Target Details
| UniProt AC | P50613 |
|---|---|
| Gene Symbol | CDK7 |
| Protein Name | Cyclin-dependent kinase 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,007
- Clinical molecules 36
- Avg pChEMBL 6.99
KEGG Pathways (3)
Active Molecules (1,007)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LAJPWWATQVPFEQ
|
7.4 | IC50 | 6 | Yes | |
OHOSYPVIDYXWQF
|
7.4 | IC50 | 2 | — | |
PIMQWRZWLQKKBJ
|
7.4 | Ki | 5 | — | |
SLKCVFPEQGHNSI
|
7.4 | Ki | 29 | — | |
XZWVOUQIYLZUCJ
|
7.4 | Ki | 23 | — | |
YCVGLKWJKIKVBI
|
7.4 | IC50 | 6 | — | |
RPGZQOOZHIEPJW
|
7.4 | Kd | 18 | — | |
RPGZQOOZHIEPJW
|
7.4 | Kd | 18 | — | |
YCVGLKWJKIKVBI
|
7.4 | IC50 | 5 | — | |
NKDOPEFRNJXAOV
|
7.4 | IC50 | 6 | — | |
SVBAJHORENGYPT
|
7.4 | IC50 | 3 | — | |
YPJSFIQDRPQLPZ
|
7.4 | Ki | 9 | — | |
HKSZLNNOFSGOKW
|
7.3 | Kd | 213 | — | |
HXEWDPLWMXRCAA
|
7.3 | Ki | 5 | — | |
BXMBIVXDTXURDF
|
7.3 | Ki | 9 | — | |
MWKSRKSEWLRPBL
|
7.3 | Kd | 1075 | — | |
XUKYEEYMPUGKNF
|
7.3 | Ki | 4 | — | |
AKDZNPFQMDRCMU
|
7.3 | IC50 | 7 | — | |
BLQYVHBZHAISJM
|
7.3 | Ki | 54 | — | |
WDARYLSSWBWVCU
|
7.3 | Ki | 49 | — | |
FSBMCTDYWXIBLM
|
7.3 | IC50 | 22 | — | |
BHDMRJQKCJHJGQ
|
7.3 | Ki | 10 | — | |
KEOUPUFVTYPQHX
|
7.3 | IC50 | 3 | — | |
KPABJHHKKJIDGX
|
7.3 | IC50 | 3 | — | |
UEFCSGDOOJJXTN
|
7.3 | IC50 | 46 | — | |
BRBJCJHJBAMBPR
|
7.3 | IC50 | 12 | — | |
BWONSNVPSAEXDY
|
7.3 | Ki | 9 | — | |
LQHMJVOJVOLFTJ
|
7.3 | IC50 | 7 | — | |
PUXKEKPYASIYGT
|
7.3 | IC50 | 7 | — | |
SCIUSXXNEKMFGZ
|
7.3 | IC50 | 3 | — | |
DVBHEDLDLJERFO
|
7.3 | Ki | 9 | — | |
FNWHPLLNMLOZTL
|
7.2 | IC50 | 3 | — | |
TWVJVNNYNNBYED
|
7.2 | Ki | 5 | — | |
AIDWTYRIDDCANO
|
7.2 | IC50 | 3 | — | |
AIPOXKONBJUOQN
|
7.2 | IC50 | 3 | — | |
GNEARXSVRDSWKT
|
7.2 | IC50 | 7 | — | |
UEQDUFKJHSOXJD
|
7.2 | IC50 | 3 | — | |
YKSDGHNGKNMUGI
|
7.2 | IC50 | 12 | — | |
YRUAMADPOZOPBF
|
7.2 | IC50 | 7 | — | |
AWLUUDKTCDEPGP
|
7.2 | Ki | 9 | — | |
OCBFHTQGXPIABP
|
7.2 | IC50 | 3 | — | |
OUSFTKFNBAZUKL
|
7.2 | IC50 | 58 | Yes | |
VUKGJVXJRDQYFA
|
7.2 | IC50 | 9 | — | |
YKCGAMRTHVAZHZ
|
7.2 | IC50 | 4 | — | |
AMJGJBCDROPOGP
|
7.2 | IC50 | 3 | — | |
BAVNIMZQZCFODD
|
7.2 | IC50 | 3 | — | |
BOBOCYVCAPAGSR
|
7.2 | IC50 | 3 | — | |
BXERJFWRHNGYKW
|
7.2 | IC50 | 3 | — | |
CFQMBAKFNZEINV
|
7.2 | IC50 | 3 | — | |
CUBDFKPNPMKIJA
|
7.2 | IC50 | 3 | — |