Target Details
| UniProt AC | P50750 |
|---|---|
| Gene Symbol | CDK9 |
| Protein Name | Cyclin-dependent kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 3,102
- Clinical molecules 43
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (3,102)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BIIVYFLTOXDAOV
|
8.2 | Kd | 29 | — | |
DLJLBQIBEFHGOE
|
8.2 | IC50 | 4 | — | |
IVEUUAYDXCENND
|
8.2 | IC50 | 4 | — | |
MPBLVVMMAMGCPJ
|
8.2 | IC50 | 4 | — | |
XLEXQTAZFDJBEA
|
8.2 | IC50 | 2 | — | |
ZLFLFYDVPNHBPQ
|
8.2 | IC50 | 2 | — | |
ANELMUPUYRZVHZ
|
8.2 | IC50 | 7 | — | |
DTHXVNCIPNCYCT
|
8.2 | IC50 | 2 | — | |
JJEJUQGQRITNHI
|
8.2 | IC50 | 2 | — | |
GNEARXSVRDSWKT
|
8.2 | IC50 | 7 | — | |
JMXKUBXNZGHANG
|
8.2 | IC50 | 2 | — | |
XCTBUXUNIXTCND
|
8.2 | IC50 | 2 | — | |
YRUAMADPOZOPBF
|
8.2 | IC50 | 7 | — | |
LIJUCWLALFXGCL
|
8.2 | IC50 | 7 | — | |
OUSFTKFNBAZUKL
|
8.2 | IC50 | 58 | Yes | |
BGPUFSMDGGQOIE
|
8.2 | Ki | 9 | — | |
BSUDUKKQFRGZBK
|
8.2 | Ki | 4 | — | |
CJJMNECGBUPMAV
|
8.2 | IC50 | 8 | Yes | |
DZHBFQMOLIUZMP
|
8.2 | Ki | 9 | — | |
GTHTUFBVEUQVRV
|
8.2 | IC50 | 2 | — | |
JONJATYOSABZNY
|
8.2 | IC50 | 4 | — | |
MCFCYLCLAYXQIZ
|
8.2 | Ki | 9 | — | |
OVPNQJVDAFNBDN
|
8.2 | IC50 | 44 | Yes | |
PJIPYWGIYRUKIG
|
8.2 | Ki | 8 | — | |
UBKCVLVAEFXGTJ
|
8.2 | Ki | 5 | — | |
YFYSQSYEQXVGJJ
|
8.2 | IC50 | 2 | — | |
YZVFJIYEYQIHIP
|
8.2 | IC50 | 15 | — | |
CCZBGFFCFFPVJL
|
8.1 | IC50 | 4 | — | |
MPVZZUVYXJBYBN
|
8.1 | IC50 | 4 | — | |
AKDZNPFQMDRCMU
|
8.1 | IC50 | 7 | — | |
BGJDLKTYVVXXRM
|
8.1 | IC50 | 2 | — | |
CHFQZGSXRCZRIQ
|
8.1 | IC50 | 2 | — | |
IPAXTZAGMDYSHM
|
8.1 | IC50 | 2 | — | |
JDIAYVMOUUKPNK
|
8.1 | IC50 | 5 | — | |
JJUAVZQHRBSKOY
|
8.1 | Ki | 4 | — | |
PMIUHCUGSNZOBV
|
8.1 | IC50 | 2 | — | |
WNONTVPKTYRAIS
|
8.1 | IC50 | 2 | — | |
XTPCYXQQIXNDST
|
8.1 | IC50 | 2 | — | |
DWBVOWNYMAESQS
|
8.1 | IC50 | 4 | — | |
AEIHOULIOWEFLO
|
8.1 | Ki | 5 | — | |
ANZDEYYSOIFTCU
|
8.1 | Ki | 8 | — | |
DIHQGMJAKVBZHN
|
8.1 | Ki | 6 | — | |
GAFYDJGFHJBXQQ
|
8.1 | Ki | 9 | — | |
GLYHKPNATCXTDU
|
8.1 | IC50 | 5 | — | |
GUFBYMCWKSZUBS
|
8.1 | Ki | 8 | — | |
GZDFPDSMIHMTRU
|
8.1 | Ki | 6 | — | |
HFDKKSOKCNZLGJ
|
8.1 | IC50 | 2 | — | |
JCQSAYNTEFQHGH
|
8.1 | IC50 | 5 | — | |
JDCMEKBYCLWBEK
|
8.1 | IC50 | 2 | — | |
KZKOIZXRAQJRPY
|
8.1 | Ki | 5 | — |