Target Details
| UniProt AC | P49841 |
|---|---|
| Gene Symbol | GSK3B |
| Protein Name | Glycogen synthase kinase-3 beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,206
- Clinical molecules 168
- Avg pChEMBL 7.19
KEGG Pathways (49)
- Alcoholic liver disease
- Alzheimer disease
- Axon guidance
- B cell receptor signaling pathway
- Basal cell carcinoma
- Breast cancer
- Cadherin signaling
- Cell cycle
- Chemokine signaling pathway
- Colorectal cancer
- Cushing syndrome
- Diabetic cardiomyopathy
- Dopaminergic synapse
- EGFR tyrosine kinase inhibitor resistance
- Endometrial cancer
- ErbB signaling pathway
- Focal adhesion
- Gastric cancer
- Growth hormone synthesis, secretion and action
- Hedgehog signaling pathway
- Hepatitis C
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human cytomegalovirus infection
- Human papillomavirus infection
- IL-17 signaling pathway
- IgSF CAM signaling
- Insulin resistance
- Insulin signaling pathway
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Melanogenesis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- PI3K-Akt signaling pathway
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Prion disease
- Prolactin signaling pathway
- Prostate cancer
- Shigellosis
- Signaling pathways regulating pluripotency of stem cells
- T cell receptor signaling pathway
- Thyroid hormone signaling pathway
- Wnt signaling pathway
- Yersinia infection
- mTOR signaling pathway
Active Molecules (2,206)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JHYRYOLAZNJFHQ
|
7.5 | Ki | 3 | — | |
JVFWYKRGQNXXST
|
7.5 | Ki | 3 | — | |
NPERTJUHSMWYIC
|
7.5 | IC50 | 3 | — | |
QPMDWYQRFWPAGE
|
7.5 | Ki | 3 | — | |
XBNWVHKGHBNRAG
|
7.5 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.5 | IC50 | 49 | Yes | |
ILJWGWQUBUXSLL
|
7.5 | IC50 | 3 | Yes | |
PFSOTOJNKFKFFB
|
7.5 | IC50 | 2 | — | |
RVUVJNIFPUHUFO
|
7.5 | Ki | 3 | — | |
XOCIRJMUBXHWBK
|
7.5 | IC50 | 2 | — | |
DABSZJYLBZJWOR
|
7.5 | Ki | 3 | — | |
CRZIGHVWJFDSFR
|
7.4 | IC50 | 5 | — | |
LDTNZBKHOOMMNR
|
7.4 | IC50 | 2 | — | |
MWLIVGPGMKTLNU
|
7.4 | Ki | 3 | — | |
RHNUSTPOMUKRCM
|
7.4 | IC50 | 2 | — | |
UEZWIGHGLPNICR
|
7.4 | IC50 | 2 | — | |
BNMDYIGEWXWOOI
|
7.4 | IC50 | 2 | — | |
FSDWOHNRBITTOF
|
7.4 | IC50 | 2 | — | |
OUSFTKFNBAZUKL
|
7.4 | Kd | 58 | Yes | |
PZSHIDRCFNBVAW
|
7.4 | IC50 | 2 | — | |
KVWDUCSNDVVLDF
|
7.4 | Ki | 3 | — | |
QBXUCZWIDBSQSN
|
7.4 | Ki | 3 | — | |
BCRZOEXVCGVQDX
|
7.4 | Ki | 3 | — | |
FPBXMXPANNHQSO
|
7.4 | IC50 | 2 | — | |
GVMDVMPNOAVKJR
|
7.4 | Ki | 26 | Yes | |
NFLNGTZCZDPIPL
|
7.4 | IC50 | 3 | — | |
RJTQBPCQZQSZFF
|
7.4 | Kd | 9 | — | |
RXQXACYMRVINQU
|
7.4 | IC50 | 5 | — | |
SRMKBWXYOWWDPG
|
7.4 | IC50 | 2 | — | |
UEZNNTQSOQVLAB
|
7.4 | Ki | 3 | — | |
AVLYNJZZQYEFEA
|
7.4 | IC50 | 8 | Yes | |
BAXKVZCDBQQQNR
|
7.4 | Ki | 3 | — | |
BOVQIKHARODWQD
|
7.4 | Ki | 4 | — | |
DQYDZCRLDYVZKY
|
7.4 | IC50 | 5 | — | |
FEMBXAAERQHQNM
|
7.4 | Ki | 3 | — | |
FPBCPISREIJULJ
|
7.4 | Ki | 3 | — | |
HZCOFZVJMJRKIB
|
7.4 | IC50 | 2 | — | |
JEYOQYMSSQZLJL
|
7.4 | Ki | 7 | — | |
JJTYLBBKGQOISV
|
7.4 | Ki | 15 | — | |
JOZIXEURKWTTSA
|
7.4 | Ki | 3 | — | |
LOMGAGWJYPGDLT
|
7.4 | Ki | 8 | — | |
LSTWFGPBNKTDIJ
|
7.4 | Ki | 3 | — | |
MOTMISLFANFCFL
|
7.4 | Ki | 3 | — | |
NCNQJLXCZQSYOX
|
7.4 | Ki | 3 | — | |
NHEQNFWGPSKRMJ
|
7.4 | Ki | 7 | — | |
OWXORKPNCHJYOF
|
7.4 | IC50 | 17 | Yes | |
PFCUZXCHLYIMTJ
|
7.4 | Ki | 18 | — | |
RCYPVQCPYKNSTG
|
7.4 | IC50 | 7 | — | |
UXUQVXDYXKMCGA
|
7.4 | Ki | 21 | — | |
UZIATSFXNVOVFE
|
7.4 | IC50 | 2 | — |