Target Details
| UniProt AC | P50750 |
|---|---|
| Gene Symbol | CDK9 |
| Protein Name | Cyclin-dependent kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 3,102
- Clinical molecules 43
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (3,102)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UAFDMWGGQQODTL
|
8.6 | Ki | 9 | — | |
UQTQEXQMIZMPDV
|
8.6 | IC50 | 2 | — | |
WOKVPTJFHFDZLP
|
8.6 | IC50 | 2 | — | |
GXDOEZRSIKWODV
|
8.6 | IC50 | 4 | — | |
CUVHRQJIXRDVGG
|
8.6 | IC50 | 4 | — | |
DEQKSXYLYYLTSY
|
8.6 | IC50 | 2 | — | |
GFAOBTBGGGZDLI
|
8.6 | IC50 | 2 | — | |
KJJKRKBRHLAFOG
|
8.6 | IC50 | 2 | — | |
MADUTGUALSLNOW
|
8.6 | IC50 | 4 | — | |
MSSWEISDYNQLGE
|
8.6 | IC50 | 4 | — | |
NLXGWLYKUXHWNP
|
8.6 | IC50 | 2 | — | |
GYGIXVNDVQQAPJ
|
8.5 | IC50 | 4 | — | |
LZVICBFRAOBQGQ
|
8.5 | IC50 | 4 | — | |
NJJPIXGNLMGEOV
|
8.5 | IC50 | 6 | — | |
LXQRFMWTQCXDPP
|
8.5 | IC50 | 4 | — | |
WIDAZACOEGHADI
|
8.5 | IC50 | 6 | — | |
YGXSGRGRLJSQDK
|
8.5 | IC50 | 4 | — | |
ACLSGVFCTLWIGY
|
8.5 | IC50 | 4 | — | |
AKVXZHCGYWIYJU
|
8.5 | IC50 | 2 | — | |
AMMBWNGMXHWBAS
|
8.5 | IC50 | 2 | — | |
AQLRQVRNKVAOOW
|
8.5 | IC50 | 2 | — | |
BQLLLVDIZXOQJD
|
8.5 | Ki | 8 | — | |
BRMDAMYZBOCCKU
|
8.5 | IC50 | 2 | — | |
CDKRFBBXZQUTDX
|
8.5 | Ki | 9 | — | |
CGBFAYLLULJFBW
|
8.5 | Ki | 8 | — | |
CODOEMQMKTTYRW
|
8.5 | IC50 | 7 | — | |
CUCBJZSGNZBKEE
|
8.5 | IC50 | 2 | — | |
FPHITTVVVWKENE
|
8.5 | Ki | 9 | — | |
HXZXJLLRGFULES
|
8.5 | Ki | 9 | — | |
LQKBDFWBLIOIGB
|
8.5 | IC50 | 2 | — | |
LWOIOAVZAUIQIB
|
8.5 | IC50 | 4 | — | |
NFTJDXGFOUFNKG
|
8.5 | IC50 | 16 | — | |
PEFQLFPPRNGLJD
|
8.5 | IC50 | 2 | — | |
XCIGDMLFQKYLKU
|
8.5 | Ki | 4 | — | |
XXPDEKKKGHCODA
|
8.5 | IC50 | 2 | — | |
YARIHEYYGBAEDE
|
8.5 | Ki | 10 | — | |
YZCUMZWULWOUMD
|
8.5 | IC50 | 2 | — | |
ZNYWIWXWOHYBON
|
8.5 | IC50 | 2 | — | |
BIKJIRVRDFVXQG
|
8.5 | IC50 | 6 | — | |
CRZXYCJOVDIWGP
|
8.5 | IC50 | 4 | — | |
DPLUHOORPHUMHS
|
8.5 | IC50 | 4 | — | |
GYFJDZVSZGIZDZ
|
8.5 | IC50 | 2 | — | |
KVXSQZZAGHGMFE
|
8.5 | IC50 | 4 | — | |
SWQLIIAAXLKOKM
|
8.5 | IC50 | 2 | — | |
BGYVWFZMYBWCNY
|
8.5 | Ki | 30 | — | |
DUPJERCDKVJCCS
|
8.5 | IC50 | 2 | — | |
WAFHXBBZJZYUIJ
|
8.5 | IC50 | 7 | — | |
ZGGIYFOLDBTZIL
|
8.5 | Ki | 27 | — | |
PFBMBYULIZGMBA
|
8.5 | IC50 | 4 | — | |
PSHJABZCSORYCH
|
8.5 | Ki | 2 | — |