Target Details
| UniProt AC | P49841 |
|---|---|
| Gene Symbol | GSK3B |
| Protein Name | Glycogen synthase kinase-3 beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,206
- Clinical molecules 168
- Avg pChEMBL 7.19
KEGG Pathways (49)
- Alcoholic liver disease
- Alzheimer disease
- Axon guidance
- B cell receptor signaling pathway
- Basal cell carcinoma
- Breast cancer
- Cadherin signaling
- Cell cycle
- Chemokine signaling pathway
- Colorectal cancer
- Cushing syndrome
- Diabetic cardiomyopathy
- Dopaminergic synapse
- EGFR tyrosine kinase inhibitor resistance
- Endometrial cancer
- ErbB signaling pathway
- Focal adhesion
- Gastric cancer
- Growth hormone synthesis, secretion and action
- Hedgehog signaling pathway
- Hepatitis C
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human cytomegalovirus infection
- Human papillomavirus infection
- IL-17 signaling pathway
- IgSF CAM signaling
- Insulin resistance
- Insulin signaling pathway
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Melanogenesis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- PI3K-Akt signaling pathway
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Prion disease
- Prolactin signaling pathway
- Prostate cancer
- Shigellosis
- Signaling pathways regulating pluripotency of stem cells
- T cell receptor signaling pathway
- Thyroid hormone signaling pathway
- Wnt signaling pathway
- Yersinia infection
- mTOR signaling pathway
Active Molecules (2,206)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QBWPHVZDFQYVMW
|
7.5 | IC50 | 2 | — | |
QKSJQYPOAQOCOW
|
7.5 | IC50 | 2 | — | |
SRUQTBWIVOVIBO
|
7.5 | Ki | 2 | — | |
XEIWUCRRAQKMAZ
|
7.5 | IC50 | 2 | — | |
BHQZGGSZRHDQFZ
|
7.5 | IC50 | 13 | Yes | |
BLTVBQXJFVRPFK
|
7.5 | Ki | 7 | — | |
NHECRIZPDJYOLQ
|
7.5 | IC50 | 2 | — | |
QTVNFRLKAGKBPS
|
7.5 | IC50 | 3 | — | |
RLESTJQOEHIBLM
|
7.5 | IC50 | 2 | — | |
RYALJKKPLGHHOZ
|
7.5 | Ki | 3 | — | |
SYILOUKHFCRMGK
|
7.5 | Ki | 3 | — | |
YNKUUJYZUJYJRR
|
7.5 | IC50 | 2 | — | |
CHTMRWQLNNRRFJ
|
7.5 | Ki | 70 | — | |
CMKYBUFVJSEEFL
|
7.5 | IC50 | 2 | — | |
DTMZXHDQZQLTHA
|
7.5 | Ki | 21 | — | |
FMUADIGMEFLZAN
|
7.5 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.5 | Ki | 118 | — | |
HWGZXYUOXGVACR
|
7.5 | Ki | 6 | — | |
IUNXLPJUYIYMBV
|
7.5 | Ki | 3 | — | |
JCSGFHVFHSKIJH
|
7.5 | IC50 | 10 | Yes | |
JMHQUQCLIVNTHT
|
7.5 | Ki | 24 | — | |
KYACBMRLQMEIAI
|
7.5 | Ki | 30 | — | |
LSLPDHNUWRDOGC
|
7.5 | Ki | 25 | — | |
NIUJTENHSPPCKO
|
7.5 | Ki | 9 | — | |
RFKYTDGEZKQNDD
|
7.5 | Ki | 3 | — | |
RQJVXILCNCEEPV
|
7.5 | Ki | 3 | — | |
SEYKIIXYLAWBHP
|
7.5 | IC50 | 4 | — | |
SWZAXOLMRPWGRZ
|
7.5 | IC50 | 2 | — | |
URNZTLZSAVLTIZ
|
7.5 | Ki | 26 | — | |
WRZNQKSBJJKEBD
|
7.5 | Ki | 6 | — | |
WVPSKSLAZQPAKQ
|
7.5 | Ki | 3 | — | |
XXSQIQBQZJHGEK
|
7.5 | IC50 | 2 | — | |
XZWVOUQIYLZUCJ
|
7.5 | Ki | 23 | — | |
BWOOIRDDVHVHNJ
|
7.5 | Ki | 2 | — | |
DKVBUSZSQFOSNU
|
7.5 | IC50 | 2 | — | |
HZKLZVWREXHXHF
|
7.5 | Ki | 3 | — | |
JXIPZFBMCRACOW
|
7.5 | Ki | 3 | — | |
ORBLRLVBONJPJG
|
7.5 | Ki | 3 | — | |
UXJMTJZHNOTAAP
|
7.5 | Ki | 3 | — | |
AYTVCTXUVCOWNN
|
7.5 | Ki | 3 | — | |
GEPLEVYEUCTLJX
|
7.5 | Ki | 3 | Yes | |
IBWNGAFCNXNEDG
|
7.5 | Ki | 4 | Yes | |
JFXBJZCDBBMRSA
|
7.5 | Ki | 3 | — | |
NOZZORCJVZKEHP
|
7.5 | IC50 | 2 | — | |
OYVBBBNYTNSCKF
|
7.5 | IC50 | 2 | — | |
SHBOZSJPVRMXBA
|
7.5 | IC50 | 7 | — | |
UXKZMYMPEYJJKA
|
7.5 | IC50 | 5 | — | |
COCQEPVUHJXQEY
|
7.5 | Ki | 3 | — | |
FIKVDYWIFLBJSG
|
7.5 | IC50 | 3 | — | |
GEATXDJAPAHPTP
|
7.5 | IC50 | 10 | — |