Target Details
| UniProt AC | P50613 |
|---|---|
| Gene Symbol | CDK7 |
| Protein Name | Cyclin-dependent kinase 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,007
- Clinical molecules 36
- Avg pChEMBL 6.99
KEGG Pathways (3)
Active Molecules (1,007)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SCJNYBYSTCRPAO
|
7.1 | IC50 | 7 | — | |
IFAKQBBVXIIUEC
|
7.1 | IC50 | 3 | — | |
KJHOORCYJSBANN
|
7.1 | IC50 | 15 | — | |
MJIALGDLOLWBRQ
|
7.1 | IC50 | 12 | — | |
UPQKBKLECVIXJR
|
7.1 | IC50 | 12 | — | |
BWRIYUPYJGGSDC
|
7.1 | IC50 | 2 | — | |
DSHAIQLEQCKJIR
|
7.1 | IC50 | 7 | — | |
PSSXVHVJRWQMQR
|
7.1 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
7.1 | Kd | 289 | Yes | |
DIHQGMJAKVBZHN
|
7.0 | Ki | 6 | — | |
IPGGHZCVPFPELS
|
7.0 | IC50 | 3 | — | |
SBNVUFMJQUOIKN
|
7.0 | IC50 | 9 | — | |
BFQBIVCJNIEQPK
|
7.0 | Ki | 5 | — | |
BGPUFSMDGGQOIE
|
7.0 | Ki | 9 | — | |
BKOYUSKBPMSUBK
|
7.0 | IC50 | 9 | — | |
GAIOPWBQKZMUNO
|
7.0 | Ki | 13 | — | |
SWAMHZPWHCCEDV
|
7.0 | IC50 | 2 | — | |
DPEBAAUPCCEJDT
|
7.0 | IC50 | 6 | — | |
NBHWQTWPQQUECJ
|
7.0 | IC50 | 2 | — | |
PHVGAEJTLZFYTO
|
7.0 | IC50 | 11 | — | |
QVGZEIMXBRBINE
|
7.0 | IC50 | 3 | — | |
DZKMAWNYSJECKX
|
7.0 | IC50 | 12 | — | |
GDZVTFLLGJNTRE
|
7.0 | IC50 | 11 | — | |
HUNWQLBOLVYRMW
|
7.0 | IC50 | 11 | — | |
JUTPXYDDNXBENH
|
7.0 | IC50 | 3 | — | |
NBSJZWFDNFWQDN
|
7.0 | IC50 | 29 | — | |
SPKWRLBKVPRPMT
|
7.0 | IC50 | 9 | — | |
BIIVYFLTOXDAOV
|
7.0 | Ki | 31 | — | |
HTFBNTYFTGIOEK
|
7.0 | IC50 | 7 | — | |
KAZJIBCOYQRDGG
|
7.0 | Ki | 16 | — | |
LNYCRXZEMSCWFG
|
7.0 | IC50 | 7 | — | |
MBIXOXMOHXFUFZ
|
7.0 | IC50 | 3 | — | |
QATMNAAQTUISJK
|
7.0 | Ki | 13 | — | |
QNUKRWAIZMBVCU
|
7.0 | Ki | 46 | — | |
RWKDVIAVTRRJIR
|
7.0 | Ki | 23 | — | |
RYYNGWLOYLRZLK
|
7.0 | Ki | 104 | — | |
SBFPHSVZEXSHTL
|
7.0 | Ki | 62 | — | |
SIGKFKBFXQQJJH
|
7.0 | IC50 | 7 | — | |
XNWKXXIGSPPPBH
|
7.0 | Ki | 31 | — | |
XUFLBSMTYMFOQH
|
7.0 | Ki | 43 | — | |
ZGGIYFOLDBTZIL
|
7.0 | Ki | 27 | — | |
ZOPGCNRZFZPRGB
|
7.0 | Ki | 9 | — | |
BIIVYFLTOXDAOV
|
7.0 | IC50 | 82 | Yes | |
JKKUZTDMJDZHEB
|
7.0 | IC50 | 7 | — | |
DSMBDRWDECFDNR
|
7.0 | IC50 | 7 | — | |
JFSGUSJACVSEKX
|
7.0 | IC50 | 7 | Yes | |
MOXBYMQBYZTOJA
|
7.0 | IC50 | 11 | — | |
AFFSZQATPPOYMW
|
7.0 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
7.0 | Kd | 64 | Yes | |
YKEMTVGDNWRGJT
|
7.0 | Ki | 5 | — |