Target Details
| UniProt AC | P49840 |
|---|---|
| Gene Symbol | GSK3A |
| Protein Name | Glycogen synthase kinase-3 alpha |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 1,262
- Clinical molecules 47
- Avg pChEMBL 7.05
KEGG Pathways (4)
Active Molecules (1,262)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HUXYBQXJVXOMKX
|
7.5 | Kd | 28 | — | |
OVYJVQMDQIHIRD
|
7.5 | IC50 | 2 | — | |
PAIFVBSOFXHAPE
|
7.5 | IC50 | 2 | — | |
POLVSVXQURZBBJ
|
7.5 | IC50 | 2 | — | |
TUOUHOOTMXWCSA
|
7.5 | IC50 | 2 | — | |
XEIWUCRRAQKMAZ
|
7.5 | IC50 | 2 | — | |
YHNDGIRYUITNSU
|
7.5 | IC50 | 2 | — | |
ZHZPUYSNZQKXRF
|
7.5 | IC50 | 2 | — | |
BHQZGGSZRHDQFZ
|
7.5 | IC50 | 13 | Yes | |
NHECRIZPDJYOLQ
|
7.5 | IC50 | 2 | — | |
AOBLBPWPSKBHSI
|
7.5 | Ki | 55 | — | |
FMUADIGMEFLZAN
|
7.5 | IC50 | 2 | — | |
OEKYVFZKBRIDJO
|
7.5 | Ki | 12 | — | |
OUJZYQBEFNDJQN
|
7.5 | Ki | 71 | — | |
QAJPIJHWTGPUNZ
|
7.5 | Ki | 37 | — | |
SRUYEOQJIXGTDT
|
7.5 | IC50 | 3 | — | |
VXYDJXMHISGSDA
|
7.5 | Ki | 59 | — | |
XXSQIQBQZJHGEK
|
7.5 | IC50 | 2 | — | |
FQNITDDDUQQKBZ
|
7.5 | IC50 | 2 | — | |
JZCWLJDSIRUGIN
|
7.5 | Ki | 16 | — | |
SMIWRILWBDJESB
|
7.5 | IC50 | 2 | — | |
BNMDYIGEWXWOOI
|
7.5 | IC50 | 2 | — | |
JCSGFHVFHSKIJH
|
7.5 | IC50 | 10 | Yes | |
NSERNZRHLGJSNF
|
7.5 | IC50 | 2 | — | |
XBNWVHKGHBNRAG
|
7.5 | IC50 | 2 | — | |
IUEJEHPLFBVXJH
|
7.5 | IC50 | 2 | — | |
XOCIRJMUBXHWBK
|
7.5 | IC50 | 2 | — | |
RHNUSTPOMUKRCM
|
7.4 | IC50 | 2 | — | |
ASLGQVPNOSGBQR
|
7.4 | IC50 | 10 | — | |
VPJUYPLDQXBZDY
|
7.4 | IC50 | 2 | — | |
KYFJPYWXCUCRPE
|
7.4 | IC50 | 2 | — | |
NFLNGTZCZDPIPL
|
7.4 | IC50 | 3 | — | |
JOZIXEURKWTTSA
|
7.4 | Ki | 3 | — | |
JWQOJVOKBAAAAR
|
7.4 | Ki | 29 | — | |
LNIDFQVRZCDVBI
|
7.4 | Ki | 16 | — | |
OIDZQWOKVFYZSD
|
7.4 | Ki | 8 | — | |
PJUVRETYCLPAFV
|
7.4 | Ki | 20 | — | |
QCLXNOBXQUWUEW
|
7.4 | IC50 | 9 | — | |
UPPGGRZNGRFDAU
|
7.4 | Ki | 21 | — | |
VJKJKZOWXJKSSK
|
7.4 | Ki | 4 | — | |
WAKGEHXTOOFEAE
|
7.4 | Ki | 27 | — | |
YNUMBZPWLHDVEX
|
7.4 | Ki | 6 | — | |
WSEQQMOTVBENFI
|
7.4 | IC50 | 2 | — | |
KRLXYVKWKDSKSA
|
7.4 | IC50 | 2 | — | |
LYADGAGFYYXXIO
|
7.4 | IC50 | 82 | — | |
QEHNJBXQNRKLAX
|
7.4 | IC50 | 2 | — | |
SJVVUBXEQRYTIE
|
7.4 | IC50 | 2 | — | |
SSBXQQAGHPLUTI
|
7.4 | IC50 | 2 | — | |
BVNDJEHETZIZCV
|
7.4 | Ki | 5 | — | |
CZPAIZKCGQCIOF
|
7.4 | IC50 | 2 | — |