Target Details
| UniProt AC | P50750 |
|---|---|
| Gene Symbol | CDK9 |
| Protein Name | Cyclin-dependent kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 3,102
- Clinical molecules 43
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (3,102)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LSLPDHNUWRDOGC
|
8.1 | Ki | 25 | — | |
MFGPPACYEFGSTK
|
8.1 | IC50 | 2 | — | |
NBOBLXOZHBALAX
|
8.1 | IC50 | 7 | — | |
NIVRVOZNYYXNJT
|
8.1 | Ki | 7 | — | |
OVOYRPVIZNJKHS
|
8.1 | Ki | 3 | — | |
PDCHCLPILDWNBF
|
8.1 | IC50 | 2 | — | |
PSNUTPHNERQRHY
|
8.1 | Ki | 4 | — | |
PUWXPMFEDYRLTM
|
8.1 | IC50 | 6 | — | |
QLQYWGHSSLXLOS
|
8.1 | IC50 | 5 | — | |
VNWYGUWLGRESFH
|
8.1 | IC50 | 2 | — | |
ZVLFDFWFDUVCGU
|
8.1 | IC50 | 2 | — | |
FGFWZFYILZKNBW
|
8.1 | IC50 | 6 | — | |
KZZDDXBCJROTIP
|
8.1 | IC50 | 8 | — | |
FUTHHRJWHRJGTO
|
8.1 | IC50 | 2 | — | |
BJBUTEFLQLIASF
|
8.1 | IC50 | 2 | — | |
HXKORJQOSCRLJP
|
8.1 | IC50 | 5 | — | |
IWSDTEGBQVXXON
|
8.1 | IC50 | 7 | — | |
MMEWHQQSISZZCB
|
8.1 | IC50 | 4 | — | |
OQWUAZIPUCLTLQ
|
8.1 | Ki | 2 | — | |
FTGMCTBSWOHGKU
|
8.1 | IC50 | 2 | — | |
SRVYTIFEXUTLAJ
|
8.1 | IC50 | 2 | — | |
VRAAFABYEISPSR
|
8.1 | IC50 | 2 | — | |
BCKLVLDQAAHMQR
|
8.1 | Ki | 9 | — | |
CUCSXQCVIUDKLI
|
8.1 | IC50 | 2 | — | |
FRCIRPZMZDFVMQ
|
8.1 | IC50 | 7 | — | |
JMMUQUKOEOPQHB
|
8.1 | IC50 | 2 | — | |
JWILUIVAYLRFIY
|
8.1 | IC50 | 14 | — | |
OWQKUKUKXLQRLY
|
8.1 | IC50 | 2 | — | |
PGVNLOUNSPQGJP
|
8.1 | IC50 | 2 | — | |
PGWURUYAKNYOPM
|
8.1 | IC50 | 4 | — | |
PMDRZLBXPGVEJA
|
8.1 | IC50 | 2 | — | |
QWDLZMUWYCLKFF
|
8.1 | IC50 | 10 | — | |
RSQPNXBTPUXMQN
|
8.1 | IC50 | 12 | — | |
RVUBWQGGWDXZIZ
|
8.1 | IC50 | 2 | — | |
RWSCYFXGWJPUQX
|
8.1 | IC50 | 15 | — | |
SCIUSXXNEKMFGZ
|
8.1 | IC50 | 3 | — | |
SSYDFQIYUKDMQD
|
8.1 | IC50 | 2 | — | |
VEJCMMPVTMQFME
|
8.1 | Ki | 8 | Yes | |
XHAWHVHQZTVHLI
|
8.1 | Ki | 4 | — | |
YXPYASILVCWNCO
|
8.1 | IC50 | 2 | — | |
ZBJGREHWROGYRW
|
8.1 | IC50 | 2 | — | |
HFKMNAUFISJBSK
|
8.0 | IC50 | 6 | — | |
HLOKDQHOCMHLLI
|
8.0 | IC50 | 7 | — | |
IPJTWBVRFFWMHE
|
8.0 | IC50 | 4 | — | |
VKXBNFWRQLNUFV
|
8.0 | IC50 | 4 | — | |
ZCSRAPNEOQVRBC
|
8.0 | IC50 | 4 | — | |
GWJUJVNEBMMNHN
|
8.0 | IC50 | 4 | — | |
PYHFRPQJHUMRSC
|
8.0 | IC50 | 2 | — | |
WYWZAULLJUBLLM
|
8.0 | IC50 | 2 | — | |
XENCJIFLJHOJNF
|
8.0 | IC50 | 2 | — |