Target Details
| UniProt AC | P50750 |
|---|---|
| Gene Symbol | CDK9 |
| Protein Name | Cyclin-dependent kinase 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 3,102
- Clinical molecules 43
- Avg pChEMBL 7.25
KEGG Pathways (2)
Active Molecules (3,102)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BFQBIVCJNIEQPK
|
9.5 | Ki | 5 | — | |
XWXGKRQCUJICNZ
|
9.4 | IC50 | 2 | — | |
HRLKJDPJDKEXFB
|
9.4 | IC50 | 4 | — | |
FBBATKKBOQLQKG
|
9.4 | IC50 | 6 | — | |
FCDMIMACOWLETE
|
9.3 | IC50 | 6 | — | |
XUDPANPGIPSBJA
|
9.3 | IC50 | 6 | — | |
ZKDRQTUQLALDNJ
|
9.3 | IC50 | 4 | — | |
VHBMYACYAMWWOX
|
9.3 | IC50 | 6 | — | |
NMLSMKNXYWXSKI
|
9.3 | IC50 | 3 | — | |
WWNMRNZJYNHSAR
|
9.3 | IC50 | 6 | — | |
SVGQRDCSVDIDOX
|
9.3 | IC50 | 6 | — | |
ZQYCLRJPFSGBEH
|
9.3 | IC50 | 6 | — | |
BIIVYFLTOXDAOV
|
9.2 | Ki | 31 | — | |
KUIAPCBDLHKMCV
|
9.2 | IC50 | 6 | — | |
YQOZIILPTSEVFV
|
9.2 | IC50 | 6 | — | |
HDSMDAXOECRDBG
|
9.2 | IC50 | 4 | — | |
QCAKOASCPYIZKI
|
9.1 | IC50 | 4 | — | |
NYQSSFSDFGEMQF
|
9.1 | IC50 | 6 | — | |
KBJYBBVTVRWYJU
|
9.1 | IC50 | 4 | — | |
PIMQWRZWLQKKBJ
|
9.1 | Ki | 5 | — | |
XUOBMFPQIZTUAZ
|
9.1 | IC50 | 6 | — | |
IALMJWAVHXWMPQ
|
9.1 | IC50 | 4 | — | |
CIVWJLUNRPRKCE
|
9.1 | IC50 | 6 | — | |
MREGZYIBCQDRSY
|
9.1 | IC50 | 4 | — | |
SOHOEERULHWXJB
|
9.0 | IC50 | 5 | — | |
OVONSEUUMQWSJD
|
9.0 | IC50 | 4 | — | |
BMXNNFIAYWHIGH
|
9.0 | IC50 | 4 | — | |
XUKYEEYMPUGKNF
|
9.0 | Ki | 4 | — | |
AYRYUMQKDYQBAS
|
9.0 | IC50 | 4 | — | |
OKLIXNGBJODOLI
|
9.0 | IC50 | 6 | — | |
SWKHRTIXNUHZMW
|
9.0 | IC50 | 4 | — | |
AULDUFVLZQNYJD
|
9.0 | IC50 | 2 | — | |
BKCOGSHTNWTZNI
|
9.0 | IC50 | 15 | — | |
CIKHZDKMTDPCLM
|
9.0 | IC50 | 2 | — | |
DTTGEKGDXFLMIL
|
9.0 | IC50 | 4 | — | |
FPPDWTSDSZADQO
|
9.0 | IC50 | 2 | — | |
OETJRQWLHMSDMD
|
9.0 | IC50 | 2 | — | |
VKFHEWRJQKNNFM
|
9.0 | IC50 | 6 | — | |
XLSYZSRXVVCHLS
|
9.0 | IC50 | 48 | — | |
IKKCTHIIEQFHBF
|
9.0 | IC50 | 4 | — | |
URJVQQWWUXRWLM
|
9.0 | IC50 | 6 | — | |
CBMDGSCTUBJWIN
|
9.0 | IC50 | 4 | — | |
FBECJLNJBCQUNR
|
9.0 | IC50 | 4 | — | |
HGTWFXKVZMIFQK
|
9.0 | IC50 | 2 | — | |
XQVDBOSCUDRTCQ
|
9.0 | IC50 | 4 | — | |
DJJBKVQCCJJIJG
|
8.9 | IC50 | 2 | — | |
FENPXPBUKNHHHM
|
8.9 | IC50 | 4 | — | |
FUMCKNCUEAQHCV
|
8.9 | Ki | 103 | — | |
OTPFZAVDWPCJLJ
|
8.9 | Ki | 9 | — | |
NMHGCPUMMGKNKO
|
8.9 | IC50 | 4 | — |