Target Details
| UniProt AC | P50281 |
|---|---|
| Gene Symbol | MMP14 |
| Protein Name | Matrix metalloproteinase-14 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11857 (DUF3377) PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 409
- Clinical molecules 255
- Avg pChEMBL 7.05
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (409)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BTMSEVQRJBBBAY
|
7.6 | IC50 | 3 | — | |
VFDSDRZNXLFCFF
|
7.6 | IC50 | 7 | Yes | |
FTPFWQRREQUXLQ
|
7.6 | IC50 | 3 | Yes | |
QURZZKPWFKUXBF
|
7.6 | IC50 | 5 | Yes | |
WVPKYEATTXWJLC
|
7.6 | IC50 | 5 | — | |
CVZIHNYAZLXRRS
|
7.6 | IC50 | 10 | Yes | |
PFIVDCYVKKFLEU
|
7.6 | IC50 | 5 | Yes | |
RHOVUJYSXPHHFW
|
7.6 | Ki | 2 | — | |
RVZWFNDDFJIWNJ
|
7.6 | Ki | 2 | — | |
QKXZKYSXPIUZEA
|
7.6 | IC50 | 2 | — | |
RZDDQWJXBRPPTM
|
7.6 | Ki | 3 | Yes | |
WNLZTTHHHYZJMB
|
7.6 | IC50 | 9 | Yes | |
XUOKZLGAMXUMSE
|
7.6 | IC50 | 3 | — | |
SLUQTAQKAIYNRS
|
7.6 | IC50 | 3 | Yes | |
WMJKIJLFVOMJDF
|
7.5 | IC50 | 6 | Yes | |
YTQYMJLEQVXIPD
|
7.5 | Ki | 4 | — | |
ZIXRMLDHKPIARA
|
7.5 | IC50 | 3 | — | |
RIOJMNDNYHZZFM
|
7.5 | Ki | 7 | Yes | |
VWKXFDZWHLCIIU
|
7.5 | IC50 | 9 | Yes | |
YOMXWXIANUYIMH
|
7.5 | IC50 | 10 | Yes | |
OVUDWXYTKUKYAX
|
7.5 | IC50 | 9 | Yes | |
RLHOCYLKSSHKMW
|
7.5 | IC50 | 6 | Yes | |
RBXJTRGTMYPRKK
|
7.4 | IC50 | 3 | Yes | |
YVCCTHCWKOIESX
|
7.4 | IC50 | 8 | Yes | |
BZKOBLHHRSTMHO
|
7.4 | Ki | 4 | — | |
GTXSRFUZSLTDFX
|
7.4 | IC50 | 8 | Yes | |
SFORRVNMTYAPLQ
|
7.4 | Ki | 4 | Yes | |
IWOFJPISTOGMII
|
7.4 | IC50 | 4 | — | |
QHHHTEGVVKPDKH
|
7.4 | IC50 | 6 | — | |
RFNUTMXSNZMOSL
|
7.4 | Ki | 7 | Yes | |
UFJUEKAJZPTZED
|
7.4 | Ki | 4 | Yes | |
WYBFHVSAXDKMJV
|
7.3 | Ki | 4 | Yes | |
BUKCBCDGRPOFJP
|
7.3 | IC50 | 9 | Yes | |
RDFQXFRQTOWZEQ
|
7.3 | IC50 | 8 | Yes | |
XFBRPTYLOIFAQR
|
7.3 | IC50 | 8 | Yes | |
UIODHSBHBXTRBO
|
7.3 | IC50 | 3 | Yes | |
GRRDUDJQILRRES
|
7.3 | Ki | 3 | — | |
LCYYUMHWMVOGPC
|
7.3 | IC50 | 8 | Yes | |
LWTYDGJEOHWGQD
|
7.3 | Ki | 4 | Yes | |
PFIFGQWOKBQYID
|
7.3 | IC50 | 9 | Yes | |
USEQZALNBFQSDH
|
7.3 | IC50 | 3 | — | |
SIEIWCDBNIGNIG
|
7.3 | IC50 | 7 | Yes | |
JAPLGNWCNXCEJT
|
7.2 | IC50 | 5 | Yes | |
OFCWIPGKPUJTDP
|
7.2 | IC50 | 7 | Yes | |
LTCNKRUYOJZZJO
|
7.2 | IC50 | 7 | Yes | |
NFDNOGJHVSTSMJ
|
7.2 | Ki | 7 | Yes | |
OJGIWNSVHKBBDS
|
7.2 | IC50 | 3 | Yes | |
BTCYLUBBXQARQV
|
7.2 | Ki | 7 | — | |
RILFWDKQYPJIOQ
|
7.2 | IC50 | 8 | Yes | |
SYNSXJHFJAEBFU
|
7.2 | IC50 | 2 | — |