Target Details
| UniProt AC | P50281 |
|---|---|
| Gene Symbol | MMP14 |
| Protein Name | Matrix metalloproteinase-14 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11857 (DUF3377) PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 409
- Clinical molecules 255
- Avg pChEMBL 7.05
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (409)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KSGNBXMXFPLVKJ
|
6.6 | IC50 | 3 | Yes | |
BBUAWDNXWDAMGY
|
6.6 | IC50 | 4 | Yes | |
GJOCABIDMCKCEG
|
6.6 | IC50 | 6 | Yes | |
GODQVOUTCHZIOJ
|
6.6 | Ki | 3 | Yes | |
HTBWAVKWLNLFGD
|
6.6 | IC50 | 2 | — | |
QOWBVKQSFCSJAK
|
6.6 | IC50 | 5 | — | |
WVSIAOYHEIZRMM
|
6.6 | IC50 | 2 | — | |
BTMGFNYLYGWAKT
|
6.6 | Ki | 7 | Yes | |
JPMXJRBHCOULJI
|
6.6 | IC50 | 4 | — | |
WJWOJAKOSRCFKB
|
6.6 | Ki | 9 | Yes | |
ZGBAPSHWPBXEKN
|
6.6 | IC50 | 10 | — | |
WPYFTDWGMAINBU
|
6.6 | IC50 | 5 | Yes | |
FANDWSFYLCHFFT
|
6.6 | Ki | 2 | — | |
LQNSDZTXHZUYKJ
|
6.6 | IC50 | 10 | Yes | |
LZYKHUZBVFGWCA
|
6.6 | IC50 | 3 | Yes | |
AMUGNOPZMAZKFD
|
6.6 | Ki | 4 | Yes | |
BMVSRGXHTJYIKY
|
6.6 | Ki | 2 | — | |
OTCWHHBFFQOWCU
|
6.6 | IC50 | 2 | — | |
QUIDRRLYQSJQMX
|
6.6 | Ki | 4 | Yes | |
UYHGJXBEWRNPQI
|
6.6 | Ki | 2 | — | |
CPYCKLJBTHKVRT
|
6.5 | IC50 | 3 | Yes | |
GPZUWAHQDYJABE
|
6.5 | Ki | 3 | — | |
OIZMOMFOLNBXHF
|
6.5 | IC50 | 9 | — | |
UVGAWIJNBYCHSP
|
6.5 | Ki | 9 | Yes | |
UVGAWIJNBYCHSP
|
6.5 | Ki | 7 | — | |
XWUCDOCUSPAHFU
|
6.5 | IC50 | 2 | — | |
XXZNXULRAJJTRV
|
6.5 | IC50 | 5 | Yes | |
BSTYDWORGHMRLI
|
6.5 | Ki | 5 | — | |
IIABJCHWKFZJBK
|
6.5 | Ki | 9 | Yes | |
IIABJCHWKFZJBK
|
6.5 | Ki | 9 | Yes | |
LKJAZJMUPQPJNA
|
6.5 | IC50 | 6 | Yes | |
ZVJILQAAQQNBOP
|
6.5 | IC50 | 6 | — | |
RPWGPXSVYLHGRZ
|
6.5 | IC50 | 7 | Yes | |
WOIMZSMDPIJLFO
|
6.5 | Ki | 7 | Yes | |
YHSMTPXGPORQER
|
6.5 | IC50 | 3 | Yes | |
HGHQBSHHIZJUCO
|
6.5 | IC50 | 2 | — | |
SBTMZMWGVVORIF
|
6.5 | IC50 | 6 | Yes | |
AKOBMMAQXVKOJR
|
6.4 | IC50 | 5 | Yes | |
KPYDTDKHTIUCAB
|
6.4 | Ki | 3 | Yes | |
LEDMBBYIVRLZAS
|
6.4 | Ki | 9 | Yes | |
UDTXDKDGZMYOBK
|
6.4 | IC50 | 5 | Yes | |
ZCRWOWSOWBMWGI
|
6.4 | IC50 | 8 | Yes | |
HYBHKZKKEGAPOP
|
6.4 | IC50 | 6 | — | |
KRFFMGOIPZCPLJ
|
6.4 | IC50 | 3 | — | |
PDKBAEDNMKVROV
|
6.4 | Ki | 8 | Yes | |
QVLRRQHYUCZYFV
|
6.4 | IC50 | 3 | — | |
RKYYWBHSYPIJKC
|
6.4 | IC50 | 4 | — | |
ZYHWVZVONQGAQS
|
6.4 | IC50 | 2 | — | |
AFXZHRNVMMQHOL
|
6.4 | IC50 | 4 | Yes | |
WAWUNJHTWVBKFW
|
6.4 | IC50 | 3 | — |