Target Details
| UniProt AC | P49841 |
|---|---|
| Gene Symbol | GSK3B |
| Protein Name | Glycogen synthase kinase-3 beta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,206
- Clinical molecules 168
- Avg pChEMBL 7.19
KEGG Pathways (49)
- Alcoholic liver disease
- Alzheimer disease
- Axon guidance
- B cell receptor signaling pathway
- Basal cell carcinoma
- Breast cancer
- Cadherin signaling
- Cell cycle
- Chemokine signaling pathway
- Colorectal cancer
- Cushing syndrome
- Diabetic cardiomyopathy
- Dopaminergic synapse
- EGFR tyrosine kinase inhibitor resistance
- Endometrial cancer
- ErbB signaling pathway
- Focal adhesion
- Gastric cancer
- Growth hormone synthesis, secretion and action
- Hedgehog signaling pathway
- Hepatitis C
- Hepatocellular carcinoma
- Hippo signaling pathway
- Human cytomegalovirus infection
- Human papillomavirus infection
- IL-17 signaling pathway
- IgSF CAM signaling
- Insulin resistance
- Insulin signaling pathway
- Integrin signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Measles
- Melanogenesis
- Neurotrophin signaling pathway
- Non-alcoholic fatty liver disease
- PI3K-Akt signaling pathway
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Prion disease
- Prolactin signaling pathway
- Prostate cancer
- Shigellosis
- Signaling pathways regulating pluripotency of stem cells
- T cell receptor signaling pathway
- Thyroid hormone signaling pathway
- Wnt signaling pathway
- Yersinia infection
- mTOR signaling pathway
Active Molecules (2,206)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AGYZUONRISUOIK
|
7.7 | Ki | 10 | — | |
AOBLBPWPSKBHSI
|
7.7 | Ki | 55 | — | |
BJOKWHXHNKPJQG
|
7.7 | IC50 | 2 | — | |
DYTKVFHLKPDNRW
|
7.7 | Ki | 23 | Yes | |
FXGHOAZJQNLNFD
|
7.7 | IC50 | 13 | Yes | |
HKECWLZKPZHUND
|
7.7 | IC50 | 8 | — | |
HULMMZPBCUBDJN
|
7.7 | Ki | 4 | — | |
IBTJHABKSWXSHB
|
7.7 | IC50 | 2 | — | |
JWQOJVOKBAAAAR
|
7.7 | Ki | 29 | — | |
NUTHTHBJRHLFCA
|
7.7 | IC50 | 2 | — | |
OTVFVCDVXUJJLL
|
7.7 | IC50 | 2 | — | |
PJUVRETYCLPAFV
|
7.7 | Ki | 20 | — | |
PNKAKGKYAQLZIY
|
7.7 | IC50 | 4 | — | |
POXGYBNJJBFCDU
|
7.7 | IC50 | 2 | — | |
QCLXNOBXQUWUEW
|
7.7 | IC50 | 9 | — | |
QOJSERWVVHZZPL
|
7.7 | IC50 | 3 | — | |
QOWGEVKZOPOWLW
|
7.7 | IC50 | 2 | — | |
QTMWRIBZHAYRNM
|
7.7 | IC50 | 2 | — | |
QTSSRGDJHWGQHI
|
7.7 | IC50 | 2 | — | |
RAUNAZYXRMQIJT
|
7.7 | IC50 | 2 | — | |
SRONQUHCRFZABC
|
7.7 | Ki | 28 | — | |
UKNGIFKYRYBARW
|
7.7 | IC50 | 3 | Yes | |
UOVCGJXDGOGOCZ
|
7.7 | Ki | 59 | — | |
VREFOIXLIFZAFY
|
7.7 | Ki | 3 | — | |
VRQYMKLREADGJR
|
7.7 | IC50 | 2 | — | |
VXYDJXMHISGSDA
|
7.7 | Ki | 59 | — | |
WUTXOFQDICTONV
|
7.7 | IC50 | 3 | — | |
XOXWOPNBJDVSJP
|
7.7 | Ki | 8 | — | |
XVHXYPREJYNIQE
|
7.7 | IC50 | 2 | — | |
ZJCKMANGHDJUQT
|
7.7 | IC50 | 3 | Yes | |
ZYERPFJFBXNWOJ
|
7.7 | IC50 | 2 | — | |
GSIAWDOQQULRPR
|
7.7 | Ki | 3 | — | |
RADBQWRTGKIKOV
|
7.7 | Ki | 3 | — | |
YRWLBOFEJRBMIO
|
7.7 | Ki | 3 | — | |
AWNNDHTUHGTAEJ
|
7.7 | IC50 | 2 | — | |
BKYUHKIVVKNZII
|
7.7 | Ki | 3 | — | |
CLNWLUWTLQVFCS
|
7.7 | IC50 | 3 | — | |
IHALLZCDYKCFIO
|
7.7 | Ki | 3 | — | |
OVTRGRMOTBJXKF
|
7.7 | IC50 | 2 | — | |
OYPIIVNTYVSCNV
|
7.7 | IC50 | 4 | — | |
VKZHSGOJYOUKNB
|
7.7 | Ki | 3 | — | |
XJVFAQKZAPQAPZ
|
7.7 | Ki | 3 | — | |
DQFJMOXVVXFSQS
|
7.7 | Ki | 3 | — | |
JEYZBDMGNTZMIQ
|
7.7 | Ki | 3 | — | |
JIUJHJMJUBLVSE
|
7.7 | Ki | 3 | — | |
KCAILKRQNNMUFI
|
7.7 | Ki | 3 | — | |
WGNHFGLWDANFBX
|
7.7 | IC50 | 4 | — | |
AYPKOBSJMAUBFQ
|
7.7 | IC50 | 2 | — | |
BRQIEVOYMRUXNP
|
7.7 | IC50 | 7 | — | |
FQCPPVRJPILDIK
|
7.7 | IC50 | 12 | — |