Target Details
| UniProt AC | P50281 |
|---|---|
| Gene Symbol | MMP14 |
| Protein Name | Matrix metalloproteinase-14 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11857 (DUF3377) PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 409
- Clinical molecules 255
- Avg pChEMBL 7.05
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (409)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NIAIEBGBRXKPAO
|
6.9 | Ki | 7 | — | |
BXLWVAKSQMYQKF
|
6.9 | Ki | 5 | Yes | |
GRRDUDJQILRRES
|
6.9 | Ki | 3 | — | |
GRRDUDJQILRRES
|
6.9 | Ki | 4 | — | |
HYDHEJPXRHGPLP
|
6.9 | IC50 | 3 | Yes | |
BVNHOVTUHKATJL
|
6.9 | Ki | 4 | Yes | |
JJTWETADXAELLS
|
6.9 | Ki | 9 | Yes | |
VKFNDAOTTJONML
|
6.9 | IC50 | 9 | Yes | |
UGRPRGWEEBXORM
|
6.9 | IC50 | 3 | — | |
CUKATAAPVFYVIL
|
6.8 | IC50 | 9 | — | |
DONMTDNLNMLOIC
|
6.8 | Ki | 13 | Yes | |
KIMAXDZENSBFAC
|
6.8 | IC50 | 3 | Yes | |
LRRAUDSVXJEODP
|
6.8 | Ki | 6 | Yes | |
PTUCPHGSAFOJAU
|
6.8 | Ki | 9 | — | |
PTUCPHGSAFOJAU
|
6.8 | Ki | 9 | Yes | |
PTUCPHGSAFOJAU
|
6.8 | Ki | 7 | — | |
STSMSPOAFPZOFC
|
6.8 | Ki | 3 | — | |
JXHAGXRDZALSLG
|
6.8 | Ki | 9 | Yes | |
IEHSRERHOYOHOA
|
6.8 | Ki | 6 | Yes | |
LTVIJEFEZVFIST
|
6.8 | IC50 | 14 | Yes | |
RODBIJLXINIENS
|
6.8 | IC50 | 3 | Yes | |
WJULIBHPWZXMJA
|
6.8 | IC50 | 10 | Yes | |
XVVZROOOIUBICS
|
6.8 | IC50 | 3 | Yes | |
DZCGIZPIPKWUIX
|
6.8 | IC50 | 7 | Yes | |
FYFJMQCWKQDEQR
|
6.8 | IC50 | 6 | Yes | |
IXKRFERDVUXQLW
|
6.8 | IC50 | 6 | Yes | |
SXSIQUOYBXOPSS
|
6.8 | IC50 | 7 | Yes | |
YDDMVPLLJTZTQL
|
6.8 | Ki | 7 | Yes | |
OBBSDCUMPDPHQF
|
6.8 | Ki | 3 | Yes | |
BGUXTVRZPYKBBN
|
6.7 | IC50 | 5 | Yes | |
NZKKRYAESABOSS
|
6.7 | IC50 | 8 | Yes | |
GINBTQGVSPUJLE
|
6.7 | Ki | 9 | Yes | |
LEBLJISYPUWAJY
|
6.7 | Ki | 2 | — | |
QJTQSHPLYJZWCK
|
6.7 | IC50 | 4 | Yes | |
WOIMZSMDPIJLFO
|
6.7 | Ki | 9 | Yes | |
ZGTPJERIIBYCFG
|
6.7 | Ki | 5 | Yes | |
ITWGWXCEGHFMHT
|
6.7 | IC50 | 10 | Yes | |
OFXJMYWLEABUGO
|
6.7 | IC50 | 3 | Yes | |
PGEMRSCSFPLCBF
|
6.7 | IC50 | 8 | Yes | |
MKGHITYLXXYNMZ
|
6.7 | IC50 | 3 | — | |
PDKBAEDNMKVROV
|
6.7 | Ki | 9 | Yes | |
VALKNOMNTXYCBM
|
6.7 | Ki | 4 | Yes | |
WLZISXXOYYGJNT
|
6.7 | IC50 | 12 | Yes | |
YAYGKNVDBLFWFW
|
6.7 | IC50 | 6 | Yes | |
BGRGANYQQMRQLM
|
6.7 | Ki | 3 | — | |
JPTZDOYPNCQOTF
|
6.7 | Ki | 4 | Yes | |
WBRQJRYOZZQHQI
|
6.7 | IC50 | 3 | Yes | |
ZHXMXRVBOZWQPF
|
6.7 | IC50 | 5 | Yes | |
ZTJUBPXNBSLSGL
|
6.7 | IC50 | 6 | Yes | |
MESQXIKYNYUZRV
|
6.7 | IC50 | 4 | Yes |