Target Details
| UniProt AC | P50613 |
|---|---|
| Gene Symbol | CDK7 |
| Protein Name | Cyclin-dependent kinase 7 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,007
- Clinical molecules 36
- Avg pChEMBL 6.99
KEGG Pathways (3)
Active Molecules (1,007)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OLEFHQBTXFCZON
|
10.8 | Ki | 2 | — | |
KAUXKMRRDIDIRK
|
10.5 | Kd | 8 | — | |
DQFXKZPDQHUJLY
|
10.2 | Kd | 8 | — | |
NUMHIIKAGFNIFT
|
10.2 | Kd | 8 | — | |
DGAWYBIEBJUVHR
|
10.1 | Kd | 8 | — | |
DIIRGFRZMVBYSW
|
10.1 | Kd | 8 | — | |
PCHKTFSWKCJOTQ
|
10.1 | Kd | 8 | — | |
JEWRIBSMLSEECE
|
10.0 | Kd | 8 | — | |
XNWQJSPBCYZFAU
|
10.0 | Kd | 8 | — | |
LSGRZENCFIIHNV
|
9.9 | IC50 | 3 | — | |
SLIFZZITPODXKX
|
9.8 | Kd | 6 | — | |
BFEWHEFVBQRIIR
|
9.7 | Kd | 8 | — | |
YSPIHUWHLMNFOV
|
9.5 | Kd | 5 | — | |
XWKQZYOSWGEGIH
|
9.5 | Kd | 9 | — | |
YDHKLKQGRRFWHD
|
9.5 | Kd | 8 | — | |
JDJOUBVVSQDIRC
|
9.4 | IC50 | 3 | — | |
DMCVVJAYVRAPRW
|
9.2 | Ki | 5 | — | |
CVWXJKQAOSCOAB
|
9.2 | IC50 | 35 | — | |
TWWKXZDIDHDHRF
|
9.0 | IC50 | 7 | — | |
YISMQBFJYDFMAL
|
9.0 | IC50 | 46 | — | |
PEMUGDMSUDYLHU
|
8.9 | IC50 | 5 | — | |
RVZJFCNYSSUDCU
|
8.9 | IC50 | 7 | — | |
GWRVGNYOXQHPMF
|
8.7 | Ki | 5 | — | |
KPABJHHKKJIDGX
|
8.7 | Ki | 3 | — | |
ODTNVBQMSINVPK
|
8.7 | Ki | 6 | — | |
GLOFAMHSVMGLKL
|
8.6 | IC50 | 4 | — | |
QTHCAAFKVUWAFI
|
8.6 | Kd | 23 | — | |
CSYVEHWJTGNMOY
|
8.6 | Ki | 7 | — | |
HZZNUWNFLHMBRW
|
8.6 | IC50 | 9 | — | |
OVPNQJVDAFNBDN
|
8.6 | Kd | 44 | Yes | |
XSKBBXDFCDHKGM
|
8.5 | Ki | 3 | — | |
ODTNVBQMSINVPK
|
8.5 | Ki | 6 | — | |
KHGPYYFCIAISBU
|
8.5 | Ki | 31 | — | |
CWZJJLMGMPZMDY
|
8.4 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
8.4 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
8.4 | Kd | 149 | — | |
ADMFLILDQJSEIK
|
8.4 | Ki | 72 | — | |
VSTRBHWJZOVRDC
|
8.4 | IC50 | 4 | — | |
LYADGAGFYYXXIO
|
8.4 | IC50 | 82 | — | |
CPZWNPKQAYBTEE
|
8.4 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
8.3 | Kd | 153 | — | |
VZQDFIKUYBSQRQ
|
8.3 | IC50 | 6 | — | |
AJNPBOWCTJZTHG
|
8.3 | IC50 | 2 | — | |
OFPXYNMQWVCVKZ
|
8.3 | Ki | 8 | — | |
ZBFCXGKZXRBIFF
|
8.3 | IC50 | 5 | — | |
QVBVFLKFEISMLZ
|
8.3 | IC50 | 9 | — | |
UZPUYHARAXYZLT
|
8.2 | IC50 | 3 | — | |
VSTRBHWJZOVRDC
|
8.2 | IC50 | 2 | — | |
XAQRVVLOLCCQEB
|
8.2 | IC50 | 3 | — | |
ACSYKUPGCXYRRO
|
8.2 | Ki | 26 | — |