Target Details
| UniProt AC | P49841 |
|---|---|
| Gene Symbol | GSK3B |
| Protein Name | Glycogen synthase kinase-3 beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,206
- Clinical molecules 168
- Avg pChEMBL 7.19
KEGG Pathways (49)
- Alcoholic liver disease
- Alzheimer disease
- Axon guidance
- B cell receptor signaling pathway
- Basal cell carcinoma
- Breast cancer
- Cadherin signaling
- Cell cycle
- Chemokine signaling pathway
- Colorectal cancer
- Cushing syndrome
- Diabetic cardiomyopathy
- Dopaminergic synapse
- EGFR tyrosine kinase inhibitor resistance
- Endometrial cancer
- ErbB signaling pathway
- Focal adhesion
- Gastric cancer
- Growth hormone synthesis, secretion and action
- Hedgehog signaling pathway
- Hepatitis C
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human cytomegalovirus infection
- Human papillomavirus infection
- IL-17 signaling pathway
- IgSF CAM signaling
- Insulin resistance
- Insulin signaling pathway
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Melanogenesis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- PI3K-Akt signaling pathway
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Prion disease
- Prolactin signaling pathway
- Prostate cancer
- Shigellosis
- Signaling pathways regulating pluripotency of stem cells
- T cell receptor signaling pathway
- Thyroid hormone signaling pathway
- Wnt signaling pathway
- Yersinia infection
- mTOR signaling pathway
Active Molecules (2,206)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QNUBZASKWDMCAQ
|
8.8 | IC50 | 2 | — | |
ZLWLGUFTYZQJRI
|
8.8 | IC50 | 3 | — | |
NCCWVYNXHZNCBA
|
8.8 | Ki | 3 | — | |
ZBLGVBFQWBVFAW
|
8.8 | IC50 | 2 | — | |
GKMDVMDXNKYJRV
|
8.8 | IC50 | 2 | — | |
LWBQXWADRRVTID
|
8.8 | IC50 | 2 | — | |
YCVNCXIPRCVVBB
|
8.8 | IC50 | 2 | — | |
VNESSNYPFIJTKU
|
8.8 | Ki | 3 | — | |
HHSIUHRARDLCPM
|
8.8 | IC50 | 5 | Yes | |
UGOONUOQGNIMGO
|
8.8 | IC50 | 2 | — | |
AASZBVWGEDIXLX
|
8.7 | IC50 | 2 | — | |
UHOXKVIMEROOGG
|
8.7 | Ki | 3 | — | |
BXQCCJUQGHRPJT
|
8.7 | IC50 | 2 | — | |
JWHJRYPMAPELPT
|
8.7 | IC50 | 2 | — | |
UHOXKVIMEROOGG
|
8.7 | Ki | 3 | — | |
VPGLALPDHBCDQS
|
8.7 | IC50 | 3 | — | |
WPOGTDAGBXNDTP
|
8.7 | Ki | 3 | — | |
CEUMAXLRGBKFQP
|
8.7 | IC50 | 2 | — | |
DENIPLMYQYHPPA
|
8.7 | IC50 | 6 | Yes | |
FGECJLIFPRCLCB
|
8.7 | Ki | 3 | Yes | |
FZHZYQRQDGJIBK
|
8.7 | Ki | 3 | Yes | |
GBYZMXCPDFNNOB
|
8.7 | Ki | 3 | Yes | |
HJYHJYGXRBYDIG
|
8.7 | Ki | 23 | — | |
IFUKBECSYNPLCY
|
8.7 | IC50 | 3 | — | |
OMGQIHJJEYTELG
|
8.7 | Ki | 4 | — | |
QGMKFIGNGWVOSE
|
8.7 | Ki | 3 | Yes | |
RGVVHQNJKUNSFQ
|
8.7 | IC50 | 2 | — | |
USLKSBWEDVVGFB
|
8.7 | IC50 | 2 | — | |
MHFIPGPJGIQNLQ
|
8.7 | Ki | 3 | — | |
XEFFULWZVBHILM
|
8.7 | IC50 | 2 | — | |
XYTBUOHYMLZOLR
|
8.7 | IC50 | 2 | — | |
YRRRHSNOXWKVDL
|
8.7 | IC50 | 5 | — | |
DVUFESKYOOBJLS
|
8.7 | IC50 | 2 | — | |
HVEXJKQESNIDLM
|
8.7 | Kd | 10 | — | |
KRULSUCANQUTLR
|
8.7 | IC50 | 2 | — | |
MHFIPGPJGIQNLQ
|
8.7 | Ki | 3 | — | |
RAWLWEKCRGSVHW
|
8.6 | Ki | 3 | — | |
XUEHEOHRTKKVET
|
8.6 | IC50 | 2 | Yes | |
ZOEPKGAWYBURFM
|
8.6 | IC50 | 2 | — | |
YUSPBPSJWMPFNQ
|
8.6 | Ki | 3 | — | |
FATYPJCFRSJVOR
|
8.6 | Ki | 3 | — | |
SGSNNFOYHPQJRM
|
8.6 | Ki | 3 | — | |
AMHWMCSHBYIXCE
|
8.6 | IC50 | 3 | — | |
AMOBEFCWUAKOSI
|
8.6 | IC50 | 2 | — | |
DZUXTQCYZWQAFQ
|
8.6 | IC50 | 2 | — | |
FAACVFRHPMNIQT
|
8.6 | IC50 | 2 | — | |
GVOOEMLKTIRYCO
|
8.6 | Ki | 7 | — | |
JAZBHABYAFZEPR
|
8.6 | IC50 | 2 | — | |
NWMPVMMGSHXANZ
|
8.6 | Ki | 58 | — | |
RVSKJUNTDGBSSS
|
8.6 | Ki | 25 | — |