Target Details
| UniProt AC | P50613 |
|---|---|
| Gene Symbol | CDK7 |
| Protein Name | Cyclin-dependent kinase 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,007
- Clinical molecules 36
- Avg pChEMBL 6.99
KEGG Pathways (3)
Active Molecules (1,007)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BEJCLDKQCNVTQR
|
7.6 | Ki | 16 | — | |
CBARNMHMGRVVLO
|
7.6 | IC50 | 11 | — | |
MEFDJWAWYLVECZ
|
7.6 | IC50 | 3 | — | |
OTPFZAVDWPCJLJ
|
7.6 | Ki | 9 | — | |
PFMZZSWRMJKBOJ
|
7.6 | IC50 | 3 | — | |
PLHUMPJXRHMFFR
|
7.6 | Ki | 28 | — | |
SCEXYAFUDMYBSF
|
7.6 | Ki | 5 | — | |
SYNHRWSDSNIWGA
|
7.6 | IC50 | 3 | — | |
UELYDGOOJPRWGF
|
7.6 | IC50 | 13 | — | |
URNZTLZSAVLTIZ
|
7.6 | Ki | 26 | — | |
XFWUTMHVDGPWLH
|
7.6 | Ki | 75 | — | |
XZONYYFHQICDAM
|
7.6 | Ki | 19 | — | |
HJAJKTBYEIGNCK
|
7.6 | IC50 | 2 | — | |
MTGSQICHLUCDIB
|
7.6 | IC50 | 3 | — | |
QUYSDNMRBIJUBA
|
7.6 | IC50 | 3 | — | |
BKCOGSHTNWTZNI
|
7.6 | IC50 | 15 | — | |
TYZYGROMFZZJSB
|
7.6 | IC50 | 3 | — | |
OTWWRAXKMZULAP
|
7.5 | IC50 | 2 | — | |
JISLYHZGPUPOHU
|
7.5 | Ki | 8 | — | |
NRKPJTBUHZKLGS
|
7.5 | Ki | 9 | — | |
UVAGZHXCVLIMPV
|
7.5 | IC50 | 2 | — | |
CGBFAYLLULJFBW
|
7.5 | Ki | 8 | — | |
OBJNFLYHUXWUPF
|
7.5 | IC50 | 17 | — | |
QNABDSWBQJKBHK
|
7.5 | IC50 | 45 | — | |
OWDGCSZIOWIQOM
|
7.5 | IC50 | 2 | — | |
HZPACYSNLOCDLW
|
7.5 | Ki | 48 | — | |
KTWBYGUSEYSRND
|
7.5 | Ki | 28 | — | |
OWRXHGAFWZFFCW
|
7.5 | Ki | 113 | — | |
ZBYGBITZFKOQTA
|
7.5 | Ki | 18 | — | |
CXEVHNQTHRJLAT
|
7.5 | IC50 | 2 | — | |
ATGAGBNTLIIJJW
|
7.5 | IC50 | 3 | — | |
DFCOQRZKYSNBAZ
|
7.5 | Ki | 5 | — | |
KMVBIPSQSSTTCJ
|
7.5 | IC50 | 11 | — | |
CKLUGGQEKTXIHN
|
7.5 | IC50 | 3 | — | |
YGHPDKYRIZDBRZ
|
7.5 | IC50 | 3 | — | |
AHKMMSOBMZWPIC
|
7.5 | IC50 | 3 | — | |
ICIRUJKCPRMGQT
|
7.5 | IC50 | 3 | — | |
CUBLXHMKEYHDBZ
|
7.5 | IC50 | 2 | — | |
UVMVCEDKKHGTIW
|
7.4 | IC50 | 7 | — | |
VHEPZOYVQIFCJY
|
7.4 | IC50 | 2 | — | |
VXBAJLGYBMTJCY
|
7.4 | IC50 | 34 | Yes | |
BCIYCFUPZKVHKU
|
7.4 | IC50 | 3 | — | |
MCUJKPPARUPFJM
|
7.4 | Kd | 11 | — | |
POTKDJWRAMHALZ
|
7.4 | IC50 | 9 | — | |
WFWFIAFTMSUDNO
|
7.4 | IC50 | 7 | — | |
PHMSPIZKLQNZQG
|
7.4 | IC50 | 2 | — | |
UTTLTLACXKGJRK
|
7.4 | IC50 | 3 | — | |
BGYVWFZMYBWCNY
|
7.4 | Ki | 30 | — | |
CDKRFBBXZQUTDX
|
7.4 | Ki | 9 | — | |
KFIMNHWHBJDDKJ
|
7.4 | IC50 | 3 | — |