Target Details
| UniProt AC | P50613 |
|---|---|
| Gene Symbol | CDK7 |
| Protein Name | Cyclin-dependent kinase 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,007
- Clinical molecules 36
- Avg pChEMBL 6.99
KEGG Pathways (3)
Active Molecules (1,007)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FELGDXDUEDTBOE
|
7.2 | IC50 | 3 | — | |
FSLNKEPUUKBMOR
|
7.2 | IC50 | 3 | — | |
GUKWPWBWSGIXJS
|
7.2 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
7.2 | Ki | 118 | — | |
HLJDDFGBLSZCEP
|
7.2 | IC50 | 3 | — | |
HSMUWLLZAZCLHF
|
7.2 | Ki | 25 | — | |
IWBAOIOMHDLFAY
|
7.2 | IC50 | 3 | — | |
JXTNBBXDHFAGLE
|
7.2 | IC50 | 3 | — | |
KDCKKNHYXJQMRS
|
7.2 | IC50 | 3 | — | |
KVOMOZYLJKQEDA
|
7.2 | IC50 | 3 | — | |
MXUFWRPGQWGALR
|
7.2 | IC50 | 3 | — | |
MXUFWRPGQWGALR
|
7.2 | IC50 | 3 | — | |
QBKUOOQFSVMDPB
|
7.2 | Ki | 31 | — | |
QRHXYRZCHFIWGD
|
7.2 | IC50 | 3 | — | |
RGOPHVZLEMGMBZ
|
7.2 | Ki | 20 | — | |
RMTHHMQLXQDQPP
|
7.2 | IC50 | 3 | — | |
SIGAKCXGEQAVJE
|
7.2 | IC50 | 3 | — | |
VVEGARMQKNYDID
|
7.2 | Ki | 24 | — | |
WEZUISMDDVGNCM
|
7.2 | IC50 | 3 | — | |
YZCXLBPFKGLDGS
|
7.2 | IC50 | 3 | — | |
ZFDZFQZUFROCDW
|
7.2 | IC50 | 3 | — | |
ZGNFJXHNIRUYHS
|
7.2 | IC50 | 3 | — | |
FPHITTVVVWKENE
|
7.2 | Ki | 9 | — | |
PDKCCNVCSBISEP
|
7.2 | IC50 | 3 | — | |
ARIOBGGRZJITQX
|
7.2 | IC50 | 24 | — | |
PBDNNWWYSHCMCH
|
7.2 | IC50 | 7 | — | |
TYSWNLQZLBRNSE
|
7.2 | IC50 | 15 | — | |
HMCJMBDXHYZRRL
|
7.2 | Ki | 9 | — | |
BPNUQXPIQBZCMR
|
7.2 | Kd | 83 | Yes | |
DYTKVFHLKPDNRW
|
7.2 | Ki | 23 | Yes | |
RSQPNXBTPUXMQN
|
7.2 | IC50 | 12 | — | |
HKSZLNNOFSGOKW
|
7.1 | IC50 | 408 | — | |
KNNCVZWOVBDOPR
|
7.1 | IC50 | 3 | — | |
LUWQTRGZKXLDSO
|
7.1 | IC50 | 11 | — | |
OEVYIGIAPVJKTQ
|
7.1 | IC50 | 2 | — | |
SDCFEWGPZJQLBA
|
7.1 | IC50 | 2 | — | |
YUXAEVQPKOFNAM
|
7.1 | IC50 | 3 | — | |
BTDWTDGMTNRFHC
|
7.1 | IC50 | 10 | — | |
DJMZUWUEYULGRB
|
7.1 | IC50 | 2 | — | |
VLAVGBDMWFWAPA
|
7.1 | IC50 | 3 | — | |
BUYAXUCATQBEKE
|
7.1 | IC50 | 3 | — | |
KFRGPUFONMCXQI
|
7.1 | IC50 | 11 | — | |
RVKNONNXSNALJV
|
7.1 | IC50 | 21 | — | |
BTIHMVBBUGXLCJ
|
7.1 | Ki | 7 | Yes | |
CHADTINFLWZSKR
|
7.1 | Ki | 26 | — | |
DQPYZHUAILXFJI
|
7.1 | Ki | 27 | — | |
LONMOKRIWNAKRA
|
7.1 | IC50 | 2 | — | |
NIUJTENHSPPCKO
|
7.1 | Ki | 9 | — | |
PNLPHGXRRNXSNB
|
7.1 | IC50 | 11 | — | |
QAJPIJHWTGPUNZ
|
7.1 | Ki | 37 | — |