Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MJZQCHSSWCBKHZ
|
7.4 | IC50 | 2 | — | |
ACWKGTGIJRCOOM
|
7.3 | IC50 | 11 | — | |
ACWKGTGIJRCOOM
|
7.3 | IC50 | 5 | — | |
AVUUHIYJPTWYNX
|
7.3 | IC50 | 9 | — | |
FBVOMJUDISSGGD
|
7.3 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
7.3 | Kd | 1075 | — | |
MYBZDSDFVPDTCR
|
7.3 | IC50 | 2 | — | |
WPLPQAPDKVSKJQ
|
7.3 | IC50 | 2 | — | |
FWRXPBSHAIFMGA
|
7.3 | IC50 | 2 | — | |
JPWPFXUIMVYLLR
|
7.3 | IC50 | 3 | — | |
ZTDVAFBPHUYMFS
|
7.3 | IC50 | 2 | — | |
BHGSKYNWCFIOHP
|
7.3 | Ki | 6 | — | |
CFIBXVQLBVNOHW
|
7.3 | Ki | 64 | — | |
DZCWNAMURCVSNJ
|
7.3 | Ki | 4 | — | |
IJMSMJUUYYSKBT
|
7.3 | IC50 | 2 | — | |
IJNGXROUMFEKDB
|
7.3 | Ki | 39 | — | |
NFKMFNBKEOQNPZ
|
7.3 | Ki | 43 | — | |
NJPWCTYVEJIQBM
|
7.3 | Ki | 72 | — | |
QLWUDWMYFSWGHK
|
7.3 | Ki | 22 | — | |
RRYFECCPZIZXEK
|
7.3 | IC50 | 2 | — | |
RUTNUZIYAWTMEA
|
7.3 | IC50 | 3 | — | |
ULVWJFBHQIXEPE
|
7.3 | Ki | 10 | — | |
UOVCGJXDGOGOCZ
|
7.3 | Ki | 59 | — | |
URNZTLZSAVLTIZ
|
7.3 | Ki | 26 | — | |
VTQQYBGURNVVFE
|
7.3 | Ki | 17 | — | |
WRZNQKSBJJKEBD
|
7.3 | Ki | 6 | — | |
YOVNFNXUCOWYSG
|
7.3 | Ki | 33 | Yes | |
FRXDRZHYTZXJJS
|
7.3 | IC50 | 2 | — | |
PMMSNAUVALVAPD
|
7.3 | IC50 | 2 | — | |
WDPWBLOFHHDUCY
|
7.3 | IC50 | 4 | — | |
XWBBKDHLSOTTLR
|
7.3 | IC50 | 2 | — | |
YAEMHJKFIIIULI
|
7.3 | IC50 | 2 | — | |
FQJGLFZIJDNUCH
|
7.3 | IC50 | 2 | — | |
IYVZGXAXYHRGQR
|
7.3 | IC50 | 2 | — | |
RQUYLFVCZMFFCI
|
7.3 | IC50 | 4 | — | |
BDRSCIWOUKYOAH
|
7.3 | IC50 | 2 | — | |
NRQCVZPNBUOBQY
|
7.3 | IC50 | 2 | — | |
WJRRGYBTGDJBFX
|
7.3 | Kd | 16 | Yes | |
XMPHNZMDLSUDQI
|
7.3 | IC50 | 2 | — | |
QQLBWGXVBLHMJR
|
7.2 | IC50 | 2 | — | |
WHASIRNOCBFBSL
|
7.2 | IC50 | 2 | — | |
SWAZORFPVNPJJA
|
7.2 | IC50 | 2 | — | |
DFYXXJJSVFEUQI
|
7.2 | Ki | 8 | — | |
GMHOTJPHDRSKTA
|
7.2 | IC50 | 4 | — | |
UJTKQLPXTHLCPC
|
7.2 | IC50 | 2 | — | |
CAKMXCJFQDYCIQ
|
7.2 | IC50 | 3 | — | |
URFXBQPKXUWFFL
|
7.2 | IC50 | 2 | — | |
BOVQIKHARODWQD
|
7.2 | Ki | 4 | — | |
CALAEFSQWBJMDU
|
7.2 | Ki | 21 | — | |
DKXHSOUZPMHNIZ
|
7.2 | Ki | 51 | Yes |