Target Details
| UniProt AC | P50750 |
|---|---|
| Gene Symbol | CDK9 |
| Protein Name | Cyclin-dependent kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 3,102
- Clinical molecules 43
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (3,102)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NFTJDXGFOUFNKG
|
8.7 | IC50 | 4 | — | |
WUIYYLQXGFFWTL
|
8.7 | IC50 | 2 | — | |
XJKTXWSMMWPNTP
|
8.7 | IC50 | 6 | — | |
XSDZPPRQLIZLDG
|
8.7 | IC50 | 6 | — | |
YGZQAQIWZFMADC
|
8.7 | IC50 | 12 | — | |
YPAQXRURXUKFGB
|
8.7 | IC50 | 4 | — | |
ZDQGFSXRMBIKKI
|
8.7 | IC50 | 4 | — | |
ZLHUAMTYKCRXDR
|
8.7 | Ki | 8 | — | |
ZMZIPHROZUBATK
|
8.7 | IC50 | 2 | — | |
FPZYYCPZIIPVNT
|
8.7 | IC50 | 4 | — | |
GBTFAVMORZGOBX
|
8.7 | IC50 | 4 | — | |
HASNZZTVQOLZGN
|
8.7 | IC50 | 2 | — | |
NACHSLSMZHMOQM
|
8.7 | IC50 | 2 | — | |
QFKHYTSJLGIBEQ
|
8.7 | IC50 | 4 | — | |
XQNOWBKVNDCBHZ
|
8.7 | IC50 | 4 | — | |
ZMTFZGPLNVXQCA
|
8.7 | IC50 | 2 | — | |
JMJVJBLTWBOIBV
|
8.7 | IC50 | 2 | — | |
PCVRDGSBSHXSIV
|
8.7 | IC50 | 4 | — | |
QPLPUYOXFJFKJQ
|
8.7 | IC50 | 2 | — | |
ZBQZKMUITVYTBN
|
8.7 | IC50 | 4 | — | |
QTLSVBHPZACPBO
|
8.7 | IC50 | 2 | — | |
VQDUCLMICBTOLT
|
8.7 | IC50 | 4 | — | |
HXOTVSDBXJSUKD
|
8.6 | IC50 | 4 | — | |
IKEGLJUOFSRILW
|
8.6 | IC50 | 2 | — | |
LZTILAJWCMPABA
|
8.6 | IC50 | 4 | — | |
MRMIZTRXAITUEN
|
8.6 | IC50 | 2 | — | |
RDOKVGWGKMHBMG
|
8.6 | IC50 | 9 | — | |
UQZLGOVFSDEYQJ
|
8.6 | IC50 | 6 | — | |
VGKOYNIMZVZLAN
|
8.6 | IC50 | 6 | — | |
ZGMXUKBNYJKTLV
|
8.6 | IC50 | 4 | — | |
OHNWBGGGJMOKIX
|
8.6 | IC50 | 4 | — | |
QTHCAAFKVUWAFI
|
8.6 | IC50 | 23 | — | |
HCWVCCMKEVZHLU
|
8.6 | IC50 | 6 | — | |
LWHMSHBMCRYSON
|
8.6 | IC50 | 2 | — | |
SSIOYGMEKCPFAV
|
8.6 | IC50 | 5 | — | |
VXBAJLGYBMTJCY
|
8.6 | IC50 | 34 | Yes | |
WJDGUKDMQOOHQB
|
8.6 | IC50 | 2 | — | |
XMQUZQUEHXAOEE
|
8.6 | IC50 | 2 | — | |
XRMXIRZGNIFUDY
|
8.6 | IC50 | 2 | — | |
CNQGNADBGYCKKV
|
8.6 | Ki | 25 | — | |
COXHFPQLBUVXLI
|
8.6 | IC50 | 2 | — | |
GNHNRVSQWNAGHC
|
8.6 | IC50 | 7 | Yes | |
JJGYTERWQYNFJU
|
8.6 | IC50 | 4 | — | |
VHAJTIDXIDFCMN
|
8.6 | IC50 | 4 | — | |
ZKLJKKASNXVQBZ
|
8.6 | Ki | 27 | — | |
DWJMXSDTTGHUTQ
|
8.6 | IC50 | 2 | — | |
LNYNSZZKFBTQRV
|
8.6 | IC50 | 2 | — | |
NOBXXQPXRRDJOJ
|
8.6 | IC50 | 6 | — | |
RIGDRWMDXNFWPV
|
8.6 | IC50 | 4 | — | |
YKSDGHNGKNMUGI
|
8.6 | IC50 | 12 | — |