Target Details
| UniProt AC | P50281 |
|---|---|
| Gene Symbol | MMP14 |
| Protein Name | Matrix metalloproteinase-14 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11857 (DUF3377) PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 409
- Clinical molecules 255
- Avg pChEMBL 7.05
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (409)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WUXSSALNWBMRKU
|
7.2 | Ki | 4 | Yes | |
FOSWRYKPHVPIDJ
|
7.2 | IC50 | 8 | Yes | |
KMXAXPCBRVZOGA
|
7.2 | IC50 | 7 | — | |
AYFCYVLVRYQGME
|
7.2 | IC50 | 8 | — | |
AYFCYVLVRYQGME
|
7.2 | IC50 | 9 | Yes | |
HJNKYGBTSGQBDU
|
7.2 | Ki | 10 | — | |
XGGNDAOPHPLHFW
|
7.2 | Ki | 4 | — | |
YTQYMJLEQVXIPD
|
7.2 | Ki | 4 | — | |
BRYABXWERJYEAH
|
7.2 | IC50 | 3 | Yes | |
KJNZDUKNEQXTSO
|
7.2 | Ki | 6 | — | |
NKGRTRASISLCCZ
|
7.2 | IC50 | 10 | Yes | |
WHHAEBOHMHRZGW
|
7.2 | IC50 | 4 | — | |
BVONHINTCXADCU
|
7.1 | Ki | 4 | Yes | |
DYKLASPWVUKEIT
|
7.1 | IC50 | 6 | Yes | |
BGBWSADVPWNBME
|
7.1 | IC50 | 9 | Yes | |
FQEZYKOXVAISOF
|
7.1 | IC50 | 3 | Yes | |
BZVYQWLRCHLAGK
|
7.1 | IC50 | 10 | Yes | |
NIQJXWLMDJIMHL
|
7.1 | IC50 | 4 | — | |
FGQTUBBIXYISNM
|
7.1 | IC50 | 4 | — | |
NJZUERVIVLYZMO
|
7.1 | IC50 | 5 | — | |
RQCBSNJRFVZHOS
|
7.1 | IC50 | 10 | Yes | |
SYYRIPAKWJBIOW
|
7.1 | IC50 | 8 | Yes | |
GHVMTHKJUAOZJP
|
7.1 | IC50 | 6 | — | |
AHDPJKYOQXMDIX
|
7.0 | Ki | 4 | — | |
MERYKHOGOUEPIA
|
7.0 | Ki | 4 | Yes | |
QSOYTCHABFMDFV
|
7.0 | IC50 | 10 | Yes | |
COMOZYQMQPSLMB
|
7.0 | Ki | 4 | Yes | |
GYETWAWIKBOMPE
|
7.0 | IC50 | 7 | Yes | |
RMPAKJHKSCQYEB
|
7.0 | Ki | 2 | — | |
ZNCKCQFPCKMNBK
|
7.0 | Ki | 2 | — | |
HFAGTNGCAZYYLZ
|
7.0 | Ki | 13 | Yes | |
NUFBSNVYZRUJSW
|
7.0 | IC50 | 6 | — | |
KUDQLMASLRCXLF
|
7.0 | IC50 | 6 | — | |
LNPBBURQSUEIHO
|
7.0 | IC50 | 5 | Yes | |
JKRVXAWKSWVVCV
|
7.0 | IC50 | 7 | Yes | |
KFOJCCXBEQXGOL
|
7.0 | IC50 | 3 | Yes | |
QVFLVOHFXMNIFB
|
7.0 | IC50 | 3 | Yes | |
JXHAGXRDZALSLG
|
7.0 | Ki | 9 | Yes | |
KEPYRBFIGNMAQF
|
7.0 | IC50 | 7 | Yes | |
LCLWTUJSVDCASO
|
7.0 | IC50 | 4 | Yes | |
LCLWTUJSVDCASO
|
7.0 | IC50 | 2 | — | |
LHVGXRIIQBVWQU
|
7.0 | Ki | 5 | — | |
YQEMFOGNUTYMTJ
|
7.0 | Ki | 4 | Yes | |
YQEMFOGNUTYMTJ
|
7.0 | Ki | 5 | — | |
YQEMFOGNUTYMTJ
|
7.0 | Ki | 5 | Yes | |
ORSWNUGKUNQTLF
|
7.0 | IC50 | 7 | Yes | |
LSONWRHLFZYHIN
|
7.0 | Ki | 4 | Yes | |
OTEWYJZEFZRZKI
|
7.0 | IC50 | 8 | Yes | |
PSLRKUXEVFQKIV
|
6.9 | IC50 | 2 | — | |
QTGQZAQZBAEHLR
|
6.9 | IC50 | 6 | Yes |