Target Details
| UniProt AC | P50281 |
|---|---|
| Gene Symbol | MMP14 |
| Protein Name | Matrix metalloproteinase-14 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11857 (DUF3377) PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 409
- Clinical molecules 255
- Avg pChEMBL 7.05
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (409)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AEOWLQGPNGMHBP
|
6.4 | Ki | 8 | — | |
YTQYMJLEQVXIPD
|
6.4 | Ki | 4 | — | |
FBLGEUMPZQFQFF
|
6.4 | IC50 | 2 | — | |
NVERRANKYVTEPN
|
6.4 | IC50 | 2 | — | |
DUPWUQYVKWCUOG
|
6.4 | Ki | 7 | — | |
YNSXKATXVIZKSB
|
6.4 | IC50 | 5 | — | |
YSYXAGMNRKARQB
|
6.4 | IC50 | 4 | Yes | |
BFJIOGLKGISOKV
|
6.4 | Ki | 8 | — | |
JOKZNFFZUNYVMR
|
6.4 | Ki | 5 | Yes | |
LEDMBBYIVRLZAS
|
6.4 | Ki | 9 | Yes | |
GCYXMFHUCWJAKI
|
6.3 | IC50 | 2 | — | |
JZZAWBZYLOHRQP
|
6.3 | IC50 | 2 | — | |
QTHGVXWBMQNWSU
|
6.3 | IC50 | 2 | — | |
LWHDLJDNHJFUSI
|
6.3 | Ki | 2 | Yes | |
MYFWCGILTGDUAM
|
6.3 | Ki | 8 | Yes | |
HNEDFPGSHTUVKZ
|
6.3 | IC50 | 7 | Yes | |
LWFCUEQJXZSHMP
|
6.3 | IC50 | 7 | Yes | |
AOPZFYOXZYZEAC
|
6.3 | IC50 | 7 | Yes | |
KNKPUUINTPWUPH
|
6.3 | IC50 | 3 | — | |
QVNZBDLTUKCPGJ
|
6.3 | IC50 | 10 | — | |
KOKCTGWRLDNNGZ
|
6.3 | IC50 | 3 | Yes | |
PPLPLBVUEJOBPI
|
6.3 | IC50 | 4 | — | |
PZJJOMPTIHBGHO
|
6.3 | IC50 | 8 | Yes | |
SDZHRLYVISHMEO
|
6.3 | IC50 | 3 | — | |
YVJXBWDNNWDVMN
|
6.3 | IC50 | 9 | Yes | |
AVBNYKAIQSRTNJ
|
6.3 | Ki | 2 | — | |
BRKOQUQULDVEDN
|
6.3 | Ki | 4 | Yes | |
CHBRRXABVNYHLG
|
6.3 | IC50 | 2 | — | |
HCCYYUWFQWPMDZ
|
6.3 | Ki | 4 | Yes | |
JDBUKSMCZPXYJU
|
6.3 | IC50 | 4 | — | |
JGWTVBVOISUVJD
|
6.3 | IC50 | 9 | — | |
JUQBJPICEZJIRQ
|
6.3 | Ki | 2 | — | |
NWYAUZLEGMZWIR
|
6.3 | IC50 | 2 | — | |
PAXQYYVHPNBESJ
|
6.3 | IC50 | 4 | — | |
QDHXNZRPVLUOML
|
6.3 | Ki | 6 | — | |
WNEMBEALMHVXIK
|
6.3 | IC50 | 7 | — | |
XLKQIIIKETWLMI
|
6.3 | Ki | 8 | — | |
OTCQKJMDFJEBFM
|
6.2 | IC50 | 6 | — | |
QAKGJAQGTQLMFN
|
6.2 | IC50 | 2 | — | |
CXKWJJJVWDMSAG
|
6.2 | Ki | 3 | — | |
DVBWYFQJLIUTJA
|
6.2 | Ki | 4 | Yes | |
MKGHITYLXXYNMZ
|
6.2 | IC50 | 3 | — | |
SFHMNFHDIRPFKM
|
6.2 | IC50 | 7 | Yes | |
VMOSDDURWLNMNG
|
6.2 | IC50 | 8 | Yes | |
VCASEBIJMMTOBI
|
6.2 | IC50 | 4 | — | |
VTRJTXRAOIMSTL
|
6.2 | Ki | 8 | Yes | |
WVAIZSKMOMDPIT
|
6.2 | IC50 | 6 | Yes | |
CBZOKXRPUYLLBY
|
6.2 | IC50 | 2 | — | |
HMJIPPQTLJLPNE
|
6.2 | IC50 | 3 | Yes | |
QPWBTJDQYIYLND
|
6.2 | IC50 | 4 | — |