Target Details
| UniProt AC | P50613 |
|---|---|
| Gene Symbol | CDK7 |
| Protein Name | Cyclin-dependent kinase 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,007
- Clinical molecules 36
- Avg pChEMBL 6.99
KEGG Pathways (3)
Active Molecules (1,007)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XPHWIERLJBFPFV
|
8.2 | Ki | 69 | — | |
ZKLJKKASNXVQBZ
|
8.2 | Ki | 27 | — | |
DHZKWPMYADCRCR
|
8.2 | IC50 | 4 | — | |
QMNWYIJJYDNVOQ
|
8.2 | IC50 | 3 | — | |
ITSPBRBMIPVDCF
|
8.2 | Ki | 5 | — | |
VWSDWOYFAZHKHK
|
8.2 | IC50 | 3 | — | |
WINYZTMONKJGNR
|
8.2 | IC50 | 3 | — | |
IVOIFGRBXZVOFK
|
8.2 | IC50 | 3 | — | |
AYCPARAPKDAOEN
|
8.2 | IC50 | 73 | — | |
FXAIHFVIKDJIAK
|
8.2 | IC50 | 2 | — | |
RKKBVXKJICHLRV
|
8.2 | IC50 | 2 | — | |
KOBLEPSVVLTMLE
|
8.1 | IC50 | 3 | — | |
LHGBWMYXJKRMIP
|
8.1 | IC50 | 3 | — | |
USDBEZRARXRGGK
|
8.1 | IC50 | 5 | — | |
FPTHHKVHJDUFEA
|
8.1 | IC50 | 3 | — | |
IOKORVXLSWJWQL
|
8.1 | IC50 | 3 | — | |
JWLWJKKNZAGESY
|
8.1 | IC50 | 3 | — | |
YIZTXJASFULJSI
|
8.1 | IC50 | 2 | — | |
VBNZZGDQJYVFDA
|
8.1 | IC50 | 3 | — | |
CGPMSCGCDRRRHS
|
8.1 | IC50 | 3 | — | |
JOPQDQBLBCRZES
|
8.1 | IC50 | 3 | — | |
QESKJLNPFAAHST
|
8.1 | IC50 | 3 | — | |
ROBBURZERULYQU
|
8.1 | IC50 | 3 | — | |
MRWKUIOLQRITLV
|
8.1 | IC50 | 3 | — | |
OIXCMADAZITJOX
|
8.1 | IC50 | 3 | — | |
JVBMCKNTDXXCTA
|
8.0 | IC50 | 3 | — | |
MZVXBMQKLXUJEV
|
8.0 | IC50 | 3 | — | |
FGNHJXSBQQICEW
|
8.0 | Ki | 7 | — | |
DKXHSOUZPMHNIZ
|
8.0 | IC50 | 51 | Yes | |
HUXYBQXJVXOMKX
|
8.0 | IC50 | 28 | — | |
JRNJNYBQQYBCLE
|
8.0 | Kd | 40 | Yes | |
NWMPVMMGSHXANZ
|
8.0 | Ki | 58 | — | |
XKFTZKGMDDZMJI
|
8.0 | Ki | 56 | — | |
ZMFBLJJBZOWLHV
|
8.0 | IC50 | 3 | — | |
LGHAAIHVITWSPZ
|
8.0 | IC50 | 3 | — | |
LHHVKIBLSJIVFI
|
8.0 | IC50 | 2 | — | |
KMCFZYFLOLCIFG
|
8.0 | IC50 | 3 | — | |
OZIBOKYMPVXMRJ
|
8.0 | IC50 | 3 | — | |
QJRKDESSUVYBDT
|
8.0 | IC50 | 3 | — | |
GLMORIZVXAPSPO
|
8.0 | IC50 | 3 | — | |
YPMOBRWHNOTUIL
|
7.9 | IC50 | 7 | — | |
LBFBGDRIHBSNMU
|
7.9 | IC50 | 2 | — | |
SOHKYLNCPBLXTM
|
7.9 | IC50 | 3 | — | |
VTTAWQQFJQXYFM
|
7.9 | IC50 | 2 | — | |
VBYGXNURPHQSPG
|
7.9 | IC50 | 5 | — | |
DQDNKGFWJQBIFN
|
7.9 | IC50 | 3 | — | |
RVSKJUNTDGBSSS
|
7.9 | Ki | 25 | — | |
VTWWRKFUHCSCEW
|
7.9 | Kd | 19 | — | |
YSKUCLKVLULVQM
|
7.9 | IC50 | 3 | — | |
UOMFAOIPQSGEDO
|
7.9 | IC50 | 3 | — |