Target Details
| UniProt AC | P50281 |
|---|---|
| Gene Symbol | MMP14 |
| Protein Name | Matrix metalloproteinase-14 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11857 (DUF3377) PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 409
- Clinical molecules 255
- Avg pChEMBL 7.05
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (409)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YKPYIPVDTNNYCN
|
9.5 | IC50 | 11 | Yes | |
GSWRTFGMHRKLKT
|
9.5 | IC50 | 14 | Yes | |
WIUDGBCTJVXBCM
|
9.5 | IC50 | 7 | — | |
ZHIRJJYNGRGHQQ
|
9.1 | IC50 | 6 | Yes | |
MTDVSXPXWCWOED
|
9.1 | IC50 | 6 | Yes | |
ROSNVSQTEGHUKU
|
9.0 | IC50 | 12 | Yes | |
OJPRZTDTKMGAMY
|
8.9 | IC50 | 3 | Yes | |
DSLRBIQFKOUGKT
|
8.9 | IC50 | 4 | Yes | |
WVUXCTUJEGJKKV
|
8.9 | IC50 | 5 | Yes | |
JDKMZILZEJPWTA
|
8.8 | IC50 | 2 | Yes | |
PKAAOTCIUWGSDS
|
8.8 | IC50 | 6 | Yes | |
OCSMOTCMPXTDND
|
8.7 | IC50 | 14 | Yes | |
LPZWIAVKYXCHGC
|
8.7 | IC50 | 7 | Yes | |
QRXOZHSEEGNRFC
|
8.7 | IC50 | 8 | Yes | |
HFLSBITWFGZVGL
|
8.7 | IC50 | 11 | Yes | |
OBJBBLBMOOBABD
|
8.7 | IC50 | 8 | Yes | |
YOZKFIDLBXLPFF
|
8.6 | IC50 | 7 | Yes | |
ONJBMYIEKPLUOX
|
8.6 | IC50 | 4 | Yes | |
FPSMXPGSVWPWCG
|
8.5 | IC50 | 8 | — | |
RLDSXGKXSYXTOQ
|
8.5 | IC50 | 3 | Yes | |
XFILPEOLDIKJHX
|
8.5 | IC50 | 12 | Yes | |
QJNGNVJSSUXWBO
|
8.5 | IC50 | 8 | Yes | |
GRSFKJZRDUZQPW
|
8.5 | IC50 | 9 | Yes | |
UZMULMICABXSNQ
|
8.4 | IC50 | 4 | Yes | |
JATUSZYMCBLDQS
|
8.4 | IC50 | 8 | Yes | |
IWQSGINKBSWILJ
|
8.4 | IC50 | 10 | — | |
KBZNOZAJAJRTII
|
8.4 | IC50 | 10 | Yes | |
WQCXDERWRJMJQA
|
8.4 | IC50 | 6 | — | |
BDONYXHHXNTUSW
|
8.4 | IC50 | 8 | Yes | |
MUWDEQLPHWVPPA
|
8.4 | Ki | 5 | — | |
YJRJYIQWWPZSTM
|
8.4 | IC50 | 6 | — | |
IXVDOEAUVAJHER
|
8.4 | IC50 | 7 | Yes | |
MWMRJYLEVAWDDL
|
8.4 | IC50 | 7 | Yes | |
KOPIIXVBCHXDHO
|
8.3 | IC50 | 8 | Yes | |
NBRBWZJMBITNBC
|
8.3 | IC50 | 8 | Yes | |
LXQUQEBAZBLBEJ
|
8.3 | IC50 | 5 | Yes | |
HXZPYZWICHZKRL
|
8.3 | IC50 | 10 | — | |
HBYRXCFAHCMHAA
|
8.2 | IC50 | 9 | Yes | |
QDPILJAKSNERSV
|
8.2 | Ki | 6 | — | |
WSFQQGCWUCOARG
|
8.2 | Ki | 6 | — | |
QHERSXDLUJOMHD
|
8.2 | Ki | 5 | — | |
ASZIRMQBBYBMMU
|
8.2 | IC50 | 7 | Yes | |
DRXVUBODYFAEED
|
8.2 | IC50 | 4 | — | |
HYIVZTPHVNIXFU
|
8.2 | IC50 | 4 | Yes | |
IMKDKHQDFFLOKK
|
8.2 | IC50 | 13 | Yes | |
QQCNGNFIZAKQDT
|
8.2 | IC50 | 4 | — | |
RYDPXGZLAKQPJB
|
8.2 | Ki | 6 | — | |
UXTZIHLCCIDADG
|
8.2 | IC50 | 2 | — | |
VMWGPLRCSWOQJR
|
8.1 | IC50 | 5 | Yes | |
ZBRHTUMWSDPCMI
|
8.1 | IC50 | 10 | Yes |