Target Details
| UniProt AC | P50579 |
|---|---|
| Gene Symbol | METAP2 |
| Protein Name | Methionine aminopeptidase 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00557 (Peptidase_M24) |
Summary
- Multi-target molecules 75
- Clinical molecules 0
- Avg pChEMBL 7.33
Active Molecules (75)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AKSQBPCRIODOMP
|
6.9 | IC50 | 2 | — | |
OKRRCGPMTODYSO
|
6.9 | IC50 | 2 | — | |
PZRVLRRTOLHQPA
|
6.9 | IC50 | 2 | — | |
VBUWQVASCOSYOA
|
6.8 | IC50 | 2 | — | |
SWVZZGKHFRKDPR
|
6.7 | IC50 | 2 | — | |
OXGKPVIBOVJKSI
|
6.7 | IC50 | 2 | — | |
FTRFOFPAMKYZPH
|
6.6 | IC50 | 4 | — | |
QPVQIYYFNNDMOE
|
6.6 | IC50 | 2 | — | |
UYXAPGZGTCWPHK
|
6.6 | IC50 | 2 | — | |
JHXYEIHBHBJJIT
|
6.5 | IC50 | 2 | — | |
NAOYSRBUEYWQNL
|
6.5 | IC50 | 3 | — | |
WSQQTUKKGLYHCD
|
6.4 | IC50 | 2 | — | |
NKASPYGDXVCCTA
|
6.4 | IC50 | 2 | — | |
XSYJUVKQRPLTAU
|
6.4 | IC50 | 2 | — | |
WDNVNCPECUHEGM
|
6.4 | IC50 | 2 | — | |
DUYDXTWDEKJZHW
|
6.3 | IC50 | 2 | — | |
KEKIZDKQHXXAEP
|
6.3 | IC50 | 2 | — | |
KZDTUSZNJHGAIW
|
6.2 | IC50 | 2 | — | |
SXTKECRQJMUZOI
|
6.2 | IC50 | 2 | — | |
YYZBXLHPDIWNHC
|
6.1 | IC50 | 2 | — | |
JYZRJSXLGQYLJB
|
6.0 | IC50 | 2 | — | |
JTJRNFGGGCLXSL
|
6.0 | IC50 | 2 | — | |
PKAMRWQMJQIISK
|
6.0 | IC50 | 2 | — | |
PJHRBUCIVIJVKT
|
6.0 | IC50 | 2 | — | |
YJVSNGVKQCPVFF
|
6.0 | IC50 | 2 | — |