLOIMG
|
8.4 | IC50 | 2 | — | |
RNHNQORGLGCJLQ
|
8.4 | IC50 | 2 | — | |
IFMLEMDUMAPODC
|
8.3 | IC50 | 2 | — | |
NWAWSQQMTQQBGL
|
8.3 | IC50 | 4 | — | |
QQMRBUUPHPWYOK
|
8.2 | IC50 | 2 | — | |
CXMJWJJNVWXSJV
|
8.2 | IC50 | 2 | — | |
LMZYNSBAUOTKJP
|
8.1 | IC50 | 7 | — | |
SECKRCOLJRRGGV
|
8.0 | IC50 | 16 | — | |
PIOIVHHIGWTEJQ
|
7.7 | IC50 | 3 | — | |
YLBRHUHHQIYMSH
|
7.5 | IC50 | 7 | — | |
IFMLEMDUMAPODC
|
7.5 | IC50 | 2 | — | |
BNRNXUUZRGQAQC
|
7.4 | IC50 | 12 | — | |
FJJLJIBQQGUEHI
|
7.3 | IC50 | 2 | — | |
ILKQRTXPJWHTCQ
|
7.2 | IC50 | 7 | — | |
ZXGQTWGCVTUQHJ
|
7.1 | IC50 | 8 | — | |
PNROCVKVRSRTPH
|
7.0 | IC50 | 2 | — | |
IZEKFCXSFNUWAM
|
6.9 | Ki | 19 | — | |
JTZIKJJODWLHHP
|
6.8 | IC50 | 2 | — | |
HVDQYPSFEUUGDN
|
6.8 | IC50 | 8 | — | |
IQOUMUUIJXJPMR
|
6.7 | IC50 | 2 | — | |
WVFZLLHYILMVBO
|
6.7 | Ki | 7 | — | |
WKEBNSYJGBPIKM
|
6.6 | IC50 | 3 | — | |
RNLNRXGCWGOQMW
|
6.6 | Ki | 7 | — | |
WDRWBLDUZZTZRV
|
6.6 | IC50 | 8 | — | |
ANFPYGBSFPVDQM
|
6.5 | IC50 | 7 | — | |
MXRCTQYKTXQWTH
|
6.5 | IC50 | 3 | — | |
OFZGCAMFVYIIHV
|
6.5 | IC50 | 24 | — | |
OTFYWELOCYDGRZ
|
6.5 | IC50 | 7 | — | |
YKLLPTMXZQKNGA
|
6.5 | IC50 | 7 | — | |
FGBIHGKWPVSHSO
|
6.5 | IC50 | 7 | — | |
MIATWQLLYKUWRD
|
6.5 | IC50 | 8 | — | |
QDPNAMRLQRQPMR
|
6.4 | IC50 | 2 | — |