Target Details
| UniProt AC | P50750 |
|---|---|
| Gene Symbol | CDK9 |
| Protein Name | Cyclin-dependent kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 3,102
- Clinical molecules 43
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (3,102)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DFVQRLLERQLHSP
|
7.7 | IC50 | 2 | — | |
DQKKUVSYKRLEBM
|
7.7 | IC50 | 10 | — | |
FLIVKVQMXOAQAK
|
7.7 | IC50 | 15 | — | |
GCVSAIBJMFPDAT
|
7.7 | IC50 | 2 | — | |
GNWQPICFCPORII
|
7.7 | IC50 | 5 | — | |
HVERIWOPBLJMDS
|
7.7 | IC50 | 2 | — | |
LQHMJVOJVOLFTJ
|
7.7 | IC50 | 7 | — | |
LYXGMLBMSIISDR
|
7.7 | IC50 | 2 | — | |
MBBABMWLFCFNPV
|
7.7 | IC50 | 2 | — | |
MBWPOBKGEBIBOJ
|
7.7 | IC50 | 2 | — | |
ONZJVSHWCHMBKN
|
7.7 | IC50 | 2 | — | |
PUXKEKPYASIYGT
|
7.7 | IC50 | 7 | — | |
QWDSCEPBJKQNGL
|
7.7 | IC50 | 2 | — | |
RHWIDIZNQRAAIU
|
7.7 | IC50 | 7 | — | |
RIUQJGVJWYACAJ
|
7.7 | IC50 | 2 | — | |
RWJDKWGWJJVDJB
|
7.7 | IC50 | 2 | — | |
SDKUHAJXRKLBEV
|
7.7 | IC50 | 2 | — | |
UNVIDDLDPDEJMZ
|
7.7 | IC50 | 2 | — | |
VCGZLNSADOXLAT
|
7.7 | Ki | 4 | — | |
VCPRPKASMPDNQA
|
7.7 | IC50 | 2 | — | |
VSIAIRQSYURWTI
|
7.7 | IC50 | 2 | — | |
WITIUJMWBTVWES
|
7.7 | IC50 | 2 | — | |
YQPUVDJEBYVXDE
|
7.7 | IC50 | 2 | — | |
ZFEUWTMEXIDLMB
|
7.7 | IC50 | 2 | — | |
ZNNREQBGMVPIDK
|
7.7 | IC50 | 2 | — | |
ZPUBPIPZFAUDSS
|
7.7 | IC50 | 2 | — | |
XDPKOVYWCYQSBM
|
7.7 | IC50 | 2 | — | |
AUNVIXGOAIFEQQ
|
7.7 | IC50 | 2 | — | |
AWYBHCVXZFMJHV
|
7.7 | IC50 | 5 | — | |
AYCKASQUVBKOMD
|
7.7 | IC50 | 3 | — | |
GIYOAWSOVWBBGQ
|
7.7 | IC50 | 2 | — | |
GJHHGLCAFGSVNF
|
7.7 | IC50 | 4 | — | |
HJVQEPUKVZEVTN
|
7.7 | IC50 | 2 | — | |
IQMPZJYDZWUWHT
|
7.7 | IC50 | 2 | — | |
JAGSBTCNHPBZIM
|
7.7 | IC50 | 2 | — | |
JZVAAEYRYPYICS
|
7.7 | IC50 | 2 | — | |
MFMGZBUGOSVXOS
|
7.7 | IC50 | 2 | — | |
MRWKUIOLQRITLV
|
7.7 | IC50 | 3 | — | |
NDQRCUOYOAPFLR
|
7.7 | IC50 | 2 | — | |
OSVJXWVRTPXQBX
|
7.7 | IC50 | 2 | — | |
OYLVPRAOMPFNAP
|
7.7 | IC50 | 2 | — | |
OZWHCAZDQNMMES
|
7.7 | IC50 | 2 | — | |
QTROMHAUINAJRE
|
7.7 | IC50 | 2 | — | |
RAFISFVOOKCYLW
|
7.7 | IC50 | 6 | — | |
SBOSVLRBKPEZMQ
|
7.7 | IC50 | 3 | — | |
SLBMMPZICNYISW
|
7.7 | IC50 | 2 | — | |
SSEDQERECATUBR
|
7.7 | Ki | 5 | — | |
SSMMYRQDZBSVCY
|
7.7 | IC50 | 7 | Yes | |
VDKLUQBZRIEHKE
|
7.7 | IC50 | 2 | — | |
XLAXFWRJQFAVQC
|
7.7 | IC50 | 2 | — |