Target Details
| UniProt AC | P50750 |
|---|---|
| Gene Symbol | CDK9 |
| Protein Name | Cyclin-dependent kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 3,102
- Clinical molecules 43
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (3,102)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UVSZGHBPMOAFSS
|
8.9 | IC50 | 6 | — | |
VRHHAMWTRSVIEX
|
8.9 | Kd | 5 | — | |
AWVIEXQGKHJISX
|
8.9 | IC50 | 4 | — | |
PYTROLIEIDFMKB
|
8.9 | IC50 | 4 | — | |
VQAQEQWKWBXYBD
|
8.9 | IC50 | 4 | — | |
CWGBJAZDOLEZBX
|
8.8 | IC50 | 4 | — | |
DQBASRYERZQRJJ
|
8.8 | IC50 | 15 | — | |
RVKNONNXSNALJV
|
8.8 | IC50 | 21 | — | |
VUKIOSRRSWOLGW
|
8.8 | IC50 | 4 | — | |
MIXKIGRNSRMTFM
|
8.8 | IC50 | 6 | — | |
WZBMGNIWAIVYPC
|
8.8 | IC50 | 4 | — | |
JMQICEYHFZDQRQ
|
8.8 | IC50 | 4 | — | |
LHXPKQBNRWZDLD
|
8.8 | IC50 | 4 | — | |
UOSJCNTXEITJHM
|
8.8 | IC50 | 4 | — | |
ADZXDTAAQTYSRZ
|
8.8 | IC50 | 2 | — | |
CPHBFPSTJMYONO
|
8.8 | IC50 | 4 | — | |
HOARYCLJOWBNCE
|
8.8 | IC50 | 4 | — | |
JSHQBITYFQKJER
|
8.8 | IC50 | 2 | — | |
FCWZPEHBEGYARS
|
8.8 | IC50 | 6 | — | |
WLTRIWCDHOZNRP
|
8.8 | Ki | 14 | — | |
XCGKNNRKGHJIBF
|
8.8 | IC50 | 4 | — | |
MRPGRAKIAJJGMM
|
8.8 | IC50 | 11 | — | |
PYICIQOHSCQPIT
|
8.8 | IC50 | 4 | — | |
HTFBNTYFTGIOEK
|
8.8 | IC50 | 7 | — | |
HEAXYWPCYLENAR
|
8.7 | IC50 | 4 | — | |
OXSBHNFOHBJSEQ
|
8.7 | IC50 | 4 | — | |
ZBQZKMUITVYTBN
|
8.7 | IC50 | 4 | — | |
ITSPBRBMIPVDCF
|
8.7 | Ki | 5 | — | |
LMIPCDJYZXYYLQ
|
8.7 | IC50 | 5 | — | |
NBSJZWFDNFWQDN
|
8.7 | IC50 | 29 | — | |
WMUYOUUBRWWBTA
|
8.7 | IC50 | 2 | — | |
CEERPSVTLJOQDZ
|
8.7 | IC50 | 4 | — | |
IKRBTPMIGDQTPT
|
8.7 | IC50 | 4 | — | |
MSZSKQDTQOXXHU
|
8.7 | IC50 | 2 | — | |
AJXDBLPSUPQKBJ
|
8.7 | IC50 | 2 | — | |
AXAQVNRYNMCZCK
|
8.7 | Ki | 10 | Yes | |
BDRPEEVXRRASAS
|
8.7 | IC50 | 2 | — | |
BFSKFHZFACZLER
|
8.7 | IC50 | 2 | — | |
BQRWVMGYVBRTGW
|
8.7 | IC50 | 2 | — | |
BRBJCJHJBAMBPR
|
8.7 | IC50 | 12 | — | |
BXMBIVXDTXURDF
|
8.7 | Ki | 9 | — | |
CXMKIWPGGSLHRE
|
8.7 | IC50 | 15 | — | |
DAXGPJQWYKFPPW
|
8.7 | IC50 | 4 | — | |
DKGCKUUOPCFNNH
|
8.7 | IC50 | 2 | — | |
IUBQEKUBWGFDHC
|
8.7 | IC50 | 4 | — | |
KHGPYYFCIAISBU
|
8.7 | Ki | 31 | — | |
LAMSOXVNXMIZHG
|
8.7 | IC50 | 2 | — | |
LRXZVWVFJCSXSV
|
8.7 | IC50 | 2 | — | |
LYJYFPJCEDSGHY
|
8.7 | IC50 | 2 | — | |
MDOPSPOMDXUNGM
|
8.7 | IC50 | 2 | — |