Target Details
| UniProt AC | P49841 |
|---|---|
| Gene Symbol | GSK3B |
| Protein Name | Glycogen synthase kinase-3 beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,206
- Clinical molecules 168
- Avg pChEMBL 7.19
KEGG Pathways (49)
- Alcoholic liver disease
- Alzheimer disease
- Axon guidance
- B cell receptor signaling pathway
- Basal cell carcinoma
- Breast cancer
- Cadherin signaling
- Cell cycle
- Chemokine signaling pathway
- Colorectal cancer
- Cushing syndrome
- Diabetic cardiomyopathy
- Dopaminergic synapse
- EGFR tyrosine kinase inhibitor resistance
- Endometrial cancer
- ErbB signaling pathway
- Focal adhesion
- Gastric cancer
- Growth hormone synthesis, secretion and action
- Hedgehog signaling pathway
- Hepatitis C
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human cytomegalovirus infection
- Human papillomavirus infection
- IL-17 signaling pathway
- IgSF CAM signaling
- Insulin resistance
- Insulin signaling pathway
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Melanogenesis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- PI3K-Akt signaling pathway
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Prion disease
- Prolactin signaling pathway
- Prostate cancer
- Shigellosis
- Signaling pathways regulating pluripotency of stem cells
- T cell receptor signaling pathway
- Thyroid hormone signaling pathway
- Wnt signaling pathway
- Yersinia infection
- mTOR signaling pathway
Active Molecules (2,206)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SSMMEOSYEUOMIT
|
6.5 | IC50 | 4 | — | |
XKNDLPMAXNMALL
|
6.5 | IC50 | 5 | — | |
YYWGDJIEQNZXDR
|
6.5 | IC50 | 3 | Yes | |
BOKIQWSDLBGRGI
|
6.5 | IC50 | 2 | — | |
CTJAMSGCMYAVCZ
|
6.5 | Ki | 14 | — | |
LLDVRUBUBPSOMY
|
6.5 | Ki | 4 | — | |
OGLXQFQATMRTEA
|
6.5 | IC50 | 2 | — | |
XDYOZBDORGQQDV
|
6.5 | IC50 | 3 | — | |
MPCYSIQJPBBOJL
|
6.5 | Ki | 2 | — | |
MPCYSIQJPBBOJL
|
6.5 | Ki | 3 | — | |
AWZFCQRICMFIES
|
6.5 | IC50 | 9 | Yes | |
AXILYJJKIDQSFE
|
6.5 | IC50 | 3 | — | |
FLDSZPYCDPPFIH
|
6.5 | IC50 | 2 | — | |
GWFCNMFOAORLDH
|
6.5 | IC50 | 2 | Yes | |
JQWXFCIJCDFZKC
|
6.5 | IC50 | 2 | — | |
PFWCEPWUHBDYJN
|
6.5 | IC50 | 3 | Yes | |
WCAYCTGIGMRVKS
|
6.5 | IC50 | 2 | — | |
XMNABEGDUNNDFW
|
6.5 | IC50 | 5 | — | |
ZHZPUYSNZQKXRF
|
6.5 | IC50 | 2 | — | |
ACXVCLUGFVYVMQ
|
6.5 | Ki | 2 | — | |
AJTBUWMKUOLMNM
|
6.5 | IC50 | 5 | — | |
HVHBXBDAWFYVOJ
|
6.5 | Ki | 2 | Yes | |
UGPDJSYAEGUOSO
|
6.5 | IC50 | 6 | — | |
VBWQPLLCGUWXEE
|
6.5 | IC50 | 5 | — | |
YFXZFROOGCONFB
|
6.5 | IC50 | 3 | — | |
YUPWBUPSOSSVKV
|
6.5 | Ki | 2 | — | |
ZDFKUJXTEZOUQT
|
6.5 | IC50 | 2 | — | |
AMQWJXRKJIUZAW
|
6.5 | IC50 | 2 | — | |
AQDWDWAYVBQMAM
|
6.5 | IC50 | 7 | — | |
BRBGAJDUHBVSLV
|
6.5 | IC50 | 2 | — | |
CYHDOETYGLKIAA
|
6.5 | IC50 | 4 | — | |
DKSNLQYRZJKYOC
|
6.5 | Ki | 51 | — | |
DPDVVGCNUWGGRS
|
6.5 | IC50 | 10 | — | |
GYPHGCGOSZJXOT
|
6.5 | IC50 | 5 | — | |
IKIFANJBLBFWHU
|
6.5 | Ki | 4 | — | |
IPTSYCYNQJITNJ
|
6.5 | Ki | 12 | — | |
IRNVMUQZQDLZAK
|
6.5 | IC50 | 5 | — | |
JGPBLWPUPCMPDV
|
6.5 | IC50 | 2 | — | |
JRLSUZIPUYDUKX
|
6.5 | Ki | 22 | — | |
KRIUNPBAQZGFQA
|
6.5 | Ki | 76 | — | |
LCKDESRGCHSHHO
|
6.5 | Ki | 18 | — | |
LRZYYIZFBXFSJB
|
6.5 | Ki | 69 | — | |
OBHMNLIBIPFXCY
|
6.5 | Ki | 15 | — | |
PDWYDOXDYRHDSC
|
6.5 | IC50 | 2 | — | |
QMHDOQLIVAHCCU
|
6.5 | IC50 | 2 | — | |
RKDYDLMULRETNX
|
6.5 | Ki | 8 | — | |
VNGYQBMDQMDALH
|
6.5 | Ki | 25 | — | |
VWTSLPZPHHTWSU
|
6.5 | Ki | 5 | — | |
XIDJQQGLLNEFTP
|
6.5 | IC50 | 2 | — | |
YFAZVYJDWIMMBA
|
6.5 | IC50 | 3 | — |