Target Details
| UniProt AC | P50281 |
|---|---|
| Gene Symbol | MMP14 |
| Protein Name | Matrix metalloproteinase-14 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11857 (DUF3377) PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 409
- Clinical molecules 255
- Avg pChEMBL 7.05
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (409)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ASSONXJFMGBTAQ
|
6.2 | IC50 | 3 | Yes | |
LHVGXRIIQBVWQU
|
6.2 | Ki | 4 | Yes | |
HEKVSVDHQDDIEK
|
6.2 | IC50 | 2 | — | |
IJHSQTQFKJCKEA
|
6.2 | IC50 | 3 | — | |
KXFPWCKTSXRQIS
|
6.2 | IC50 | 4 | — | |
QNKSDDQPRLWOEC
|
6.2 | Ki | 5 | Yes | |
UDTINYVLJDOKAN
|
6.2 | IC50 | 3 | — | |
NMPGSGFXAAVWRZ
|
6.2 | IC50 | 2 | — | |
OUZMHHWAGJCAFA
|
6.2 | Ki | 8 | — | |
YZKJTNXYLZWHHJ
|
6.2 | IC50 | 7 | Yes | |
ANZVEJFIFVKQAS
|
6.2 | IC50 | 3 | — | |
DJZNIZCARKSSDE
|
6.2 | IC50 | 9 | Yes | |
DUONGMKIDQRGNH
|
6.1 | IC50 | 6 | — | |
JOBBURWSJZOPNT
|
6.1 | IC50 | 4 | Yes | |
MTSOZTJGECJILJ
|
6.1 | IC50 | 6 | Yes | |
NIPJJOWPCLBDGS
|
6.1 | IC50 | 8 | Yes | |
FIPYOKGRSDJCAR
|
6.1 | IC50 | 9 | Yes | |
JOKZNFFZUNYVMR
|
6.1 | Ki | 5 | Yes | |
RCQCNSNJGRCTSZ
|
6.1 | IC50 | 3 | — | |
BIHFFXMAAJBXAB
|
6.1 | IC50 | 2 | — | |
CKZHFOKQZRZCPF
|
6.1 | IC50 | 9 | Yes | |
XIQNNSMTTLQUTR
|
6.1 | IC50 | 6 | Yes | |
IQVPMSHPSMKSIK
|
6.1 | Ki | 3 | Yes | |
QASGJNZOZYCBGQ
|
6.1 | IC50 | 4 | — | |
QTWBSNWADUEERO
|
6.1 | IC50 | 2 | — | |
VVZFBVIPGIVQRI
|
6.1 | IC50 | 7 | Yes | |
CPUBMGYGVNFLPZ
|
6.1 | IC50 | 8 | Yes | |
ITXQTOBRXFVFDQ
|
6.1 | IC50 | 2 | — | |
QGMPTSWHSCMOJI
|
6.1 | IC50 | 3 | — | |
SSXHPSBZPUTJCO
|
6.1 | IC50 | 3 | — | |
JOGYGVFUVCZABB
|
6.1 | IC50 | 9 | Yes | |
LBVBVIKJOWWVJX
|
6.1 | IC50 | 4 | — | |
NVCCYYKMLFBFPP
|
6.1 | IC50 | 3 | — | |
KFGJNQLPIZMSFB
|
6.0 | IC50 | 5 | Yes | |
KREIDOPERSNSKP
|
6.0 | IC50 | 3 | — | |
LIJQQAFTSYEDRO
|
6.0 | IC50 | 6 | Yes | |
LSRFXDADRHAGGZ
|
6.0 | IC50 | 2 | — | |
NILIMKWDWHKQOZ
|
6.0 | IC50 | 7 | Yes | |
PHMPGOJWLISPFK
|
6.0 | Ki | 4 | Yes | |
WVHOOIOSMOLBGZ
|
6.0 | IC50 | 4 | — | |
BBUFBPSZYHVWGA
|
6.0 | IC50 | 5 | Yes | |
JGTIIKHYSZFICL
|
6.0 | IC50 | 5 | Yes | |
UGZBIMMKYPYEOY
|
6.0 | IC50 | 3 | — | |
UUVAUHUMINHXNV
|
6.0 | IC50 | 2 | — | |
IVQNYNVXTUYYFR
|
6.0 | IC50 | 4 | — | |
KDIPAKUGVJEBFC
|
6.0 | IC50 | 2 | — | |
MDNBGABATBOAOY
|
6.0 | IC50 | 6 | Yes | |
NFPKLGKUZSGXBR
|
6.0 | IC50 | 6 | Yes | |
YYBFXMXFWMJGLB
|
6.0 | IC50 | 8 | Yes | |
HHHJVFVJVOPDRT
|
6.0 | IC50 | 3 | — |