Target Details
| UniProt AC | P50750 |
|---|---|
| Gene Symbol | CDK9 |
| Protein Name | Cyclin-dependent kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 3,102
- Clinical molecules 43
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (3,102)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QZUWGDSAAXXRKW
|
8.5 | Ki | 2 | — | |
RSWRXLOFPCNDID
|
8.5 | IC50 | 2 | — | |
VZRBGAXSPYVRRB
|
8.5 | IC50 | 4 | — | |
YOJWDXJAIHIGAD
|
8.5 | Ki | 2 | — | |
CWZFOZMXEIEENA
|
8.5 | IC50 | 2 | — | |
FRUDYEUOYPWKKU
|
8.5 | IC50 | 5 | — | |
IBHADHHDWIADDZ
|
8.5 | IC50 | 2 | — | |
WDXRGXOFKKTSHX
|
8.5 | IC50 | 4 | — | |
DBOXIXXMMCQDIQ
|
8.5 | IC50 | 2 | — | |
FCJBTZIGPFCDBX
|
8.5 | IC50 | 2 | — | |
IECCMARSLUQALN
|
8.5 | IC50 | 4 | — | |
PGJSFHVYYFKSRH
|
8.5 | IC50 | 4 | — | |
RUSDDQSVRZWWRP
|
8.5 | IC50 | 4 | — | |
FHPOPNDOFQGPBB
|
8.5 | IC50 | 2 | — | |
HFCLVEWUMOPUHL
|
8.5 | IC50 | 2 | — | |
UYWLJKDPGSPEFI
|
8.5 | IC50 | 2 | — | |
YZCUMZWULWOUMD
|
8.5 | IC50 | 4 | — | |
CLHZKZYRISNUNI
|
8.4 | IC50 | 4 | — | |
FDDRHWAVGSBKFR
|
8.4 | IC50 | 2 | — | |
MWYWPRFDCPIKNI
|
8.4 | IC50 | 2 | — | |
SNEZQLJYUBSJBP
|
8.4 | IC50 | 2 | — | |
XWQVQSXLXAXOPJ
|
8.4 | IC50 | 7 | — | |
HQVRFXBZJOXOKH
|
8.4 | IC50 | 2 | — | |
KWDKPWGMOHUDFP
|
8.4 | IC50 | 2 | — | |
WNONTVPKTYRAIS
|
8.4 | IC50 | 2 | — | |
XNCHAOOIMXRRBN
|
8.4 | IC50 | 2 | — | |
XTPCYXQQIXNDST
|
8.4 | IC50 | 2 | — | |
YAAYHLMEILEMJC
|
8.4 | IC50 | 2 | — | |
ZMFLCQAMPNGORA
|
8.4 | IC50 | 6 | — | |
HYPSIGLBLBWTCY
|
8.4 | IC50 | 2 | — | |
QIIDDOABFUKHBM
|
8.4 | IC50 | 6 | — | |
GKXBSZQJUPTJLA
|
8.4 | IC50 | 2 | — | |
XMDAGFVARVIRGW
|
8.4 | IC50 | 4 | — | |
ACSYKUPGCXYRRO
|
8.4 | Ki | 26 | — | |
AIOFXERAXQYANK
|
8.4 | IC50 | 9 | — | |
BYUAPXZEZUYLJI
|
8.4 | IC50 | 4 | — | |
CKIFWVSQRJHDKI
|
8.4 | Ki | 9 | — | |
DDDXJQXLEOFIHJ
|
8.4 | IC50 | 6 | — | |
DORFHNBANBXCGZ
|
8.4 | IC50 | 5 | — | |
DYTKVFHLKPDNRW
|
8.4 | Ki | 23 | Yes | |
DZKMAWNYSJECKX
|
8.4 | IC50 | 12 | — | |
GAIOPWBQKZMUNO
|
8.4 | Ki | 13 | — | |
HQVUAGCBAZOMFE
|
8.4 | IC50 | 2 | — | |
KCKWQKDFLCMFNR
|
8.4 | IC50 | 4 | — | |
LEOFXMFOPINZOR
|
8.4 | IC50 | 2 | — | |
LHEDETRRIJTKNJ
|
8.4 | IC50 | 2 | — | |
LPILBMJJRGTKOQ
|
8.4 | Ki | 27 | — | |
NDLAFOKSJSLKGG
|
8.4 | IC50 | 4 | — | |
OCBFHTQGXPIABP
|
8.4 | IC50 | 3 | — | |
ODRITQGYYWHQGM
|
8.4 | IC50 | 4 | — |