Target Details
| UniProt AC | P50750 |
|---|---|
| Gene Symbol | CDK9 |
| Protein Name | Cyclin-dependent kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 3,102
- Clinical molecules 43
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (3,102)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PIMQWRZWLQKKBJ
|
8.4 | IC50 | 4 | — | |
PIMQWRZWLQKKBJ
|
8.4 | IC50 | 36 | — | |
POHPLECFWMXLII
|
8.4 | IC50 | 2 | — | |
PUBSTGHGWFWUTL
|
8.4 | Ki | 4 | — | |
RUFKAIQMVPWHCQ
|
8.4 | IC50 | 4 | — | |
RVZJFCNYSSUDCU
|
8.4 | IC50 | 7 | — | |
RVZJFCNYSSUDCU
|
8.4 | Kd | 2 | — | |
UPQKBKLECVIXJR
|
8.4 | IC50 | 12 | — | |
XRANJRXEZLWYJP
|
8.4 | IC50 | 2 | — | |
YKCGAMRTHVAZHZ
|
8.4 | IC50 | 4 | — | |
YZCUMZWULWOUMD
|
8.4 | IC50 | 2 | — | |
YZRRSIPTHDIILM
|
8.4 | Ki | 9 | — | |
HUKJRDDXELSRFT
|
8.4 | IC50 | 4 | — | |
WECKVHKRXUSKCN
|
8.4 | IC50 | 2 | — | |
DFPJSLJLOKWVCD
|
8.4 | IC50 | 6 | — | |
IQNFHQLDSXSHGX
|
8.4 | IC50 | 4 | — | |
IUMDSEQXNBJVCE
|
8.4 | IC50 | 4 | — | |
NZJQEKXXVRBRKU
|
8.4 | IC50 | 2 | — | |
QEYANDLEJXFZFA
|
8.4 | IC50 | 2 | — | |
MPLSNQAHULTSPR
|
8.4 | Ki | 5 | — | |
YKEMTVGDNWRGJT
|
8.4 | Ki | 5 | — | |
FNCMAUYJEUVBTB
|
8.4 | IC50 | 2 | — | |
GZHOQLMULXEMDB
|
8.4 | IC50 | 2 | — | |
IFAKQBBVXIIUEC
|
8.4 | IC50 | 3 | — | |
IAPISFUJUUDVNW
|
8.3 | IC50 | 15 | — | |
JJEJNNOEHSRLAW
|
8.3 | IC50 | 2 | — | |
NYJBTSYJXIHYOP
|
8.3 | IC50 | 2 | — | |
TWVJVNNYNNBYED
|
8.3 | Ki | 5 | — | |
ZVYXVPZGGHYOJL
|
8.3 | IC50 | 2 | — | |
GCZXMBAUDPVPSA
|
8.3 | IC50 | 6 | — | |
JRYOXRWZTSUWMQ
|
8.3 | IC50 | 4 | — | |
UQDHAMQNTWHVFF
|
8.3 | IC50 | 2 | — | |
BNVGYGOBIHDVET
|
8.3 | IC50 | 4 | — | |
BWONSNVPSAEXDY
|
8.3 | Ki | 9 | — | |
CBARNMHMGRVVLO
|
8.3 | IC50 | 11 | — | |
CELCCCWTAADGDV
|
8.3 | IC50 | 15 | — | |
CSIAVORBNYKYNX
|
8.3 | Ki | 4 | — | |
FMOZXIOQQZEZNP
|
8.3 | IC50 | 4 | — | |
HMCJMBDXHYZRRL
|
8.3 | Ki | 9 | — | |
HOYRWTWZUFFACV
|
8.3 | Ki | 28 | — | |
JRNXAQINDCOHGS
|
8.3 | IC50 | 13 | — | |
JRNXAQINDCOHGS
|
8.3 | IC50 | 15 | — | |
KMRJEIFKFAGWAW
|
8.3 | IC50 | 2 | — | |
LVJZZDNNQXAXPX
|
8.3 | Ki | 7 | — | |
MJIALGDLOLWBRQ
|
8.3 | IC50 | 12 | — | |
MLTGOCWSTUBXGD
|
8.3 | IC50 | 2 | — | |
QSFLJKWUAIYKRN
|
8.3 | IC50 | 3 | — | |
SLKCVFPEQGHNSI
|
8.3 | Ki | 29 | — | |
TYSWNLQZLBRNSE
|
8.3 | IC50 | 15 | — | |
UELYDGOOJPRWGF
|
8.3 | IC50 | 13 | — |