Target Details
| UniProt AC | P50281 |
|---|---|
| Gene Symbol | MMP14 |
| Protein Name | Matrix metalloproteinase-14 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11857 (DUF3377) PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 409
- Clinical molecules 255
- Avg pChEMBL 7.05
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (409)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MEGFCBVTRXVKDO
|
8.1 | IC50 | 6 | Yes | |
PKVXJRTWUNPBJP
|
8.1 | IC50 | 6 | Yes | |
PKVXJRTWUNPBJP
|
8.1 | IC50 | 4 | — | |
PENUDEJHXUSMIL
|
8.1 | IC50 | 4 | Yes | |
JHSGRRNCQDDQBC
|
8.1 | IC50 | 9 | — | |
YPHZFHQBHSELGO
|
8.1 | IC50 | 7 | Yes | |
QDGVTWBFTFHWOG
|
8.1 | IC50 | 8 | Yes | |
OTKHAYOLIGHFRB
|
8.0 | IC50 | 5 | Yes | |
DGZZVIWCMGVHGV
|
8.0 | IC50 | 11 | Yes | |
GKHRDWHFKKUYAX
|
8.0 | Ki | 9 | — | |
IHERVMJHCHNTKO
|
8.0 | IC50 | 7 | Yes | |
YTQYMJLEQVXIPD
|
8.0 | Ki | 4 | — | |
NUTUARVYQWFZAA
|
8.0 | IC50 | 6 | Yes | |
CJTUBZULFXKTAT
|
8.0 | IC50 | 10 | Yes | |
HUAZIQKZKFNJLA
|
8.0 | IC50 | 6 | — | |
KLCHUAUMSZUJEX
|
8.0 | IC50 | 5 | Yes | |
QLTNWLFWQKKDEO
|
8.0 | IC50 | 7 | Yes | |
RVKPGECPCLBLDB
|
8.0 | IC50 | 10 | Yes | |
TUUOOTOFTLPOMW
|
8.0 | IC50 | 3 | Yes | |
UJWXVGWYDPXCST
|
8.0 | Ki | 5 | — | |
BXOTYZMFPUKYAU
|
7.9 | IC50 | 5 | Yes | |
JIRXORZYIXSWOB
|
7.9 | IC50 | 11 | Yes | |
NITYDPDXAAFEIT
|
7.9 | IC50 | 20 | Yes | |
RHWGGEKVTPKRQW
|
7.9 | IC50 | 4 | Yes | |
SFEPJGMZSMIONR
|
7.9 | IC50 | 7 | Yes | |
NXUHVWMBPOFLMA
|
7.9 | IC50 | 6 | Yes | |
DYMSXYKQOWNDKR
|
7.8 | IC50 | 4 | — | |
ZRAUMSIZBNBIFE
|
7.8 | IC50 | 8 | Yes | |
LMIHEFSBOIGKDH
|
7.8 | IC50 | 8 | Yes | |
ICCZTDHQUXGJEO
|
7.8 | IC50 | 3 | Yes | |
KLOYCYLPVRADHA
|
7.8 | IC50 | 5 | Yes | |
DNSIVPJNRUSHDP
|
7.8 | IC50 | 4 | Yes | |
BGEFVHSKSARWDE
|
7.7 | IC50 | 3 | Yes | |
FRIYTZJGYCAFHL
|
7.7 | IC50 | 3 | Yes | |
GJLVFYXHGPXLCC
|
7.7 | IC50 | 7 | Yes | |
AHXGZLJBINZPQZ
|
7.7 | IC50 | 3 | Yes | |
GTBJTISRJIZWKE
|
7.7 | IC50 | 7 | Yes | |
PLCRCZGBQOTIFV
|
7.7 | IC50 | 3 | Yes | |
WXNWNNKHEJMQOM
|
7.7 | IC50 | 8 | Yes | |
SPEYRVQKGFNUCY
|
7.7 | IC50 | 8 | Yes | |
ZXVWNUSVQOQAIY
|
7.7 | Ki | 5 | — | |
FSSPDFKSDKXWQO
|
7.7 | IC50 | 3 | Yes | |
KKRBZYCHOUTMBU
|
7.7 | Ki | 4 | Yes | |
BIHSFSZDPRDVEE
|
7.6 | IC50 | 3 | Yes | |
BSIZUMJRKYHEBR
|
7.6 | IC50 | 15 | Yes | |
GFUITADOEPNRML
|
7.6 | IC50 | 11 | Yes | |
OCENTDLFDAKGHV
|
7.6 | IC50 | 3 | Yes | |
QHCDOFQMQJCFGF
|
7.6 | IC50 | 4 | — | |
UJKKQEHHLXCTJE
|
7.6 | IC50 | 6 | — | |
XRSYNYGEEYTXJV
|
7.6 | IC50 | 2 | — |