Target Details
| UniProt AC | P49841 |
|---|---|
| Gene Symbol | GSK3B |
| Protein Name | Glycogen synthase kinase-3 beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,206
- Clinical molecules 168
- Avg pChEMBL 7.19
KEGG Pathways (49)
- Alcoholic liver disease
- Alzheimer disease
- Axon guidance
- B cell receptor signaling pathway
- Basal cell carcinoma
- Breast cancer
- Cadherin signaling
- Cell cycle
- Chemokine signaling pathway
- Colorectal cancer
- Cushing syndrome
- Diabetic cardiomyopathy
- Dopaminergic synapse
- EGFR tyrosine kinase inhibitor resistance
- Endometrial cancer
- ErbB signaling pathway
- Focal adhesion
- Gastric cancer
- Growth hormone synthesis, secretion and action
- Hedgehog signaling pathway
- Hepatitis C
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human cytomegalovirus infection
- Human papillomavirus infection
- IL-17 signaling pathway
- IgSF CAM signaling
- Insulin resistance
- Insulin signaling pathway
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Melanogenesis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- PI3K-Akt signaling pathway
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Prion disease
- Prolactin signaling pathway
- Prostate cancer
- Shigellosis
- Signaling pathways regulating pluripotency of stem cells
- T cell receptor signaling pathway
- Thyroid hormone signaling pathway
- Wnt signaling pathway
- Yersinia infection
- mTOR signaling pathway
Active Molecules (2,206)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DZIPQNPWTUXXSJ
|
7.0 | Ki | 18 | — | |
FDBPGAHVEGEARY
|
7.0 | Ki | 19 | — | |
FIQAVSYFYGVUJT
|
7.0 | IC50 | 2 | — | |
IABDKYMGRMDGMM
|
7.0 | Ki | 10 | — | |
IFQICUARAXVEIQ
|
7.0 | Ki | 18 | — | |
IJNGXROUMFEKDB
|
7.0 | Ki | 39 | — | |
KBDRSPRFXNCQAM
|
7.0 | Ki | 8 | — | |
KIETZCMQSGWUQA
|
7.0 | Ki | 2 | — | |
LKUJDAHYLPICSE
|
7.0 | Ki | 24 | — | |
LPILBMJJRGTKOQ
|
7.0 | Ki | 27 | — | |
NBQJSDZRPFLUGK
|
7.0 | IC50 | 2 | — | |
NERQMDXDVAZVNX
|
7.0 | Ki | 13 | — | |
NQPMSSAUJYNSOR
|
7.0 | Ki | 3 | — | |
ORASXEURMWARRB
|
7.0 | IC50 | 2 | — | |
ORUUEFDGYYTXAF
|
7.0 | Ki | 26 | — | |
OXFMTURCMJXJOI
|
7.0 | IC50 | 6 | — | |
OYEBWUJVTCQTJD
|
7.0 | IC50 | 2 | — | |
PFAAZWLEKZPBLT
|
7.0 | IC50 | 2 | — | |
PTZQSGFNHIVQKV
|
7.0 | Ki | 8 | — | |
RXVOXSGTUROJOL
|
7.0 | Ki | 11 | — | |
SMRWVXLSRJWVBF
|
7.0 | Ki | 25 | — | |
VGMDAWVZNAXVDG
|
7.0 | IC50 | 5 | Yes | |
VIZWJTHWUUQVGO
|
7.0 | Ki | 9 | — | |
VTQQYBGURNVVFE
|
7.0 | Ki | 17 | — | |
XZBJACSADMRYGX
|
7.0 | IC50 | 3 | — | |
YEHCNYAQEBQCCS
|
7.0 | Ki | 74 | — | |
ZCXXFPLQFFRMPN
|
7.0 | Ki | 12 | — | |
ZGGIYFOLDBTZIL
|
7.0 | Ki | 27 | — | |
BREKJDOOMHOYCU
|
7.0 | Ki | 3 | — | |
ISFRHUBPXUQPEV
|
7.0 | IC50 | 2 | — | |
NDIUYMHNCUTVGE
|
7.0 | Ki | 25 | — | |
SJWUVVGOTOMGOH
|
7.0 | IC50 | 10 | — | |
VPJUYPLDQXBZDY
|
7.0 | IC50 | 2 | — | |
VVVCUWUORGMTNG
|
7.0 | IC50 | 3 | — | |
YAEMHJKFIIIULI
|
7.0 | IC50 | 2 | — | |
ZOVCAZRXVNBAFS
|
7.0 | IC50 | 2 | — | |
JXJHPQHLHQTQQI
|
7.0 | IC50 | 15 | — | |
UQWUWIJSRXLIKA
|
7.0 | Ki | 3 | — | |
ACBZAFIQJQQSBY
|
7.0 | IC50 | 2 | — | |
CNPLEVGVGWVFGT
|
7.0 | IC50 | 2 | — | |
FHLBVJLTLSPLLV
|
7.0 | Ki | 3 | — | |
IBRKDXNYRBZUGZ
|
7.0 | IC50 | 2 | — | |
IDSINMBICXAPEL
|
7.0 | IC50 | 4 | — | |
PYFNOGGEKLQDLR
|
7.0 | IC50 | 2 | — | |
UKLODWPLBDVRPZ
|
7.0 | Ki | 4 | Yes | |
VRQZQKQMJJRPDA
|
7.0 | Ki | 2 | — | |
XBFRRCZSSOFGAI
|
7.0 | IC50 | 3 | — | |
ZTDVAFBPHUYMFS
|
7.0 | IC50 | 2 | — | |
ZWXBEUSAAVHLFW
|
7.0 | IC50 | 8 | — | |
FMNWOBLAZAYOSG
|
7.0 | IC50 | 5 | — |