Target Details
| UniProt AC | P50750 |
|---|---|
| Gene Symbol | CDK9 |
| Protein Name | Cyclin-dependent kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 3,102
- Clinical molecules 43
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (3,102)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UXEWCQUEOJJYLF
|
7.9 | IC50 | 6 | — | |
WZYMEKZRUAABBC
|
7.9 | IC50 | 2 | — | |
JRDXBFKOJWSWAB
|
7.9 | IC50 | 2 | — | |
XOTQSFMYDHXIOI
|
7.9 | IC50 | 2 | — | |
ZWWTZNLYKPWLQS
|
7.9 | IC50 | 2 | — | |
NNMRZPOMVQNXMS
|
7.9 | Ki | 8 | — | |
PBDNNWWYSHCMCH
|
7.9 | IC50 | 7 | — | |
CJABJKHMLIRNNF
|
7.9 | IC50 | 2 | — | |
LNSQQXAMSPLGOU
|
7.9 | IC50 | 2 | — | |
RXLKGKJSOZFSEN
|
7.9 | IC50 | 2 | — | |
ABAHFFAFDXIWSH
|
7.8 | IC50 | 2 | — | |
AFYLTDZJAWPVBM
|
7.8 | Ki | 8 | — | |
BHDZLFHFYYIDMB
|
7.8 | IC50 | 2 | — | |
CQLFRGIYOHYSJV
|
7.8 | IC50 | 7 | — | |
CWBNKHNBBDYRLV
|
7.8 | IC50 | 2 | — | |
GVUHDEMSKMOPHW
|
7.8 | IC50 | 9 | — | |
GZEWMDYKYJQWHT
|
7.8 | IC50 | 2 | — | |
HAOOVLDCSQZODX
|
7.8 | Ki | 8 | — | |
HATMRDUPPAWOII
|
7.8 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.8 | IC50 | 408 | — | |
JPLLQSBSTHWUIK
|
7.8 | IC50 | 7 | — | |
LRUBSVFNLJTGJA
|
7.8 | IC50 | 2 | — | |
MQWRXIFGIPESEO
|
7.8 | IC50 | 2 | — | |
NJCLIBSGAOCZBH
|
7.8 | IC50 | 2 | — | |
OVSXVWXYBBOHGF
|
7.8 | IC50 | 2 | — | |
PBDNNWWYSHCMCH
|
7.8 | IC50 | 7 | — | |
POSUMUOPXKYTPR
|
7.8 | IC50 | 2 | — | |
WKDOKJKUKSSFSB
|
7.8 | IC50 | 2 | — | |
WLIJQAGXRURARW
|
7.8 | IC50 | 6 | — | |
WQCXLUNOPQPYFK
|
7.8 | IC50 | 3 | — | |
WQZVTNFUNLTGDW
|
7.8 | Ki | 4 | — | |
WUXSDCABLMGOMN
|
7.8 | IC50 | 2 | — | |
XYSDSNJAODYESD
|
7.8 | IC50 | 2 | — | |
YRNFLVUMZIRYKY
|
7.8 | IC50 | 2 | — | |
BRYMZSSAIDEFEM
|
7.8 | IC50 | 4 | — | |
OAAHCIALZYFQLH
|
7.8 | IC50 | 2 | — | |
WXRXZJOVLMBRSB
|
7.8 | IC50 | 2 | — | |
AIYUXSKIUKFZIR
|
7.8 | IC50 | 2 | — | |
FPBKUBUKBWJEMH
|
7.8 | IC50 | 7 | — | |
ROMAHJZEHBXJSU
|
7.8 | IC50 | 7 | — | |
BLUORUUGUNHQIW
|
7.8 | IC50 | 2 | — | |
BLUORUUGUNHQIW
|
7.8 | IC50 | 2 | — | |
FIOUSIQCBJHCSJ
|
7.8 | IC50 | 2 | — | |
GSRHVOVIIWBRTN
|
7.8 | IC50 | 5 | — | |
IYJUXBLZDNMMKD
|
7.8 | IC50 | 2 | — | |
JCWDLMMDEICJNN
|
7.8 | IC50 | 2 | — | |
JRNJNYBQQYBCLE
|
7.8 | Kd | 40 | Yes | |
JYXQKMTVNRMKPN
|
7.8 | Ki | 6 | — | |
KOFUCJJVAIILNY
|
7.8 | IC50 | 2 | — | |
NWFSYTHPSDOPRY
|
7.8 | IC50 | 2 | — |